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Journal of Medicinal Chemistry

Volumn 58, Issue 20, 2015, Pages 7928-7930

Discovery of the First Selective, Nonpeptidic Orexin 2 Receptor Agonists

(3) Heifetz, Alexander a Bodkin, Mike J a Biggin, Philip C b

a EVOTEC UK LTD (United Kingdom)

b UNIVERSITY OF OXFORD (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

AGENTS INTERACTING WITH TRANSMITTER, HORMONE OR DRUG RECEPTORS; OREXIN; OREXIN 2 RECEPTOR; OREXIN 2 RECEPTOR AGONIST; UNCLASSIFIED DRUG; BENZAMIDE DERIVATIVE; OREXIN RECEPTOR; SULFONAMIDE;

AGONIST POTENCY; CRYSTAL STRUCTURE; DRUG CONFORMATION; DRUG EFFICACY; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; HUMAN; MOLECULAR DOCKING; REVIEW; STRUCTURE ACTIVITY RELATION; X RAY CRYSTALLOGRAPHY; AGONISTS; ANIMAL; SYNTHESIS;

ANIMALS; BENZAMIDES; HUMANS; OREXIN RECEPTORS; SULFONAMIDES;

EID: 84945589012 PISSN: 00222623 EISSN: 15204804 Source Type: Journal
DOI: 10.1021/acs.jmedchem.5b01394 Document Type: Review

Times cited : (14)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.