Microemulsion based topical hydrogel of sertaconazole: Formulation, characterization and evaluation

Colloids and Surfaces B: Biointerfaces

Volumn 120, Issue , 2014, Pages 193-199

  Sahoo, Susijit ^a   Pani, Nihar Ranjan ^a   Sahoo, Sunit Kumar ^b  

^a Gayatri College of Pharmacy   (India)

^b UTKAL UNIVERSITY   (India)

Author keywords

Antifungal effect; Hydrogel; Microemulsion; Sertaconazole

Indexed keywords

HYDROGELS; OLEIC ACID; POLYOLS;

ANTIFUNGAL EFFECT; ENHANCING EFFECT; FUNGAL INFECTION; PROPYLENE GLYCOLS; PSEUDOTERNARY PHASE DIAGRAMS; SERTACONAZOLE; SKIN SENSITIVITY; ZONE OF INHIBITIONS;

MICROEMULSIONS;

CARBOPOL 940; OLEIC ACID; POLYSORBATE 80; PROPYLENE GLYCOL; SERTACONAZOLE; WATER; ANTIFUNGAL AGENT; EMULSION; HYDROGEL; IMIDAZOLE DERIVATIVE; SURFACTANT; THIOPHENE DERIVATIVE;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ANTIFUNGAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; CREAM; DRUG DELIVERY SYSTEM; DRUG DETERMINATION; DRUG EFFECT; DRUG FORMULATION; DRUG SCREENING; DRUG STABILITY; EX VIVO STUDY; GROWTH INHIBITION; HYDROGEL; MALE; MICROEMULSION; MOUSE; NONHUMAN; PH MEASUREMENT; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; RABBIT; REFRACTION INDEX; SKIN PERMEABILITY; SKIN SENSITIVITY; VISCOSITY; ANIMAL; CHEMISTRY; DRUG EFFECTS; EMULSION; IN VITRO STUDY; MEDICINAL CHEMISTRY; MICROBIAL SENSITIVITY TEST; PERMEABILITY; PHASE TRANSITION; TOPICAL DRUG ADMINISTRATION;

ADMINISTRATION, TOPICAL; ANIMALS; ANTIFUNGAL AGENTS; CANDIDA ALBICANS; CHEMISTRY, PHARMACEUTICAL; EMULSIONS; HYDROGEL; IMIDAZOLES; IN VITRO TECHNIQUES; MALE; MICE; MICROBIAL SENSITIVITY TESTS; PERMEABILITY; PHASE TRANSITION; RABBITS; SURFACE-ACTIVE AGENTS; THIOPHENES;

EID: 84904695244     PISSN: 09277765     EISSN: 18734367     Source Type: Journal    
DOI: 10.1016/j.colsurfb.2014.05.022     Document Type: Article

References (36)

