Mucoadhesive cellulosic derivative sponges as drug delivery system for vaginal application

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 95, Issue , 2015, Pages 128-135

  Furst, Tania ^a   Piette, Marie ^a   Lechanteur, Anna ^a   Evrard, Brigitte ^a   Piel, Géraldine ^a  

^a UNIVERSITY OF LIÈGE   (Belgium)

Author keywords

Cellulosic derivative; Hydrogel; Lyophilization; Mucoadhesion; Sponge; Vaginal

Indexed keywords

HYDROXYETHYLCELLULOSE; HYDROXYETHYLCELLULOSE 250 M; MACROGOL 400; MICONAZOLE; UNCLASSIFIED DRUG; CELLULOSE; HYDROGEL; TISSUE ADHESIVE;

ARTICLE; DRUG DELIVERY SYSTEM; FREEZE DRYING; FREEZING; HYDROGEL; IN VITRO STUDY; MUCOADHESION; REHYDRATION; SCANNING ELECTRON MICROSCOPY; SURFACE AREA; TEMPERATURE; VAGINA DISCHARGE; VISCOSITY; WATER LOSS; ADMINISTRATION AND DOSAGE; ANIMAL; CHEMISTRY; FEMALE; HUMAN; INTRAVAGINAL DRUG ADMINISTRATION; METABOLISM; PROCEDURES;

ADMINISTRATION, INTRAVAGINAL; ANIMALS; CELLULOSE; DRUG DELIVERY SYSTEMS; FEMALE; HUMANS; HYDROGELS; TISSUE ADHESIVES;

EID: 84944274678     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2015.01.019     Document Type: Article

References (24)

1. A. Aka-Any-Grah, K. Bouchemal, A. Koffi, F. Agnely, M. Zhang, M. Djabourov, and et al. Formulation of mucoadhesive vaginal hydrogels insensitive to dilution with vaginal fluids Eur. J. Pharm. Biopharm. 76 2 2010 296 303
2. J. das Neves, and M.F. Bahia Gels as vaginal drug delivery systems Int. J. Pharmaceut. 318 1-2 2006 1 14
3. L.M. Ensign, R. Cone, and J. Hanes Nanoparticle-based drug delivery to the vagina: a review J. Control. Release 190 2014 500 514
4. Z. Vanic, and N. Skalko-Basnet Nanopharmaceuticals for improved topical vaginal therapy: can they deliver? Eur. J. Pharm. Sci. 50 1 2013 29 41
5. S. Yang, Y. Chen, R. Ahmadie, and E.A. Ho Advancements in the field of intravaginal siRNA delivery J. Control. Release 167 1 2013 29 39
6. T. Bríd, R.L.S. Burruano, and Daniel Malamud In vitro test to evaluate the interaction between synthetic cervical mucus and vaginal formulations AAPS PharmSciTech. 5 1 2004 (Article 17)
7. J. das Neves, M. Amiji, and B. Sarmento Mucoadhesive nanosystems for vaginal microbicide development: friend or foe? Nanomed. Nanobiotechnol. 3 4 2011 389 399
8. R. Margareth, and C. Marques Simulated biological fluids with possible application in dissolution testing Dissolution Technol. 2011 15 28
9. H.H. Sigurdsson, J. Kirch, and C.M. Lehr Mucus as a barrier to lipophilic drugs Int. J. Pharm. 453 1 2013 56 64
10. K.J. Whaley, J. Hanes, R. Shattock, R.A. Cone, and D.R. Friend Novel approaches to vaginal delivery and safety of microbicides: biopharmaceuticals, nanoparticles, and vaccines Antiviral Res. 88 Suppl. 1 2010 S55 S66
11. K. Berginc, S. Suljakovic, N. Skalko-Basnet, and A. Kristl Mucoadhesive liposomes as new formulation for vaginal delivery of curcumin Eur. J. Pharm. Biopharm. 87 1 2014 40 46
12. J.D. Smart The basics and underlying mechanisms of mucoadhesion Adv. Drug Deliv. Rev. 57 11 2005 1556 1568
13. S. David, A.D.W. Jones, and Andrew F. Brown Textural, viscoelastic and mucoadhesive properties of pharmaceutical gels composed of cellulose polymers Int. J. Pharm. 151 1997 223 233
14. A. Tachaprutinun, P. Pan-In, and S. Wanichwecharungruang Mucosa-plate for direct evaluation of mucoadhesion of drug carriers Int. J. Pharm. 441 1-2 2013 801 808
15. K.H. Matthews, H.N. Stevens, A.D. Auffret, M.J. Humphrey, and G.M. Eccleston Lyophilised wafers as a drug delivery system for wound healing containing methylcellulose as a viscosity modifier Int. J. Pharm. 289 1-2 2005 51 62
16. O. Labovitiadi, A.J. Lamb, and K.H. Matthews Lyophilised wafers as vehicles for the topical release of chlorhexidine digluconate-release kinetics and efficacy against Pseudomonas aeruginosa Int. J. Pharm. 439 1-2 2012 157 164
17. M. Piette, I. Coia, B. Evrard, Composition and Method for treating HPV, Belgium, US2014 017 0219 A1.
18. P.N. Gupta, A. Pattani, R.M. Curran, V.L. Kett, G.P. Andrews, R.J. Morrow, and et al. Development of liposome gel based formulations for intravaginal delivery of the recombinant HIV-1 envelope protein CN54gp140 Eur. J. Pharm. Sci. 46 5 2012 315 322
19. S.F. Ng, and N. Jumaat Carboxymethyl cellulose wafers containing antimicrobials: a modern drug delivery system for wound infections Eur. J. Pharm. Sci. 51 2014 173 179
20. J.S. Boateng, A.D. Auffret, K.H. Matthews, M.J. Humphrey, H.N. Stevens, and G.M. Eccleston Characterisation of freeze-dried wafers and solvent evaporated films as potential drug delivery systems to mucosal surfaces Int. J. Pharm. 389 1-2 2010 24 31
21. E. Josef, and H. Bianco-Peled Sponges carrying self-microemulsifying drug delivery systems Int. J. Pharm. 458 1 2013 208 217
22. C. María, M.L.F. Gutiérrez, and Monte Francisco del Ice-templated materials sophisticated structures exhibiting enhanced functionalities obtained after unidirectional freezing and ice-segregation-induced self-assembly Chem. Mater. 20 2007 634 648
23. J.C. Kasper, and W. Friess The freezing step in lyophilization: physico-chemical fundamentals, freezing methods and consequences on process performance and quality attributes of biopharmaceuticals Eur. J. Pharm. Biopharm. 78 2 2011 248 263
24. J.C. Kasper, G. Winter, and W. Friess Recent advances and further challenges in lyophilization Eur. J. Pharm. Biopharm. 85 2 2013 162 169