Microwave assisted synthesis and docking study of N-(2-oxo-2-(4-oxo-2-substituted thiazolidin-3ylamino)ethyl)benzamide derivatives as anticonvulsant agents

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 24, 2014, Pages 5558-5562

  Nikalje, Anna Pratima G ^a   Shaikh, Arfat N ^a   Shaikh, Sameer I ^a   Kalam Khan, Firoz A ^a   Sangshetti, Jaiprakash N ^a   Shinde, Devanand B ^b  

^a Y B CHAVAN COLLEGE OF PHARMACY   (India)

^b DR BABASAHEB AMBEDKAR MARATHWADA UNIVERSITY   (India)

Author keywords

Anticonvulsant evaluation; Benzamide; Computational studies; Microwave irradiation; Thiazolidinone

Indexed keywords

ANTICONVULSIVE AGENT; BENZAMIDE DERIVATIVE; DIAZEPAM; PHENYTOIN; SODIUM CHANNEL; THIAZOLIDINE DERIVATIVE;

ANIMAL BEHAVIOR; ANIMAL EXPERIMENT; ANIMAL TISSUE; ANTICONVULSANT ACTIVITY; ARTICLE; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG ABSORPTION; DRUG BINDING; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ELECTROSHOCK SEIZURE; HISTOPATHOLOGY; HYDROGEN BOND; HYDROPHILICITY; HYDROPHOBICITY; LOCOMOTION; MAXIMAL ELECTROSHOCK SEIZURE; MICROWAVE ASSISTED SYNTHESIS; MICROWAVE IRRADIATION; MOLECULAR DOCKING; MOLECULAR WEIGHT; MOUSE; NEUROTOXICITY; NONHUMAN; ANIMAL; BINDING SITE; CHEMISTRY; DISEASE MODEL; DRUG EFFECTS; HALF LIFE TIME; LIVER; METABOLISM; MICROWAVE RADIATION; MOTOR ACTIVITY; PATHOLOGY; PROTEIN TERTIARY STRUCTURE; SEIZURES; SYNTHESIS;

ANIMALS; ANTICONVULSANTS; BENZAMIDES; BINDING SITES; DISEASE MODELS, ANIMAL; HALF-LIFE; LIVER; MICE; MICROWAVES; MOLECULAR DOCKING SIMULATION; MOTOR ACTIVITY; PROTEIN STRUCTURE, TERTIARY; SEIZURES; SODIUM CHANNELS; THIAZOLIDINES;

EID: 84911918344     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2014.11.016     Document Type: Article

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