메뉴 건너뛰기




Volumn 75, Issue 2, 2015, Pages 387-393

In vivo radioimaging of bradykinin receptor B1, a widely overexpressed molecule in human cancer

Author keywords

[No Author keywords available]

Indexed keywords

BRADYKININ B1 RECEPTOR; ENALAPRILAT; GALLIUM TETRAXETAN AMINOHEXANOIC ACID [4 HYDROXYPROLINE 6 CHA 9 LEUCINE 10 DESARGININE]KALLIDIN GA 68; GALLIUM TETRAXETAN AMINOHEXANOIC ACID [9 LEUCIN 10 DESARGININE]KALLIDIN GA 68; GALLIUM TETRAXETAN POLYETHYLENE GLYCOL 2 [4 HYDROXYPROLINE 6 CHA 9 LEUCINE 10 DESARGININE]KALLIDIN GA 68; KALLIDIN DERIVATIVE; PEPTIDASE; PHOSPHORAMIDON; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG; GALLIUM; ORGANOMETALLIC COMPOUND; PEPTIDE;

EID: 84920997436     PISSN: 00085472     EISSN: 15387445     Source Type: Journal    
DOI: 10.1158/0008-5472.CAN-14-1603     Document Type: Article
Times cited : (51)

References (20)
  • 1
    • 6444236841 scopus 로고    scopus 로고
    • Bradykinin receptor ligands: Therapeutic perspectives
    • Marceau F, Regoli D. Bradykinin receptor ligands: therapeutic perspectives. Nat Rev Drug Discov 2004;3:845-52.
    • (2004) Nat Rev Drug Discov , vol.3 , pp. 845-852
    • Marceau, F.1    Regoli, D.2
  • 2
    • 84893805673 scopus 로고    scopus 로고
    • The role of kinin receptors in cancer and therapeutic opportunities
    • da Costa PL, Sirois P, Tannock IF, ChammasR. The role of kinin receptors in cancer and therapeutic opportunities. Cancer Lett 2014;345:27-38.
    • (2014) Cancer Lett , vol.345 , pp. 27-38
    • Da Costa, P.L.1    Sirois, P.2    Tannock, I.F.3    Chammasr4
  • 3
    • 70449561221 scopus 로고    scopus 로고
    • Stimulation of the bradykinin B(1) receptor induces the proliferation of estrogen-sensitive breast cancer cells and activates the ERK1/2 signaling pathway
    • Molina L, Matus CE, Astroza A, Pavicic F, Tapia E, Toledo C, et al. Stimulation of the bradykinin B(1) receptor induces the proliferation of estrogen-sensitive breast cancer cells and activates the ERK1/2 signaling pathway. Breast Cancer Res Treat 2009;118:499-510.
    • (2009) Breast Cancer Res Treat , vol.118 , pp. 499-510
    • Molina, L.1    Matus, C.E.2    Astroza, A.3    Pavicic, F.4    Tapia, E.5    Toledo, C.6
  • 4
    • 0037729000 scopus 로고    scopus 로고
    • Bradykinin receptor subtype 1 expression and function in prostate cancer
    • Taub JS, Guo R, Leeb-Lundberg LM, Madden JF, Daaka Y. Bradykinin receptor subtype 1 expression and function in prostate cancer. Cancer Res 2003;63:2037-41.
    • (2003) Cancer Res , vol.63 , pp. 2037-2041
    • Taub, J.S.1    Guo, R.2    Leeb-Lundberg, L.M.3    Madden, J.F.4    Daaka, Y.5
  • 5
    • 78650558263 scopus 로고    scopus 로고
    • Activation of kinin B1 receptor increases the release of metalloproteases-2 and-9 from both estrogen-sensitive and-insensitive breast cancer cells
    • Ehrenfeld P, Conejeros I, Pavicic MF, Matus CE, Gonzalez CB, Quest AF, et al. Activation of kinin B1 receptor increases the release of metalloproteases-2 and-9 from both estrogen-sensitive and-insensitive breast cancer cells. Cancer Lett 2011;301:106-18.
    • (2011) Cancer Lett , vol.301 , pp. 106-118
