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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 20, 2014, Pages 4871-4875

The design and implementation of a generic lipopeptide scanning platform to enable the identification of 'locally acting' agonists for the apelin receptor

(8) McKeown, Stephen C a Zecri, Frederic J a Fortier, Eric a Taggart, Andrew a Sviridenko, Lilya a Adams, Christopher M a McAllister, Kathryn H a Pin, Sokhom S a

a NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH (United States)

Author keywords

Apelin; APJ agonist; Lipopeptide; Pepducin; Peptide; Protein protein interactions

Indexed keywords

APLNR PROTEIN, HUMAN; G PROTEIN COUPLED RECEPTOR; LIPOPEPTIDE;

AGONISTS; CHEMISTRY; CONFORMATION; DOSE RESPONSE; DRUG DESIGN; GENETICS; HUMAN; STRUCTURE ACTIVITY RELATION;

DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; HUMANS; LIPOPEPTIDES; MOLECULAR CONFORMATION; RECEPTORS, G-PROTEIN-COUPLED; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84908680936 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.08.045 Document Type: Article

Times cited : (12)

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