-
1
-
-
34447646495
-
Developing early formulations: Practice and perspective
-
L. Ping, and L. Zhao Developing early formulations: practice and perspective Int. J. Pharm. 341 2007 1 19
-
(2007)
Int. J. Pharm.
, vol.341
, pp. 1-19
-
-
Ping, L.1
Zhao, L.2
-
2
-
-
84859734219
-
Modification of physicochemical characteristics of active pharmaceutical ingredients and application of supersaturatable dosage forms for improving bioavailability of poorly absorbed drugs
-
K. Kawakami Modification of physicochemical characteristics of active pharmaceutical ingredients and application of supersaturatable dosage forms for improving bioavailability of poorly absorbed drugs Adv. Drug Deliv. Rev. 64 2012 480 495
-
(2012)
Adv. Drug Deliv. Rev.
, vol.64
, pp. 480-495
-
-
Kawakami, K.1
-
3
-
-
0031024171
-
Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
-
C.A. Lipinski, F. Lombardo, B.W. Dominy, and P.J. Feeney Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings Adv. Drug. Deliv. Rev. 23 1997 3 25
-
(1997)
Adv. Drug. Deliv. Rev.
, vol.23
, pp. 3-25
-
-
Lipinski, C.A.1
Lombardo, F.2
Dominy, B.W.3
Feeney, P.J.4
-
4
-
-
84860658314
-
Bridging solubility between drug discovery and development
-
L. Di, P.V. Fish, and T. Mano Bridging solubility between drug discovery and development Drug Discov. Today 17 2012 486 495
-
(2012)
Drug Discov. Today
, vol.17
, pp. 486-495
-
-
Di, L.1
Fish, P.V.2
Mano, T.3
-
5
-
-
68249128120
-
Supersaturating drug delivery systems: The answer to solubility-limited oral bioavailability?
-
J. Brouwers, M.E. Brewrter, and P. Augustijns Supersaturating drug delivery systems: the answer to solubility-limited oral bioavailability? J. Pharm. Sci. 98 2009 2549 2572
-
(2009)
J. Pharm. Sci.
, vol.98
, pp. 2549-2572
-
-
Brouwers, J.1
Brewrter, M.E.2
Augustijns, P.3
-
6
-
-
34548040152
-
High throughput solubility measurement in drug discovery and development
-
J. Alsenz, and M. Kansy High throughput solubility measurement in drug discovery and development Adv. Drug. Deliv. Rev. 59 2007 546 567
-
(2007)
Adv. Drug. Deliv. Rev.
, vol.59
, pp. 546-567
-
-
Alsenz, J.1
Kansy, M.2
-
7
-
-
12244263506
-
Comparison of a miniaturized shake-flask solubility method with automated potentiometric acid/base titrations and calculated solubilities
-
A. Glomme, J. März, and J.B. Dressman Comparison of a miniaturized shake-flask solubility method with automated potentiometric acid/base titrations and calculated solubilities J. Pharm. Sci. 94 2005 1 16
-
(2005)
J. Pharm. Sci.
, vol.94
, pp. 1-16
-
-
Glomme, A.1
März, J.2
Dressman, J.B.3
-
8
-
-
33750000906
-
-
K. Sugano, T. Kato, K. Suzuki, K. Keiko, T. Sujaku, and T. Mano J. Pharm. Sci. 95 2006 2115 2122
-
(2006)
J. Pharm. Sci.
, vol.95
, pp. 2115-2122
-
-
Sugano, K.1
Kato, T.2
Suzuki, K.3
Keiko, K.4
Sujaku, T.5
Mano, T.6
-
9
-
-
84884142861
-
Aqueous solubility: Simple predictive methods (in silico, in vitro and bio-relevantapproaches)
-
D. Eldera, and R. Holm Aqueous solubility: simple predictive methods (in silico, in vitro and bio-relevantapproaches) Int. J. Pharm. 453 2013 3 11
-
(2013)
Int. J. Pharm.
, vol.453
, pp. 3-11
-
-
Eldera, D.1
Holm, R.2
-
10
-
-
0036238280
-
A comparative study of artificial membrane permeability assay for high throughput profiling of drug absorption potential
-
C. Zhu, L. Jiang, T. Chen, and K. Hwang A comparative study of artificial membrane permeability assay for high throughput profiling of drug absorption potential Eur. J. Med. Chem. 37 2002 399 407
-
(2002)
Eur. J. Med. Chem.
, vol.37
, pp. 399-407
-
-
Zhu, C.1
Jiang, L.2
Chen, T.3
Hwang, K.4
-
11
-
-
0031024171
-
Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
-
C.A. Lipinski, F. Lombardo, B.W. Dominy, and P.J. Feeney Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings Adv. Drug. Deliv. Rev. 23 1997 3 25
-
(1997)
Adv. Drug. Deliv. Rev.
, vol.23
, pp. 3-25
-
-
Lipinski, C.A.1
Lombardo, F.2
Dominy, B.W.3
Feeney, P.J.4
-
12
-
-
80054697161
-
Formulation design for poorly water-soluble drugs based on biopharmaceutics classification system: Basic approaches and practical applications
-
Y. Kawabata, K. Wada, M. Nakatani, and S.Y.S. Onoue Formulation design for poorly water-soluble drugs based on biopharmaceutics classification system: basic approaches and practical applications Int. J. Pharm. 420 2011 1 10
-
(2011)
Int. J. Pharm.
