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Angewandte Chemie - International Edition

Volumn 54, Issue 8, 2015, Pages 2501-2504

Orchestrated triple C-H activation reactions using two directing groups: Rapid assembly of complex pyrazoles

(8) Yang, Weibo a Ye, Shengqing a Fanning, Dewey b Coon, Timothy b Schmidt, Yvonne b Krenitsky, Paul b Stamos, Dean b Yu, Jin Quan a

a SCRIPPS RESEARCH INSTITUTE (United States)

b VERTEX PHARMACEUTICALS (United States)

Author keywords

Benzo e indazoles; C H activation; Cascade reactions; Pyrazole

Indexed keywords

ACTIVATION ANALYSIS; REACTION KINETICS; SYNTHESIS (CHEMICAL);

AMIDE GROUPS; BENZO[E]INDAZOLES; C-H ACTIVATION; CASCADE REACTIONS; DIRECTING GROUPS; INDAZOLE; PYRAZOLES; STERICALLY CONGESTED;

CHEMICAL ACTIVATION;

CARBON; HYDROGEN; PALLADIUM; PYRAZOLE DERIVATIVE;

CATALYSIS; CHEMISTRY; SYNTHESIS;

CARBON; CATALYSIS; HYDROGEN; PALLADIUM; PYRAZOLES;

EID: 84922660479 PISSN: 14337851 EISSN: 15213773 Source Type: Journal
DOI: 10.1002/anie.201410462 Document Type: Article

Times cited : (61)

References (44)

1
- 72449170089
- a) L. Ackermann, R. Vicente, A. R. Kapdi, Angew. Chem. Int. Ed. 2009, 48, 9792;
- (2009) Angew. Chem. Int. Ed. , vol.48 , pp. 9792
- Ackermann, L.¹ Vicente, R.² Kapdi, A.R.³

2
- 84860612002
- Angew. Chem. 2009, 121, 9976;
- (2009) Angew. Chem. , vol.121 , pp. 9976

3
- 34250655628
- b) I. V. Seregin, V. Gevorgyan, Chem. Soc. Rev. 2007, 36, 1173;
- (2007) Chem. Soc. Rev. , vol.36 , pp. 1173
- Seregin, I.V.¹ Gevorgyan, V.²

4
- 68949185025
- c) O. Daugulis, H.-Q. Do, D. Shabashov, Acc. Chem. Res. 2009, 42, 1074;
- (2009) Acc. Chem. Res. , vol.42 , pp. 1074
- Daugulis, O.¹ Do, H.-Q.² Shabashov, D.³

5
- 77949381429
- d) T.W. Lyons, M. S. Sanford, Chem. Rev. 2010, 110, 1147;
- (2010) Chem. Rev. , vol.110 , pp. 1147
- Lyons, T.W.¹ Sanford, M.S.²

6
- 67649488045
- e) X. Chen, K. M. Engle, D.-H. Wang, J.-Q. Yu, Angew. Chem. Int. Ed. 2009, 48, 5094;
- (2009) Angew. Chem. Int. Ed. , vol.48 , pp. 5094
- Chen, X.¹ Engle, K.M.² Wang, D.-H.³ Yu, J.-Q.⁴

7
- 79960605080
- Angew. Chem. 2009, 121, 5196;
- (2009) Angew. Chem. , vol.121 , pp. 5196

8
- 80054728269
- f) S.-H. Cho, J. Y. Kim, J. Kwak, S. Chang, Chem. Soc. Rev. 2011, 40, 5068;
- (2011) Chem. Soc. Rev. , vol.40 , pp. 5068
- Cho, S.-H.¹ Kim, J.Y.² Kwak, J.³ Chang, S.⁴

9
- 80054972215
- g) O. Baudoin, Chem. Soc. Rev. 2011, 40, 4902;
- (2011) Chem. Soc. Rev. , vol.40 , pp. 4902
- Baudoin, O.¹

10
- 84886793220
- h) G. Rouquet, N. Chatani, Angew. Chem. Int. Ed. 2013, 52, 11726;
- (2013) Angew. Chem. Int. Ed. , vol.52 , pp. 11726
- Rouquet, G.¹ Chatani, N.²

11
- 84915753366
- Angew. Chem. 2013, 125, 11942.
- (2013) Angew. Chem. , vol.125 , pp. 11942

12
- 84868581721
- a) T. Piou, L. Neuville, J. Zhu, Angew. Chem. Int. Ed. 2012, 51, 11561;
- (2012) Angew. Chem. Int. Ed , vol.51 , pp. 11561
- Piou, T.¹ Neuville, L.² Zhu, J.³

13
- 84875311188
- Angew. Chem. 2012, 124, 11729;
- (2012) Angew. Chem. , vol.124 , pp. 11729

