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Volumn 1099, Issue , 2012, Pages 323-338

Use of in vitro data in PBPK models: An example of in vitro to in vivo extrapolation with carbaryl

Author keywords

[No Author keywords available]

Indexed keywords

COMPUTATIONAL CHEMISTRY; EXTRAPOLATION; RATS; RISK ASSESSMENT;

EID: 84905638162     PISSN: 00976156     EISSN: 19475918     Source Type: Book Series    
DOI: 10.1021/bk-2012-1099.ch020     Document Type: Conference Paper
Times cited : (8)

References (33)
  • 1
    • 59149106151 scopus 로고    scopus 로고
    • Toxicity testing in the 21st century: Bringing the vision to life
    • Andersen, M. E.; Krewski, D. Toxicity testing in the 21st century: Bringing the vision to life. Toxicol. Sei. 2009, 707(2), 324-30.
    • (2009) Toxicol. Sei. , vol.707 , Issue.2 , pp. 324-330
    • Andersen, M.E.1    Krewski, D.2
  • 2
    • 85122905591 scopus 로고    scopus 로고
    • Vitro to in vivo extrapolation of metabolic rate constants for physiologically based pharmacokinetic models
    • Lipscomb, J. C, Ohanian, E. V, Eds.; Informa Healthcare: New York
    • Kedderis, G. L. In Vitro to In Vivo Extrapolation of Metabolic Rate Constants for Physiologically Based Pharmacokinetic Models. In Toxicokinetics and Risk Assessment; Lipscomb, J. C, Ohanian, E. V, Eds.; Informa Healthcare: New York, 2007; pp 185-210.
    • (2007) Toxicokinetics and Risk Assessment , pp. 185-210
    • Kedderis, G.L.1
  • 3
    • 42649085362 scopus 로고    scopus 로고
    • Vitro measurements of metabolism for application in pharmacokinetic modeling
    • Lipscomb, J. C.; Poet, T. S. In vitro measurements of metabolism for application in pharmacokinetic modeling. Pharmacol. Ther. 2008, 118 (1), 82-103.
    • (2008) Pharmacol. Ther. , vol.118 , Issue.1 , pp. 82-103
    • Lipscomb, J.C.1    Poet, T.S.2
  • 5
    • 79956192126 scopus 로고    scopus 로고
    • Cytochrome P450-specific human PBPK/PD models for the organophosphorus pesticides: Chlorpyrifos and parathion
    • Foxenberg, R. J.; Ellison, C. A.; Knaak, J. B.; Ma, C.; Olson, J. R. Cytochrome P450-specific human PBPK/PD models for the organophosphorus pesticides: Chlorpyrifos and parathion. Toxicology 2011, 285 (1-2), 57-66.
    • (2011) Toxicology , vol.285 , Issue.1-2 , pp. 57-66
    • Foxenberg, R.J.1    Ellison, C.A.2    Knaak, J.B.3    Ma, C.4    Olson, J.R.5
  • 6
    • 33748745121 scopus 로고    scopus 로고
    • Development of a physiologically based pharmacokinetic model for deltamethrin in the adult male Sprague-Dawley rat
    • Mirfazaelian, A.; Kim, K. B.; Anand, S. S.; Kim, H. J.; Tornero-Velez, R.; Bruckner, J. V.; Fisher, J. W. Development of a physiologically based pharmacokinetic model for deltamethrin in the adult male Sprague-Dawley rat. Toxicol. Sei. 2006, 93 (2), 432-12.
    • (2006) Toxicol. Sei. , vol.93 , Issue.2 , pp. 432-512
    • Mirfazaelian, A.1    Kim, K.B.2    Anand, S.S.3    Kim, H.J.4    Tornero-Velez, R.5    Bruckner, J.V.6    Fisher, J.W.7
  • 9
    • 9244257295 scopus 로고    scopus 로고
    • Vitro metabolism of carbofuran by human, mouse, and rat cytochrome P450 and interactions with chlorpyrifos, testosterone, and estradiol
    • Usmani, K. A.; Hodgson, E.; Rose, R. L. In vitro metabolism of carbofuran by human, mouse, and rat cytochrome P450 and interactions with chlorpyrifos, testosterone, and estradiol. Chem. Biol. Interact. 2004, 150(3), 221-32.
    • (2004) Chem. Biol. Interact. , vol.150 , Issue.3 , pp. 221-232
    • Usmani, K.A.1    Hodgson, E.2    Rose, R.L.3
  • 10
    • 0037051175 scopus 로고    scopus 로고
    • Enzymes involved in the detoxification of organophosphorus, carbamate and pyrethroid insecticides through hydrolysis
    • Sogorb, M. A.; Vilanova, E. Enzymes involved in the detoxification of organophosphorus, carbamate and pyrethroid insecticides through hydrolysis. Toxicol. Lett. 2002, 128 (1-3), 215-28.
    • (2002) Toxicol. Lett. , vol.128 , Issue.1-3 , pp. 215-228