, vol.420
, pp. 1-10
-
-
Kawabata, Y.1
Wada, K.2
Nakatani, M.3
Onoue, S.Y.S.4
-
13
-
-
2342635206
-
Application of high-performance liquid chromatography based measurements of lipophilicity to model biological distribution
-
K. Valko Application of high-performance liquid chromatography based measurements of lipophilicity to model biological distribution J. Chromatogr. A 1037 2004 299 310
-
(2004)
J. Chromatogr. A
, vol.1037
, pp. 299-310
-
-
Valko, K.1
-
14
-
-
67349086295
-
Analytical tools for the physicochemical profiling of drug candidates to predict absorption/distribution
-
Y. Henchoz, B. Bard, D. Guillarme, P. Carrupt, J. Veuthey, and S. Martel Analytical tools for the physicochemical profiling of drug candidates to predict absorption/distribution Anal. Bioanal. Chem. 394 2009 707 729
-
(2009)
Anal. Bioanal. Chem.
, vol.394
, pp. 707-729
-
-
Henchoz, Y.1
Bard, B.2
Guillarme, D.3
Carrupt, P.4
Veuthey, J.5
Martel, S.6
-
17
-
-
67349254634
-
An interesting relationship between drug absorption and melting point
-
K.A. Chu, and S.H. Yalkowsky An interesting relationship between drug absorption and melting point Int. J. Pharm. 373 2009 24 40
-
(2009)
Int. J. Pharm.
, vol.373
, pp. 24-40
-
-
Chu, K.A.1
Yalkowsky, S.H.2
-
18
-
-
84929174916
-
-
P. Sanphui, D.V. Kusum, D. Clara, N. Malviya, S. Ganguly, and G.R. Desiraju Mol. Pharm. 12 2015 1615 1622
-
(2015)
Mol. Pharm.
, vol.12
, pp. 1615-1622
-
-
Sanphui, P.1
Kusum, D.V.2
Clara, D.3
Malviya, N.4
Ganguly, S.5
Desiraju, G.R.6
-
19
-
-
84889087023
-
Current trends and future perspectives of solid dispersions containing poorly water-soluble drugs
-
L.V. Chau, C. Park, and L.B. Lee Current trends and future perspectives of solid dispersions containing poorly water-soluble drugs Eur. J. Pharm. Biopharm. 85 2013 799 813
-
(2013)
Eur. J. Pharm. Biopharm.
, vol.85
, pp. 799-813
-
-
Chau, L.V.1
Park, C.2
Lee, L.B.3
-
20
-
-
34848888967
-
Solubility and dissolution profile assessment in drug discovery, drug metab
-
K. Sugano, A. Okazaki, S. Sugimoto, S. Tavornvipas, A. Omura, and T. Mano Solubility and dissolution profile assessment in drug discovery, drug metab Pharmacokinet 22 2007 225 254
-
(2007)
Pharmacokinet
, vol.22
, pp. 225-254
-
-
Sugano, K.1
Okazaki, A.2
Sugimoto, S.3
Tavornvipas, S.4
Omura, A.5
Mano, T.6
-
21
-
-
34548032742
-
Salt formation to improve drug solubility
-
Abu T.M. Serajuddin Salt formation to improve drug solubility Adv. Drug Deliv. Rev. 59 2007 603 616
-
(2007)
Adv. Drug Deliv. Rev.
, vol.59
, pp. 603-616
-
-
Serajuddin, A.T.M.1
-
22
-
-
79959906965
-
The BCS, BDDCS, and regulatory guidances
-
Mei-Ling Chen, Gordon L. Amidon, Leslie Z. Benet, Hans Lennernas, and Lawrence X. Yu The BCS, BDDCS, and regulatory guidances Pharm. Res. 28 2011 1774 1778
-
(2011)
Pharm. Res.
, vol.28
, pp. 1774-1778
-
-
Chen, M.-L.1
Amidon, G.L.2
Benet, L.Z.3
Lennernas, H.4
Yu, L.X.5
-
23
-
-
84941889664
-
Development of self-emulsifying lipid formulations of BCS class II drugs with low to medium lipophilicity
-
V. Jannina, S. Chevriera, M. Michenauda, C. Dumonta, S. Belottia, Y. Chavanta, and F. Demarne Development of self-emulsifying lipid formulations of BCS class II drugs with low to medium lipophilicity Int. J. Pharm. 495 2015 385 392
-
(2015)
Int. J. Pharm.
, vol.495
, pp. 385-392
-
-
Jannina, V.1
Chevriera, S.2
Michenauda, M.3
Dumonta, C.4
Belottia, S.5
Chavanta, Y.6
Demarne, F.7
-
24
-
-
40149088986
-
Prodrugs: Design and clinical applications
-
J. Rautio, H. Kumpulainen, T. Heimbach, R. Oliyai, D. Oh, T. Järvinen, and J. Savolainen Prodrugs: design and clinical applications Nat. Rev. Drug Discov. 7 2008 255 270
-
(2008)
Nat. Rev. Drug Discov.
, vol.7
, pp. 255-270
-
-
Rautio, J.1
Kumpulainen, H.2
Heimbach, T.3
Oliyai, R.4
Oh, D.5
Järvinen, T.6
Savolainen, J.7
-
25
-
-
84876055612
-
Permeability enhancement techniques for poorly permeable drugs: A review
-
S.I. Ms, N.C. Derle, and R. Bhamber Permeability enhancement techniques for poorly permeable drugs: a review J. Appl. Pharm. Sci. 2 2012 34 39
-
(2012)
J. Appl. Pharm. Sci.
, vol.2
, pp. 34-39
-
-
Ms, S.I.1
Derle, N.C.2
Bhamber, R.3
|