14
- 84887535835
- b) T. Piou, A. Bunescu, Q. Wang, L. Neuville, J. Zhu, Angew. Chem. Int. Ed. 2013, 52, 12385;
- (2013) Angew. Chem. Int. Ed , vol.52 , pp. 12385
- Piou, T.¹ Bunescu, A.² Wang, Q.³ Neuville, L.⁴ Zhu, J.⁵

15
- 84941599510
- Angew. Chem. 2013, 125, 12611.
- (2013) Angew. Chem. , vol.125 , pp. 12611

16
- 77953892735
- c) P. Gandeepan, K. Parthasarathy, C.-H. Cheng, J. Am. Chem. Soc. 2010, 132, 8569;
- (2010) J. Am. Chem. Soc. , vol.132 , pp. 8569
- Gandeepan, P.¹ Parthasarathy, K.² Cheng, C.-H.³

17
- 79551664541
- d) G.-W. Wang, T.-T. Yuan, D.-D. Li, Angew. Chem. Int. Ed. 2011, 50, 1380;
- (2011) Angew. Chem. Int. Ed. , vol.50 , pp. 1380
- Wang, G.-W.¹ Yuan, T.-T.² Li, D.-D.³

18
- 84937518480
- Angew. Chem. 2011, 123, 1416;
- (2011) Angew. Chem. , vol.123 , pp. 1416

19
- 84900022748
- e) M. Sickert, H. Weinstabl, B. Peters, X. Hou, M. Lautens, Angew. Chem. Int. Ed. 2014, 53, 5147;
- (2014) Angew. Chem. Int. Ed. , vol.53 , pp. 5147
- Sickert, M.¹ Weinstabl, H.² Peters, B.³ Hou, X.⁴ Lautens, M.⁵

20
- 84944280244
- Angew. Chem. 2014, 126, 5247;
- (2014) Angew. Chem. , vol.126 , pp. 5247

21
- 2942643950
- f) Q. Huang, A. Fazio, G. Dai, M. A. Campo, R. C. Larock, J. Am. Chem. Soc. 2004, 126, 7460;
- (2004) J. Am. Chem. Soc. , vol.126 , pp. 7460
- Huang, Q.¹ Fazio, A.² Dai, G.³ Campo, M.A.⁴ Larock, R.C.⁵

22
- 75749123423
- g) Z. Lu, C. Hu, J. Guo, J. Li, Y. Cui, Y. Jia, Org. Lett. 2010, 12, 480;
- (2010) Org. Lett. , vol.12 , pp. 480
- Lu, Z.¹ Hu, C.² Guo, J.³ Li, J.⁴ Cui, Y.⁵ Jia, Y.⁶

23
- 80955179609
- h) Z. Lu, Y. Cui, Y. Jia, Synthesis 2011, 2595.
- (2011) Synthesis , pp. 2595
- Lu, Z.¹ Cui, Y.² Jia, Y.³

24
- 84884931642
- a) V. Kumar, K. Kaur, G. K. Gupta, A. K. Sharma, Eur. J. Med. Chem. 2013, 69, 735;
- (2013) Eur. J. Med. Chem. , vol.69 , pp. 735
- Kumar, V.¹ Kaur, K.² Gupta, G.K.³ Sharma, A.K.⁴

25
- 84896877886
- b) A. El-Mekabaty, Synth. Commun. 2014, 44, 875;
- (2014) Synth. Commun. , vol.44 , pp. 875
- El-Mekabaty, A.¹

26
- 23044434912
- c) D. Marcic, Exp. Appl. Acarol. 2005, 36, 177;
- (2005) Exp. Appl. Acarol. , vol.36 , pp. 177
- Marcic, D.¹

27
- 84906234396
- d) R. Román, A. Navarro, D. Wodka, M. Alvim-Gaston, S. Husain, N. Franklin, A. Simoìn-Fuentes, S. Fustero, Org. Process Res. Dev. 2014, 18, 1027;
- (2014) Org. Process Res. Dev. , vol.18 , pp. 1027
- Román, R.¹ Navarro, A.² Wodka, D.³ Alvim-Gaston, M.⁴ Husain, S.⁵ Franklin, N.⁶ Simoìn-Fuentes, A.⁷ Fustero, S.⁸

28
- 72249108384
- e) M. Tao, C. H. Park, K. Josef, R. L. Hudkins, J. Heterocycl. Chem. 2009, 46, 1185;
- (2009) J. Heterocycl. Chem. , vol.46 , pp. 1185
- Tao, M.¹ Park, C.H.² Josef, K.³ Hudkins, R.L.⁴

29
- 84877581275
- f) M. Nayaka, N. Rastogi, S. Batra, Tetrahedron 2013, 69, 5029.
- (2013) Tetrahedron , vol.69 , pp. 5029
- Nayaka, M.¹ Rastogi, N.² Batra, S.³