    • Sogorb, M.A.1    Vilanova, E.2
  • 11
    • 0037145411 scopus 로고    scopus 로고
    • Vitro metabolism of carbaryl by human cytochrome P450 and its inhibition by chlorpyrifos
    • Tang, J.; Cao, Y.; Rose, R. L.; Hodgson, E. In vitro metabolism of carbaryl by human cytochrome P450 and its inhibition by chlorpyrifos. Chem. Biol. Interact. 2002, 141 (3), 229-41.
    • (2002) Chem. Biol. Interact. , vol.141 , Issue.3 , pp. 229-241
    • Tang, J.1    Cao, Y.2    Rose, R.L.3    Hodgson, E.4
  • 14
    • 49649113402 scopus 로고    scopus 로고
    • 3rd Bayesian calibration of a physiologically based pharmacokinetic/ pharmacodynamic model of carbaryl Cholinesterase inhibition
    • Nong, A.; Tan, Y. M.; Krolski, M. E.; Wang, J.; Lunchick, C.; Conolly, R. B.; Clewell, H. J., 3rd Bayesian calibration of a physiologically based pharmacokinetic/pharmacodynamic model of carbaryl Cholinesterase inhibition. J. Toxicol. Environ. Health, Part A 2008, 71 (20), 1363-81.
    • (2008) J. Toxicol. Environ. Health, Part A , vol.71 , Issue.20 , pp. 1363-1381
    • Nong, A.1    Tan, Y.M.2    Krolski, M.E.3    Wang, J.4    Lunchick, C.5    Conolly, R.B.6    Clewell, H.J.7
  • 16
    • 0043092060 scopus 로고    scopus 로고
    • Human hepatocytes as a tool for studying toxicity and drug metabolism
    • Gomez-Lechon, M. J.; Donate, M. T.; Castell, J. V.; Jover, R. Human hepatocytes as a tool for studying toxicity and drug metabolism. Curr Drug Metab. 2003, 4 (4), 292-312.
    • (2003) Curr Drug Metab. , vol.4 , Issue.4 , pp. 292-312
    • Gomez-Lechon, M.J.1    Donate, M.T.2    Castell, J.V.3    Jover, R.4
  • 18
    • 0027449673 scopus 로고
    • Nature and role of xenobiotic metabolizing esterases in rat liver, lung, skin and blood
    • McCracken, N. W.; Blain, P. G.; Williams, F. M. Nature and role of xenobiotic metabolizing esterases in rat liver, lung, skin and blood. Biochem. Pharmacol. 1993, 45 (1), 31-6.
    • (1993) Biochem. Pharmacol. , vol.45 , Issue.1 , pp. 31-36
    • McCracken, N.W.1    Blain, P.G.2    Williams, F.M.3
  • 19
    • 0029134578 scopus 로고
    • Regulatory and research issues related to Cholinesterase inhibition
    • Padilla, S. Regulatory and research issues related to Cholinesterase inhibition. Toxicology 1995, 102 (1-2), 215-20.
    • (1995) Toxicology , vol.102 , Issue.1-2 , pp. 215-220
    • Padilla, S.1
  • 20
    • 34547851657 scopus 로고    scopus 로고
    • Comparison of acute neurobehavioral and Cholinesterase inhibitory effects of N-methylcarbamates in rat
    • McDaniel, K. L.; Padilla, S.; Marshall, R. S.; Phillips, P. M.; Podhorniak, L.; Qian, Y.; Moser, V. C. Comparison of acute neurobehavioral and Cholinesterase inhibitory effects of N-methylcarbamates in rat. Toxicol. Sei. 2007, 98 (2), 552-60.
    • (2007) Toxicol. Sei. , vol.98 , Issue.2 , pp. 552-560
    • McDaniel, K.L.1    Padilla, S.2    Marshall, R.S.3    Phillips, P.M.4    Podhorniak, L.5    Qian, Y.6    Moser, V.C.7
  • 21
    • 0014690011 scopus 로고
    • Kinetics of Cholinesterase inhibition by organophosphate and carbamate insecticides
    • Main, A. R. Kinetics of Cholinesterase inhibition by organophosphate and carbamate insecticides. Can. Med. Assoc. J. 1969, 700(4), 161-7.
    • (1969) Can. Med. Assoc. J. , vol.700 , Issue.4 , pp. 161-167
    • Main, A.R.1
  • 22
    • 9644310412 scopus 로고    scopus 로고
    • Structural and functional organization of synaptic acetylcholinesterase
    • Aldunate, R.; Casar, J. C.; Brandan, E.; Inestrosa, N. C. Structural and functional organization of synaptic acetylcholinesterase. Brain Res. Brain Res. Rev. 2004, 47 (1-3), 96-104.
    • (2004) Brain Res. Brain Res. Rev. , vol.47 , Issue.1-3 , pp. 96-104
    • Aldunate, R.1    Casar, J.C.2    Brandan, E.3    Inestrosa, N.C.4
  • 23
    • 0021978929 scopus 로고
    • Acetylcholinesterase molecular forms in serum and erythrocytes of laboratory animals
    • Skau, K. A. Acetylcholinesterase molecular forms in serum and erythrocytes of laboratory animals. Comp. Biochem. Physiol, Part C 1985, 80 (1), 207-10.
