Microwave-Assisted synthesis of novel 1,2,3-triazole derivatives and their antimicrobial activity

Medicinal Chemistry Research

Volumn 23, Issue 6, 2014, Pages 3005-3018

  Ashok, D ^a   Mohan Gandhi, D ^a   Srinivas, G ^a   Vikas Kumar, A ^a  

^a OSMANIA UNIVERSITY   (India)

Author keywords

1 2 3 Triazoles; Antimicrobial activity; Click chemistry; Microwave irradiation

Indexed keywords

1,2,3 TRIAZOLE DERIVATIVE; ALKYNE DERIVATIVE; AZIDE; COPPER DERIVATIVE;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; CATALYSIS; CATALYST; CYCLOADDITION; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; MICROWAVE ASSISTED SYNTHESIS; MICROWAVE IRRADIATION; PURIFICATION;

EID: 84898888852     PISSN: 10542523     EISSN: 15548120     Source Type: Journal    
DOI: 10.1007/s00044-013-0880-1     Document Type: Article

References (19)

1. Alvarez R, Velazquez S, San-Felix A, Aquaro S, De Clercq E, Perno CF, Karlsson A, Balzarini J, Camarasa MJ (1994) 1,2,3-Triazole-[2,5-bis-O(tertbutyl dimethylsilyl)-β-d-ribofuranosyl]-3-spiro-5-(4-Amino-l,2-oxathiole2, 2-dioxide) (TSAO) Analogues: Synthesis and Anti-HIV-1 Activity. J Med Chem 37:4185-4194.
2. Anto RJ, Sukumaran K, Kuttan G, Rao MNA, Subbaraju V, Kuttan R (1995) Anticancer and antioxidant activity of synthetic chalcones and related compounds. Cancer Lett 97:33-37
3. Ashok D, Shravani D (2008) One-pot synthesis of novel spiro 2,3,7,8-tetrahydro-benzo[1,2-b:5,4-b']-dipyran-4,6-dione and 2,3,8,9-tetrahydro-benzo[1,2-b:4,3-b']dipyran-4,10-dione derivatives. Tetrahedron Lett 49:7227-7229
4. Ashok D, Sudershan K, Khalilullah M (2012) Solvent-free microwave-Assisted synthesis of E-(1)-(6-benzoyl 3,5dimethylfuro [3',2':4,5]benzo[b]furan-2-yl)3-(aryl)-2-propen-1-ones and their antibacterial activity. Green Chem Lett Rev 5(2):121-125. doi: 10.1080/17518253.2011.584912
5. Bergmann R, Gericke R (1990) Synthesis and antihypertensive activity of 4-(1,2-dihydro-2-oxo-1-pyridyl)-2H-1-benzopyrans and related compounds, new potassium channel activators. J Med Chem 33:492-504
6. Burrell G, Cassidy F, Evans JM, Ightowler D, Stemo G (1990) Variation in the aromatic ring of cromakalim: antihypertensive activity of pyranopyridines and 6-Alkyl-2H-1-benzopyans. J Med Chem 33:3023-3027
7. Chen H, Zuo S, Wang X, Tang X, Zhao M, Lu Y, Chen L, Liu J, Liu Y, Liu D, Zhang S, Li T (2011) Synthesis of 4b-triazole-podophyllotoxin derivatives by azide-Alkyne cycloaddition and biological evaluation as potential antitumor agents. Eur J Med Chem 46:1714-4709
8. Demaray JA, Thuener JE, Dawson MN, Sucheck SJ (2008) Synthesis of triazole-oxazolidinones via a one-pot reaction and evaluations of their antimicrobial activity. Bioorg Med Chem Lett 18:4868-4871
9. Gericke R, Harting J, Lues I, Schittenhelm C (1991) 3-Methyl-2H-1- benzopyran potassium channel activators. J Med Chem 34:3074-3085
10. Hsieh HK, Tsao LT, Wang JP, Lin CN (2000) Synthesis and anti-inflammatory effect of chalcones. J Pharm Pharmacol 52(2):163-171
11. Kalena GP, Jain A, Banerji A (1997) Amberlyst 15 Catalyzed prenylation of phenols: one-step synthesis of benzopyrans. Molecules 2(7):100-105. doi: 10.3390/20700100
12. Khan I, Ali S, Hameed S, Rama NH, Hussain MT, Wadood A, Ul-Haq Z, Khan A, Ali S, Choudhary MI (2010) Synthesis, antioxidant activities and urease inhibition of some new 1,2,4-triazole and 1,3,4-thiadiazole derivatives. Euro J Med Chem 45:5200-5207
13. Lazrek HB, Taourirte M, Oulih Barascut JL, Imbach JL, Pannecouqe C, Witrouw M, Clercq ED (2001) Synthesis and Anti-HIV activity of new modified 1,2,3-triazole acyclonucleosides. Nucleosides, Nucleotides Nucleic Acids 20:1949-1960
14. Mukherjee S, Kumar V, Prasad AK, Raj HG, Bracke ME, Olsen CE, Jain SC, Parmar VS (2001) Synthetic biological activity evolution studies on Novel 1,3-diarylpropanones. Bioorg Med Chem 9:337-345
15. Ram VJ, Saxena AS, Srivastava S, Chandra S (2000) Oxygenated chalcones and bischalcones as potential antimalarial agents. Bioorg Med Chem Lett 10:2159-2161
16. Ray S, Grover PK, Kamboj VP, Setty BS, Kar AB, Anand N (1976) Antifertility agents. 12. Structure-Activity relationship of 3,4-diphenylchromenes and chromans. J Med Chem 19:276-279. doi: 10.1021/jm00224a014
17. Revol-Junelles A-M, Mathis R, Krier F, Delfour A, Lefebvre G (1996) Leuconostoc mesenteroides subsp. mesenteroides FR52 synthesizes two distinct bacteriocins. Lett Appl Microbiol 23:120-124
18. Satyanarayana M, Tiwari P, Tripathi BK, Srivastava AK, Pratap R (2004) Synthesis and antiperglycemic activity of chalcone based aryloxypropanolamines. Bioorg Med Chem 12:883-889
19. Zhai L, Chen M, Blam J, Theander TG, Chiristensen SB, Kharazmi A (1999) The antileishmanial activity of novel oxygenated chalcones and their mechanism of action. J Antimicrob Chemother 43:793-803