    • Ehrenfeld, P.1    Conejeros, I.2    Pavicic, M.F.3    Matus, C.E.4    Gonzalez, C.B.5    Quest, A.F.6
  • 6
    • 84870481545 scopus 로고    scopus 로고
    • Bradykinin enhances cell migration in human prostate cancer cells through B2 receptor/PKCdelta/c-Src dependent signaling pathway
    • Yu HS, Lin TH, Tang CH. Bradykinin enhances cell migration in human prostate cancer cells through B2 receptor/PKCdelta/c-Src dependent signaling pathway. Prostate 2013;73:89-100.
    • (2013) Prostate , vol.73 , pp. 89-100
    • Yu, H.S.1    Lin, T.H.2    Tang, C.H.3
  • 7
    • 84878154975 scopus 로고    scopus 로고
    • The kinin-kallikrein system: Physiological roles, pathophysiology and its relationship to cancer biomarkers
    • Kashuba E, Bailey J, Allsup D, Cawkwell L. The kinin-kallikrein system: physiological roles, pathophysiology and its relationship to cancer biomarkers. Biomarkers 2013;18:279-96.
    • (2013) Biomarkers , vol.18 , pp. 279-296
    • Kashuba, E.1    Bailey, J.2    Allsup, D.3    Cawkwell, L.4
  • 8
    • 0036097190 scopus 로고    scopus 로고
    • Bradykinin antagonist dimer, CU201, inhibits the growth of human lung cancer cell lines in vitro and in vivo and produces synergistic growth inhibition in combination with other antitumor agents
    • Chan DC, Gera L, Stewart JM, Helfrich B, Zhao TL, Feng WY, et al. Bradykinin antagonist dimer, CU201, inhibits the growth of human lung cancer cell lines in vitro and in vivo and produces synergistic growth inhibition in combination with other antitumor agents. Clin Cancer Res 2002;8:1280-7.
    • (2002) Clin Cancer Res , vol.8 , pp. 1280-1287
    • Chan, D.C.1    Gera, L.2    Stewart, J.M.3    Helfrich, B.4    Zhao, T.L.5    Feng, W.Y.6
  • 10
    • 63849308514 scopus 로고    scopus 로고
    • Fluorescent ligands of the bradykinin B1 receptors: Pharmacologic characterization and application to the study of agonist-induced receptor translocation and cell surface receptor expression
    • Bawolak MT, Gera L, Morissette G, Bouthillier J, Stewart JM, Gobeil LA, et al. Fluorescent ligands of the bradykinin B1 receptors: pharmacologic characterization and application to the study of agonist-induced receptor translocation and cell surface receptor expression. J Pharmacol Exp Ther 2009;329:159-68.
    • (2009) J Pharmacol Exp Ther , vol.329 , pp. 159-168
    • Bawolak, M.T.1    Gera, L.2    Morissette, G.3    Bouthillier, J.4    Stewart, J.M.5    Gobeil, L.A.6
  • 11
    • 84859433492 scopus 로고    scopus 로고
    • N-terminal extended conjugates of the agonists and antagonists of both bradykinin receptor subtypes: Structure-activity relationship, cell imaging using ligands conjugated with fluorophores and prospect for functionally active cargoes
    • Gera L, Roy C, Bawolak MT, Charest-Morin X, Marceau F. N-terminal extended conjugates of the agonists and antagonists of both bradykinin receptor subtypes: structure-activity relationship, cell imaging using ligands conjugated with fluorophores and prospect for functionally active cargoes. Peptides 2012;34:433-46.
    • (2012) Peptides , vol.34 , pp. 433-446
