Carbapenem-resistant Enterobacteriaceae: Epidemiology and Prevention
Gupta, N.; Limbago, B. M.; Patel, J. B.; Kallen, A. J. Carbapenem-resistant Enterobacteriaceae: Epidemiology and Prevention Clin. Infect. Dis. 2011, 53, 60 - 67
Methicillin-Resistant Staphylococcus aureus: A Consensus Review of the Microbiology, Pathogenesis, and Epidemiology with Implications for Prevention and Management
Mulligan, M. E.; Murray-Leisure, K. A.; Ribner, B. S.; Standiford, H. C.; John, J. F.; Korvick, J. A.; Kauffman, C. A.; Yu, Y. L. Methicillin-Resistant Staphylococcus aureus: A Consensus Review of the Microbiology, Pathogenesis, and Epidemiology with Implications for Prevention and Management Am. J. Med. 1993, 94, 313 - 328
Conover, L H. Discovery of Drugs from Microbiological Sources. In Drug Discovery, Science and Development in a Changing Society; American Chemical Society: Washington, DC, 1971; Vol. 108, pp 33 - 80.
Glycylcyclines. 1. A New Generation of Potent Antibacterial Agents through Modification of 9-Aminotetracyclines
Sum, P.-E.; Lee, V. J.; Testa, R. T.; Hlavka, J. J.; Ellestad, G. A.; Bloom, J. D.; Gluzman, Y.; Tally, F. P. Glycylcyclines. 1. A New Generation of Potent Antibacterial Agents through Modification of 9-Aminotetracyclines J. Med. Chem. 1994, 37, 184 - 188
Phase 2, Randomized, Double-blind Study of the Efficacy and Safety of Two Dose Regimens of Eravacycline versus Ertapenem for Adult Community-Acquired Complicated Intra-abdominal Infections
Solomkin, J. S.; Ramesh, M. K.; Cesnauskas, G.; Novikovs, N.; Stefanova, P.; Sutcliffe, J. A.; Walpole, S. M.; Horn, P. T. Phase 2, Randomized, Double-blind Study of the Efficacy and Safety of Two Dose Regimens of Eravacycline versus Ertapenem for Adult Community-Acquired Complicated Intra-abdominal Infections Antimicrob. Agents Chemother. 2014, 58, 1847 - 1854
Synthesis and Antibacterial Activity of Pentacyclines: A Novel Class of Tetracycline Analogs
Sun, C.; Hunt, D. K.; Clark, R. B.; Lofland, D.; O'Brien, W. J.; Plamondon, L.; Xiao, X.-Y. Synthesis and Antibacterial Activity of Pentacyclines: A Novel Class of Tetracycline Analogs J. Med. Chem. 2011, 54, 3704 - 3731
A Robust Platform for the Synthesis of New Tetracycline Antibiotics
Sun, C.; Wang, Q.; Brubaker, J. D.; Wright, P. M.; Lerner, C. D.; Noson, K.; Charest, M.; Siegel, D. R.; Wang, Y.-M.; Myers, A. G. A Robust Platform for the Synthesis of New Tetracycline Antibiotics J. Am. Chem. Soc. 2008, 130, 17913 - 17927
8-Azatetracyclines: Synthesis and Evaluation of a Novel Class of Tetracycline Antibacterial Agents
Clark, R. B.; He, M.; Fyfe, C.; Lofland, D.; O'Brien, W. J.; Plamondon, L.; Xiao, X.-Y. 8-Azatetracyclines: Synthesis and Evaluation of a Novel Class of Tetracycline Antibacterial Agents J. Med. Chem. 2011, 54, 1511 - 1528
Fluorocyclines. 2. Optimization of the C-9 Side-Chain for Antibacterial Activity and Oral Efficacy
Clark, R. B.; Hunt, D. K.; Me, H.; Achorn, C.; Chen, C.-L.; Deng, D.; Fyfe, C.; Grossman, T. H.; Hogan, P. C.; O'Brien, W. J.; Plamondon, L.; Ronn, M.; Sutcliffe, J. A.; Zhu, Z.; Xiao, X.-Y. Fluorocyclines. 2. Optimization of the C-9 Side-Chain for Antibacterial Activity and Oral Efficacy J. Med. Chem. 2012, 55, 606 - 622
Synthesis and Biological Evaluation of 8-Aminomethyltetracycline Derivatives as Novel Antibacterial Agents
Clark, R. B.; He, M.; Deng, D.; Sun, C.; Chen, C.-L.; Hunt, D. K.; O'Brien, W. J.; Fyfe, C.; Grossman, T. H.; Sutcliffe, J. A.; Achorn, C.; Hogan, P. C.; Katz, C. E.; Niu, J.; Zhang, W.-Y.; Zhu, Z.; Ronn, M.; Xiao, X.-Y. Synthesis and Biological Evaluation of 8-Aminomethyltetracycline Derivatives as Novel Antibacterial Agents J. Med. Chem. 2013, 56, 8112 - 8138
A Convergent Enantioselective Route to Structurally Diverse 6-Deoxytetracycline Antibiotics
Charest, M. G.; Lerner, C. D.; Brubaker, J. D.; Siegel, D. R.; Myers, A. G. A Convergent Enantioselective Route to Structurally Diverse 6-Deoxytetracycline Antibiotics Science 2005, 308, 395 - 398
A Practical, Enantioselective Synthetic Route to a Key Precursor to the Tetracycline Antibiotics
Brubaker, J. D.; Myers, A. G. A Practical, Enantioselective Synthetic Route to a Key Precursor to the Tetracycline Antibiotics Org. Lett. 2007, 9, 3523 - 3525
Cyclization Reactions of N -Acryloyl-2-aminobenzaldehyde Derivatives: Formal Total Synthesis of Martinellic Acid
He, Y.; Mahmud, H.; Moningka, R.; Lovely, C. J.; Dias, H. V. R. Cyclization Reactions of N -Acryloyl-2-aminobenzaldehyde Derivatives: Formal Total Synthesis of Martinellic Acid Tetrahedron 2006, 62, 8755 - 8769
Tetracycline Analogs and Their Therapeutic Use against Infections
PCT Int. Appl. WO, 2102
Chen, C.-L.; Clark, R. B.; Deng, Y.; Plamondon, L.; Sun, C.; Xiao, X.-Y. Tetracycline Analogs and Their Therapeutic Use against Infections. PCT Int. Appl. WO 201202712, 2102.
Development and Characterization of a Pseudomonas aeruginosa in Vitro Coupled Transcription-Translation Assay System for Evaluation of Translation Inhibitors
Fyfe, C.; Sutcliffe, J. A.; Grossman, T. H. Development and Characterization of a Pseudomonas aeruginosa in Vitro Coupled Transcription-Translation Assay System for Evaluation of Translation Inhibitors J. Microbiol. Methods 2012, 90, 256 - 261
Methods for Dilution Antimicrobial Susceptibility for Bacteria That Grow Aerobically: Approved Standard
9th ed. Clinical and Laboratory Standards Institute (CLSI): 940 West Valley Road, Suite 1400, Wayne, Pennsylvania
Methods for Dilution Antimicrobial Susceptibility for Bacteria That Grow Aerobically: Approved Standard, 9th ed.; CLSI document M07-A9E; Clinical and Laboratory Standards Institute (CLSI): 940 West Valley Road, Suite 1400, Wayne, Pennsylvania, 2012; Vol. 32, no. 2.