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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 14, 2014, Pages 3100-3103

Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120)

(18) Sparks, Steven M a Chen, Grace a Collins, Jon L a Danger, Dana a Dock, Steven T a Jayawickreme, Channa a Jenkinson, Stephen a Laudeman, Christopher a Leesnitzer, M Anthony a Liang, Xi a Maloney, Patrick a McCoy, David C a Moncol, David a Rash, Vincent a Rimele, Thomas a Vulimiri, Padmaja a Way, James M a Ross, Sean a

a GLAXOSMITHKLINE (United States)

Author keywords

FFA4; Free fatty acid receptor 4; Free fatty acid receptor 4 agonist; Free fatty acid receptor 4 antagonist; GPR120

Indexed keywords

ANTIDIABETIC AGENT; DIARYLSULFONAMIDE DERIVATIVE; FATTY ACID; FREE FATTY ACID RECEPTOR 4; G PROTEIN COUPLED RECEPTOR 120; GLIBENCLAMIDE; GLUCOSE; INSULIN; LINOLEIC ACID; SULFONAMIDE; UNCLASSIFIED DRUG; ANILINE; FREE FATTY ACID RECEPTOR 4 AGONIST; GSK 137647A; G PROTEIN COUPLED RECEPTOR; O3FAR1 PROTEIN, HUMAN;

AGONIST; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG IDENTIFICATION; DRUG STRUCTURE; GENE EXPRESSION; HUMAN; HUMAN CELL; IN VITRO STUDY; INSULIN RELEASE; INSULINOMA CELL LINE; MOUSE; NONHUMAN; ROOM TEMPERATURE; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SYNTHESIS; HEK293 CELL LINE; SUBSTITUTION REACTION; AGONISTS; ANIMAL; CELL LINE; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ANIMALS; CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; HEK293 CELLS; HUMANS; INSULIN; MICE; MOLECULAR STRUCTURE; RECEPTORS, G-PROTEIN-COUPLED; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 84902544474 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.05.012 Document Type: Article

Times cited : (96)

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