Comparison of lipid and detergent enzyme environments for identifying inhibitors of membrane-bound energy-transducing proteins

Journal of Microbiological Methods

Volumn 120, Issue , 2016, Pages 41-43

  Dunn, Elyse A ^a   Cook, Gregory M ^a,b   Heikal, Adam ^a,b  

^a UNIVERSITY OF OTAGO   (New Zealand)

^b UNIVERSITY OF AUCKLAND   (New Zealand)

Author keywords

Antibiotic; Drug discovery; High throughput screening (HTS); Proteoliposomes; Type II NADH dehydrogenase (NDH 2)

Indexed keywords

DETERGENT; MEMBRANE PROTEIN; PHOSPHATIDYLCHOLINE; PROTEIN INHIBITOR; PROTEOLIPOSOME; REDUCED NICOTINAMIDE ADENINE DINUCLEOTIDE DEHYDROGENASE; ANTIINFECTIVE AGENT; LIPID; NADH DEHYDROGENASE II; PROTEOLIPID; PROTEOLIPOSOMES;

ARTICLE; COMPARATIVE STUDY; DRUG RESEARCH; DRUG TARGETING; ENERGY TRANSFER; HIGH THROUGHPUT SCREENING; LIPOPHILICITY; POLYACRYLAMIDE GEL ELECTROPHORESIS; PRIORITY JOURNAL; PROTEIN ANALYSIS; ANTAGONISTS AND INHIBITORS; CELL MEMBRANE; CHEMISTRY; DRUG DEVELOPMENT; DRUG EFFECTS; ISOLATION AND PURIFICATION; KINETICS; PRECLINICAL STUDY; PROCEDURES;

ANTI-INFECTIVE AGENTS; CELL MEMBRANE; DETERGENTS; DRUG DISCOVERY; DRUG EVALUATION, PRECLINICAL; ELECTROPHORESIS, POLYACRYLAMIDE GEL; HIGH-THROUGHPUT SCREENING ASSAYS; KINETICS; LIPIDS; MEMBRANE PROTEINS; NADH DEHYDROGENASE; PROTEOLIPIDS;

EID: 84947976325     PISSN: 01677012     EISSN: 18728359     Source Type: Journal    
DOI: 10.1016/j.mimet.2015.11.012     Document Type: Article

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