메뉴 건너뛰기




Volumn 56, Issue 23, 2015, Pages 3486-3488

Selective synthesis of either enantiomer of an anti-breast cancer agent via a common enantioenriched intermediate

Author keywords

Anti cancer agent; Cross coupling; Nickel; Stereospecific; Triarylmethane

Indexed keywords


EID: 84939556860     PISSN: 00404039     EISSN: 18733581     Source Type: Journal    
DOI: 10.1016/j.tetlet.2015.02.121     Document Type: Article
Times cited : (18)

References (41)
  • 5
    • 84903976004 scopus 로고    scopus 로고
    • For an overview of synthesis and medicinal properties of triarylmethanes, see
    • For an overview of synthesis and medicinal properties of triarylmethanes, see: F.S. Mondal, and G. Panda RSC Adv. 4 2014 28317
    • (2014) RSC Adv , vol.4 , pp. 28317
    • Mondal, F.S.1    Panda, G.2
  • 11
    • 84939977330 scopus 로고    scopus 로고
    • Anti-diabetes: U.S. Pat. Appl
    • Anti-diabetes: Ellsworth, B. A.; Ewing, W. R.; Jurica, E. U.S. Pat. Appl. 2011/0082165 A1, 2011.
    • (2011)
    • Ellsworth, B.A.1    Ewing, W.R.2    Jurica, E.3
  • 16
    • 36849061646 scopus 로고    scopus 로고
    • For more recent advances in transition-metal catalyzed Friedel-Crafts reactions: (a)
    • For more recent advances in transition-metal catalyzed Friedel-Crafts reactions: (a) S. Lin, and X. Lu J. Org. Chem. 72 2007 9757
    • (2007) J. Org. Chem. , vol.72 , pp. 9757
    • Lin, S.1    Lu, X.2
  • 21
    • 33751569703 scopus 로고    scopus 로고
    • For cross-coupling strategies that provide racemic products, see: (a)
    • For cross-coupling strategies that provide racemic products, see: (a) G.A. Molander, and M.D. Elia J. Org. Chem. 71 2006 9198
    • (2006) J. Org. Chem. , vol.71 , pp. 9198
    • Molander, G.A.1    Elia, M.D.2
  • 24
    • 73349133684 scopus 로고    scopus 로고
    • For chiral phosphoric acid catalyzed Friedel-Crafts alkylations, see: (a)
    • For chiral phosphoric acid catalyzed Friedel-Crafts alkylations, see: (a) F.-L. Sun, X.-J. Zheng, Q. Gu, Q.-L. He, and S.-L. You Eur. J. Org. Chem. 2010 47
    • (2010) Eur. J. Org. Chem. , pp. 47
    • Sun, F.-L.1    Zheng, X.-J.2    Gu, Q.3    He, Q.-L.4    You, S.-L.5
  • 27
    • 48849108176 scopus 로고    scopus 로고
    • For pyridine-directed enantioselective palladium-catalyzed C-H bond activation, see
    • For pyridine-directed enantioselective palladium-catalyzed C-H bond activation, see: B.-F. Shi, N. Maugel, Y.-H. Zhang, and J.-Q. Yu Angew. Chem., Int. Ed. 47 2008 4882
    • (2008) Angew. Chem., Int. Ed. , vol.47 , pp. 4882
    • Shi, B.-F.1    Maugel, N.2    Zhang, Y.-H.3    Yu, J.-Q.4
  • 39
    • 70350509058 scopus 로고    scopus 로고
    • es = enantiospecificity = (ee starting material)/(ee product) see
    • es = enantiospecificity = (ee starting material)/(ee product) see, S.E. Denmark, and T. Vogler Chem. Eur. J. 15 2009 11737
    • (2009) Chem. Eur. J. , vol.15 , pp. 11737
    • Denmark, S.E.1    Vogler, T.2
  • 40
    • 84949923857 scopus 로고    scopus 로고
    • 2 and SIMes resulted in 10% yield of triarylmethane 5. See Ref. 15b
    • 2 and SIMes resulted in 10% yield of triarylmethane 5. See Ref. 15b.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.