    • Gera, L.1    Roy, C.2    Bawolak, M.T.3    Charest-Morin, X.4    Marceau, F.5
  • 13
  • 14
    • 0034044596 scopus 로고    scopus 로고
    • Posttranscriptional regulation of bradykinin B1 and B2 receptor gene expression in human lung fibroblasts by tumor necrosis factor-alpha: Modulation by dexamethasone
    • Haddad EB, Fox AJ, Rousell J, Burgess G, McIntyre P, Barnes PJ, et al. Posttranscriptional regulation of bradykinin B1 and B2 receptor gene expression in human lung fibroblasts by tumor necrosis factor-alpha: modulation by dexamethasone. Mol Pharmacol 2000;57:1123-31.
    • Mol Pharmacol 2000 , vol.57 , pp. 1123-1131
    • Haddad, E.B.1    Fox, A.J.2    Rousell, J.3    Burgess, G.4    McIntyre, P.5    Barnes, P.J.6
  • 15
    • 0021211465 scopus 로고
    • The metabolism of neuropeptides: The hydrolysis of peptides, including enkephalins, tachykinins and their analogues, by endopeptidase-24. 11
    • Matsas R, Kenny AJ, Turner AJ. The metabolism of neuropeptides. The hydrolysis of peptides, including enkephalins, tachykinins and their analogues, by endopeptidase-24. 11. Biochem J 1984;223:433-40.
    • (1984) Biochem J , vol.223 , pp. 433-440
    • Matsas, R.1    Kenny, A.J.2    Turner, A.J.3
  • 16
    • 84894728566 scopus 로고    scopus 로고
    • To serve and protect": Enzyme inhibitors as radiopeptide escorts promote tumor targeting
    • Nock BA, Maina T, Krenning EP, de Jong M. "To serve and protect": enzyme inhibitors as radiopeptide escorts promote tumor targeting. J Nucl Med 2014;55:121-7.
    • (2014) J Nucl Med , vol.55 , pp. 121-127
    • Nock, B.A.1    Maina, T.2    Krenning, E.P.3    De Jong, M.4
  • 18
    • 79953708503 scopus 로고    scopus 로고
    • Renal uptake of different radiolabelled peptides is mediated by megalin: SPECT and biodistribution studies in megalin-deficient mice
    • Vegt E, Melis M, Eek A, de Visser M, BromM, Oyen WJ, et al. Renal uptake of different radiolabelled peptides is mediated by megalin: SPECT and biodistribution studies in megalin-deficient mice. Eur J Nucl Med Mol Imaging 2011;38:623-32.
    • (2011) Eur J Nucl Med Mol Imaging , vol.38 , pp. 623-632
    • Vegt, E.1    Melis, M.2    Eek, A.3    De Visser, M.4    Brom, M.5    Oyen, W.J.6
  • 19
    • 84885304780 scopus 로고    scopus 로고
    • Effects of chelator modifications on (68)Galabeled [Tyr (3)]octreotide conjugates
    • Lin M, Welch MJ, Lapi SE. Effects of chelator modifications on (68)Galabeled [Tyr (3)]octreotide conjugates. Mol Imaging Biol 2013;15: 606-13.
    • (2013) Mol Imaging Biol , vol.15 , pp. 606-613
    • Lin, M.1    Welch, M.J.2    Lapi, S.E.3
  • 20
    • 84866184119 scopus 로고    scopus 로고
    • Unexpected sensitivity of sst2 antagonists to N-terminal radiometal modifications
    • Fani M, Braun F, Waser B, Beetschen K, Cescato R, Erchegyi J, et al. Unexpected sensitivity of sst2 antagonists to N-terminal radiometal modifications. J Nucl Med 2012;53:1481-9.
    • (2012) J Nucl Med , vol.53 , pp. 1481-1489
    • Fani, M.1    Braun, F.2    Waser, B.3    Beetschen, K.4    Cescato, R.5    Erchegyi, J.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.