    • (1985) Comp. Biochem. Physiol, Part C , vol.80 , Issue.1 , pp. 207-210
    • Skau, K.A.1
  • 25
    • 77954008507 scopus 로고    scopus 로고
    • Biokinetic modeling and in vitro-in vivo extrapolations
    • Blaauboer, B. J. Biokinetic modeling and in vitro-in vivo extrapolations. J. Toxicol. Environ. Health, Part B 2010, 13 (2-4), 242-52.
    • (2010) J. Toxicol. Environ. Health, Part B , vol.13 , Issue.2-4 , pp. 242-252
    • Blaauboer, B.J.1
  • 26
    • 79955021414 scopus 로고    scopus 로고
    • Mechanisms underlying differences in systemic exposure of structurally similar active metabolites: Comparison of two preclinical hepatic models
    • Yan, G. Z.; Brouwer, K. L.; Pollack, G. M.; Wang, M. Z.; Tidwell, R. R.; Hall, J. E.; Paine, M. F. Mechanisms underlying differences in systemic exposure of structurally similar active metabolites: Comparison of two preclinical hepatic models. J. Pharmacol. Exp. Ther 2011, 337(2), 503-12.
    • (2011) J. Pharmacol. Exp. Ther , vol.337 , Issue.2 , pp. 503-512
    • Yan, G.Z.1    Brouwer, K.L.2    Pollack, G.M.3    Wang, M.Z.4    Tidwell, R.R.5    Hall, J.E.6    Paine, M.F.7
  • 27
    • 0023444429 scopus 로고
    • Differences in the glycolipid membrane anchors of bovine and human erythrocyte acetylcholinesterases
    • Roberts, W. L.; Kim, B. H.; Rosenberry, T. L. Differences in the glycolipid membrane anchors of bovine and human erythrocyte acetylcholinesterases. Proc. Natl. Acad. Sei. U.S.A. 1987, 84 (22), 7817-21.
    • (1987) Proc. Natl. Acad. Sei. U.S.A. , vol.84 , Issue.22 , pp. 7817-7821
    • Roberts, W.L.1    Kim, B.H.2    Rosenberry, T.L.3
  • 28
    • 0026794615 scopus 로고
    • Cimetidine-carbaryl interaction in humans: Evidence for an active metabolite of carbaryl
    • May, D. G.; Naukam, R. J.; Kambam, J. R.; Branch, R. A. Cimetidine-carbaryl interaction in humans: Evidence for an active metabolite of carbaryl. J. Pharmacol. Exp. Ther. 1992, 262 (3), 1057-61.
    • (1992) J. Pharmacol. Exp. Ther. , vol.262 , Issue.3 , pp. 1057-1061
    • May, D.G.1    Naukam, R.J.2    Kambam, J.R.3    Branch, R.A.4
  • 29
    • 0019039022 scopus 로고
    • Gastrointestinal metabolism and transport of pesticidal carbamates
    • Pekas, J. C. Gastrointestinal metabolism and transport of pesticidal carbamates. Crit. Rev. Toxicol. 1980, 7(1), 37-101.
    • (1980) Crit. Rev. Toxicol. , vol.7 , Issue.1 , pp. 37-101
    • Pekas, J.C.1
  • 30
    • 0016747720 scopus 로고
    • Pharmacokinetics and metabolism of two carbamate insecticides, carbaryl and landrin, in the rat
    • Houston, J. B.; Upshall, D. G.; Bridges, J. W. Pharmacokinetics and metabolism of two carbamate insecticides, carbaryl and landrin, in the rat. Xenobiotica 1975, 5 (10), 637-48.
    • (1975) Xenobiotica , vol.5 , Issue.10 , pp. 637-648
    • Houston, J.B.1    Upshall, D.G.2    Bridges, J.W.3
  • 31
    • 0342437515 scopus 로고    scopus 로고
    • Enzyme-catalyzed processes of first-pass hepatic and intestinal drug extraction
    • Shen, D. D.; Kunze, K. L.; Thummel, K. E. Enzyme-catalyzed processes of first-pass hepatic and intestinal drug extraction. Adv. Drug Delivery Rev. 1997, 27 (2-3), 99-127.
    • (1997) Adv. Drug Delivery Rev. , vol.27 , Issue.2-3 , pp. 99-127
    • Shen, D.D.1    Kunze, K.L.2    Thummel, K.E.3
  • 33
    • 22944464763 scopus 로고    scopus 로고
    • Identification of esterases expressed in Caco-2 cells and effects of their hydrolyzing activity in predicting human intestinal absorption
    • Imai, T.; Imoto, M.; Sakamoto, H.; Hashimoto, M. Identification of esterases expressed in Caco-2 cells and effects of their hydrolyzing activity in predicting human intestinal absorption. Drug Metab. Dispos. 2005, 33 (8), 1185-90.
    • (2005) Drug Metab. Dispos. , vol.33 , Issue.8 , pp. 1185-1190
    • Imai, T.1    Imoto, M.2    Sakamoto, H.3    Hashimoto, M.4


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