30
- 3042704672
- T. Asaumi, T. Matsuo, T. Fukuyama, Y. Ie, F. Kakiuchi, N. Chatani, J. Org. Chem. 2004, 69, 4433.
- (2004) J. Org. Chem. , vol.69 , pp. 4433
- Asaumi, T.¹ Matsuo, T.² Fukuyama, T.³ Ie, Y.⁴ Kakiuchi, F.⁵ Chatani, N.⁶

31
- 84877292512
- a) H. Wang, N. Schrc¸der, F. Glorius, Angew. Chem. Int. Ed. 2013, 52, 5386;
- (2013) Angew. Chem. Int. Ed , vol.52 , pp. 5386
- Wang, H.¹ Schrc¸der, N.² Glorius, F.³

32
- 84930627298
- Angew. Chem. 2013, 125, 5495;
- (2013) Angew. Chem. , vol.125 , pp. 5495

33
- 84897060105
- b) F. Xie, Z. Qi, S. Yu, X. Li, J. Am. Chem. Soc. 2014, 136, 4780;
- (2014) J. Am. Chem. Soc. , vol.136 , pp. 4780
- Xie, F.¹ Qi, Z.² Yu, S.³ Li, X.⁴

34
- 84880851657
- c) T.-J. Gong, B. Xiao, W.-M. Cheng,W. Su, J. Xu, Z.-J. Liu, L. Liu, Y. Fu, J. Am. Chem. Soc. 2013, 135, 10630;
- (2013) J. Am. Chem. Soc. , vol.135 , pp. 10630
- Gong, T.-J.¹ Xiao, B.² Cheng, W.-M.³ Su, W.⁴ Xu, J.⁵ Liu, Z.-J.⁶ Liu, L.⁷ Fu, Y.⁸

35
- 33746307336
- d) L. Ackermann, A. Althammer, R. Born, Angew. Chem. Int. Ed. 2006, 45, 2619;
- (2006) Angew. Chem. Int. Ed. , vol.45 , pp. 2619
- Ackermann, L.¹ Althammer, A.² Born, R.³

36
- 84899478383
- Angew. Chem. 2006, 118, 2681;
- (2006) Angew. Chem. , vol.118 , pp. 2681

37
- 53549115668
- e) L. V. Desai, K. J. Stowers, M. S. Sanford, J. Am. Chem. Soc. 2008, 130, 13285;
- (2008) J. Am. Chem. Soc. , vol.130 , pp. 13285
- Desai, L.V.¹ Stowers, K.J.² Sanford, M.S.³

38
- 84875698071
- f) M. Schinkel, I. Marek, L. Ackermann, Angew. Chem. Int. Ed. 2013, 52, 3977;
- (2013) Angew. Chem. Int. Ed. , vol.52 , pp. 3977
- Schinkel, M.¹ Marek, I.² Ackermann, L.³

39
- 84903210543
- Angew. Chem. 2013, 125, 4069;
- (2013) Angew. Chem. , vol.125 , pp. 4069

40
- 84865263016
- g) K. Muralirajan, K. Parthasarathy, C.-H. Cheng, Org. Lett. 2012, 14, 4262;
- (2012) Org. Lett. , vol.14 , pp. 4262
- Muralirajan, K.¹ Parthasarathy, K.² Cheng, C.-H.³

41
- 84872564556
- h) Y. Hashimoto, K. Hirano, T. Satoh, F. Kakiuchi, M. Miura, J. Org. Chem. 2013, 78, 638.
- (2013) J. Org. Chem. , vol.78 , pp. 638
- Hashimoto, Y.¹ Hirano, K.² Satoh, T.³ Kakiuchi, F.⁴ Miura, M.⁵

42
- 33947644069
- R. Giri, N. Maugel, J.-J. Li, D.-H. Wang, S. P. Breazzano, L. B. Saunders, J.-Q. Yu, J. Am. Chem. Soc. 2007, 129, 3510.
- (2007) J. Am. Chem. Soc. , vol.129 , pp. 3510
- Giri, R.¹ Maugel, N.² Li, J.-J.³ Wang, D.-H.⁴ Breazzano, S.P.⁵ Saunders, L.B.⁶ Yu, J.-Q.⁷

43
- 80052602187
- M. Wasa, K. S. L. Chan, J.-Q. Yu, Chem. Lett. 2011, 40, 1004.
- (2011) Chem. Lett. , vol.40 , pp. 1004
- Wasa, M.¹ Chan, K.S.L.² Yu, J.-Q.³

44
- 54849436434
- M. Wasa, J.-Q. Yu, J. Am. Chem. Soc. 2008, 130, 14058.
- (2008) J. Am. Chem. Soc. , vol.130 , pp. 14058
- Wasa, M.¹ Yu, J.-Q.²

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