Caffeine inhibits glucose transport by binding at the GLUT1 nucleotide-binding site

American Journal of Physiology - Cell Physiology

Volumn 308, Issue 10, 2015, Pages C827-C834

  Sage, Jay M ^a   Cura, Anthony J ^a   Lloyd, Kenneth P ^a   Carruthers, Anthony ^a  

^a UNIVERSITY OF MASSACHUSETTS MEDICAL SCHOOL   (United States)

Author keywords

ATP; Caffeine; Erythrocyte; Glucose transport; GLUT1

Indexed keywords

3 METHYLGLUCOSE; ADENOSINE PHOSPHATE; ADENOSINE TRIPHOSPHATE; ADENOSINE TRIPHOSPHATE DERIVATIVE; CAFFEINE; CYTOCHALASIN B; GLUCOSE; GLUCOSE TRANSPORTER 1; SLC2A1 PROTEIN, HUMAN;

ANTIGEN BINDING; ARTICLE; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; CRYSTAL STRUCTURE; DOSE RESPONSE; ERYTHROCYTE GHOST; GLUCOSE TRANSPORT; HUMAN; HUMAN CELL; NUCLEOTIDE BINDING SITE; PRIORITY JOURNAL; PROTEIN BINDING; SUGAR TRANSPORT; BINDING SITE; DRUG EFFECTS; ERYTHROCYTE; ERYTHROCYTE MEMBRANE; METABOLISM; PHYSIOLOGY; SIGNAL TRANSDUCTION; TRANSPORT AT THE CELLULAR LEVEL;

3-O-METHYLGLUCOSE; ADENOSINE TRIPHOSPHATE; BINDING SITES; BIOLOGICAL TRANSPORT; CAFFEINE; CYTOCHALASIN B; ERYTHROCYTE MEMBRANE; ERYTHROCYTES; GLUCOSE; GLUCOSE TRANSPORTER TYPE 1; HUMANS; SIGNAL TRANSDUCTION;

EID: 84930899862     PISSN: 03636143     EISSN: 15221563     Source Type: Journal    
DOI: 10.1152/ajpcell.00001.2015     Document Type: Article

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