1. Kreilgaard M. Influence of microemulsions on cutaneous drug delivery. Adv. Drug Deliv. Rev. 2002, 54:77-98.
2. Lawrence M.J., Rees G.D. Microemulsion-based media as novel drug delivery systems. Adv. Drug Deliv. Rev. 2000, 45:89-121.
3. Mohammed C., Manoj V., Aerosol-OT Microemulsions as transdermal carriers of tatracaine hydrochloride. Drug Dev. Ind. Pharm. 2000, 26:507-512.
4. Baroli B., Lopez-Quintela M.A., Delgado-Charro M.B., Fadda A.M., Blanco-Mendez J. Microemulsions for topical delivery of 8-methoxsalen. J. Control. Release 2000, 69:209-218.
5. Rhee Y.S., Choi J.G., Park E.S., Chi S.C. Transdermal delivery of ketoprofen using microemulsions. Int. J. Pharm. 2001, 228:161-170.
6. Kreilgaard M., Pedersen E.J., Jaroszewski J.W. NMR characterisation and transdermal drug delivery potential of microemulsion systems. Control. Release 2000, 69:421-433.
7. Baboota S., Al-Azaki A., Kohl K., Ali J., Dixit N., Shakeel F. Development and evaluation of a microemulsion formulation for transdermal delivery of terbinafine PDA. J. Pharm. Sci. Technol. 2007, 61:276-285.
8. Kamal M.A., Iimura N., Nabekura T., Kitagawa S. Enhanced skin permeation of diclofenac by ion-pair formation and further enhancement by microemulsion. Chem. Pharm. Bull. 2007, 55:368-371.
9. Fan Y., Ma L., Zhang W., Xu Y., Suolangzhaxi, Zhi X., Cui E., Song X. Microemulsion can improve the immune-enhancing activity of propolis flavonoid on immunosuppression and immune response. Int. J. Biol. Macromol. 2014, 63:126-132.
10. Zhao X., Liu J.P., Zhang X., Li Y. Enhancement of transdermal delivery of theophylline using microemulsion vehicle. Int. J. Pharm. 2006, 327:58-64.
11. Paolino D., Ventura C.A., Nisti S., Puglisi G., Fresta M. Lecithin microemulsion for the topical administration of ketoprofen: percutaneous adsorption through human skin and in vivo human skin tolerability. Int. J. Pharm. 2002, 244:21-31.
12. Delgado-Charro M.B., Iglesias-Vilas G., Blanco-Ménde J., López-Quintela M.A., Marty J.P., Guy R.H. Delivery of a hydrophilic solute through the skin from novel microemulsion systems. Eur. J. Pharm. Biopharm. 1997, 43:37-42.
13. Das B., Nayak A.K., Nanda U. Topical gels of lidocaine HCl using cashew gum and Carbopol 940: preparation and in vitro skin permeation. Int. J. Biol. Macromol. 2013, 62:514-517.
14. Carnali J.O., Naser M.S. The use of dilute solution viscometry to characterize the network properties of carbopol microgels. Colloids Polym. Sci. 1992, 270:183-193.
15. Carrillo-Muñoz A.J., Giusiano G., Ezkurra P.A., Quindós G. Sertaconazole: updated review of a topical antifungal agent. Expert Rev. Anticancer 2005, 3:333-342.
16. Hilton J., Woollen B.H., Scott R.C., Auton T.R., Trbilcock K.L., Wilks M.F. Vehicles effect on in-vitro percutaneous absorption through mice and human skin. Pharm. Res. 1994, 11:396-1400.
17. Patel A., Patel J. Design development and in vitro evaluation of sertaconazole mucoadhesive vaginal tablet. Der Pharmacia Lettre 2012, 4:418-427.
18. Zhu W., Yu A., Wang W., Dong R., Wu W., Zhai G. Formulation design of microemulsion for dermal delivery of penciclovir. Int. J. Pharm. 2008, 360:184-190.
19. Zhu W., Guo C., Yu A., Gao Y., Cao F., Zhai G. Microemulsion-based hydrogel formulation of penciclovir for topical delivery. Int. J. Pharm. 2009, 378:152-215.
20. Chen H., Mou D., Du D., Chang X., Zhu D., Liu J., Xu H., Yang X. Hydrogel-thickened microemulsion for topical administration of drug molecule at an extremely low concentration. Int. J. Pharm. 2007, 341:78-84.
21. Valenta C., Schultz K. Influence of carrageenan on the rheology and skin permeation of microemulsion formulations. J. Control. Release 2004, 95:257-265.
22. Peltola S., Saarinen-Savolainen P., Kiesvaara J., Suhonen T.M., Urtti A. Microemulsions for topical delivery of estradiol. Int. J. Pharm. 2003, 254:99-107.
23. Geoffroy J.M., Fredrickson J.K., Shelton J.T. A mixture experiment approach for controlling the dissolution rate of a sustained-release tablet. Drug Dev. Ind. Pharm. 1998, 24:799-806.
24. Hamed E., Sakr A. Application of multiple response optimization technique to extended release formulation design. J. Control. Release 2001, 73:329-338.
25. Korsmeyer R.W., Doelker G.E.P., Peppas N.A. Mechanisms of potassium chloride from compressed, hydrophilic, polymeric matrices: effect of entrapped air. J. Pharm. Sci. 1983, 72:1189Y1191.
26. Draize J., Woodard G., Calvery H. Methods for the study of irritation and toxicity of substances topically applied to skin and mucous membranes. J. Pharmacol. Exp. Ther. 1944, 82:377-390.
27. Osborne D.W., Ward A.J., O'Neill K.J. Microemulsions as topical drug delivery vehicles: in-vitro transdermal studies of a model hydrophilic drug. J. Pharm. Pharmacol. 1991, 43:450-454.
28. Richardson S.E., Bannatyne R.M., Summerbell R.C., Milliken J., Gold R., Weitzman S.S. Disseminated fusarial infection in the immunocompromised host. Rev. Infect. Dis. 1988, 10:1171-1181.
29. Jain G.K., Sharma A., Agrawal S. Transdermal controlled administration of verapamil-enhancement of skin permeability. Int. J. Pharm. 1996, 130:169-177.
30. Dreher F., Walde P., Luisi P., Elsner P. Human skin irritation studies of a lecithin microemulsion gel and of lecithin liposomes. Skin Pharmacol. 1996, 9:124-129.
31. Paolino D., Ventura C.A., Nistico S., Puglisi G., Fresta M. Lecithin microemulsions for the topical administration of ketoprofen: percutaneous adsorption through human skin and in vivo human skin tolerability. Int. J. Pharm. 2002, 244:21-31.
32. Butani D., Yewale C., Misra A. Amphotericin B topical microemulsion: formulation, characterization and evaluation. Colloids Surf. B: Biointerfaces 2014, 10.1016/j.colsurfb.2014.01.014.
33. Alam M.A., Ahmad F.J., Khan Z.I., Khar R.K., Ali M. Development and evaluation of acidbuffering bioadhesive vaginal tablet for mixed vaginal infections. AAPS PharmSciTech 2007, 8(4). Article 109.
34. Kogan A., Garti N. Microemulsions as transdermal drug delivery vehicles. Adv. Colloid Interface Sci. 2006, 123-126:369-385.
35. Li L., Nandi I., Kim K.H. Development of an ethyl laurate based microemulsion for rapid-onset intranasal delivery of diazepam. Int. J. Pharm. 2002, 237:77-85.
36. Chen H.B., Chang X.L., Du D.R., Li J., Xu H.B., Yang X.L. Microemulsion based hydrogel formulation of ibuprofen for topical delivery. Int. J. Pharm. 2006, 315:52-58.