Solid phospholipid nano-particles: Investigations into formulation and dissolution properties of griseofulvin

International Journal of Pharmaceutics

Volumn 467, Issue 1-2, 2014, Pages 42-47

  Brinkmann Trettenes, Ulla ^a   Bauer Brandl, Annette ^a  

^a UNIVERSITY OF SOUTHERN DENMARK   (Denmark)

Author keywords

Bio relevant media; B chi B 90; FaSSIF; Griseofulvin; Pancreatin; Spray drying

Indexed keywords

ALCOHOL; EXCIPIENT; GRISEOFULVIN; NANOPARTICLE; PANCREATIN; PHOSPHATE BUFFERED SALINE; PHOSPHOLIPID; WATER; BUFFER; DRUG CARRIER;

AEROSOL; ARTICLE; CONTROLLED STUDY; DRUG FORMULATION; DRUG SOLUBILITY; PRIORITY JOURNAL; SOLID STATE; SPRAY DRYING; CHEMISTRY; COMPARATIVE STUDY; INTESTINAL SECRETIONS; KINETICS; MEDICINAL CHEMISTRY; NANOTECHNOLOGY; PH; PHARMACEUTICS; PROCEDURES; SOLUBILITY;

BUFFERS; CHEMISTRY, PHARMACEUTICAL; DRUG CARRIERS; EXCIPIENTS; GRISEOFULVIN; HYDROGEN-ION CONCENTRATION; INTESTINAL SECRETIONS; KINETICS; NANOPARTICLES; NANOTECHNOLOGY; PANCREATIN; PHOSPHOLIPIDS; SOLUBILITY; TECHNOLOGY, PHARMACEUTICAL;

EID: 84898420206     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2014.03.023     Document Type: Article

References (20)

1. A. Balakrishnan, B.D. Rege, G.L. Amidon, and J.E. Polli Surfactant-mediated dissolution: contributions of solubility enhancement and relatively low micelle diffusivity Journal of Pharmaceutical Sciences 93 2004 2064 2075 (Pubitemid 39045487)
2. 31P NMR Journal of Pharmaceutical and Biomedical Analysis 70 2012 708 712
3. U. Brinkmann-Trettenes, S. Barnert, and A. Bauer-Brandl Single step bottom-up process to generate solid phospholipid nano-particles Pharmaceutical Development and Technology 19 2014 326 332
4. J.M. Butler, and J.B. Dressman The developability classification system: application of biopharmaceutics concepts to formulation development Journal of Pharmaceutical Sciences 99 2010 4940 4954
5. J.H. De Smidt, J.C. Offringa, and D.J. Crommelin Dissolution rate of griseofulvin in bile salt solutions Journal of Pharmaceutical Sciences 80 1991 399 401
6. P.H. Elworthy, and F.J. Lipscomb A note on the solubility of griseofulvin Journal of Pharmacy and Pharmacology 20 1968 790 792
7. J.H. Fagerberg, Y. Al-Tikriti, G. Ragnarsson, and C.A.S. Bergström Ethanol effects on apparent solubility of poorly soluble drugs in simulated intestinal fluid Molecular Pharmaceutics 9 2012 1942 1952
8. K.J. Frank, K.M. Rosenblatt, U. Westedt, P. Hölig, J. Rosenberg, M. Mägerlein, G. Fricker, and M. Brandl Amorphous solid dispersion enhances permeation of poorly soluble ABT-102: true supersaturation vs. apparent solubility enhancement International Journal of Pharmaceutics 437 2012 288 293
9. E. Galia, D. Nicolaides, D. Horter, R. Lobenberg, C. Reppas, and J.B. Dressman Evaluation of various dissolution media for predicting in vivo performance of class I and II drugs Pharmaceutical Research 15 1998 698 705 (Pubitemid 28275645)
10. B. Kloefer, P. Van Hoogevest, R. Moloney, M. Kuentz, M.L.S. Leigh, and J. Dressman Study of a standardized taurocholate-lecithin powder for preparing the biorelevant media FeSSIF and FaSSIF Dissolution Technologies 17 2010 6 13
11. W. Liu, A. Ye, C. Liu, W. Liu, and H. Singh Structure and integrity of liposomes prepared from milk- or soybean-derived phospholipids during in vitro digestion Food Research International 48 2012 499 506
12. V.M. Rao, M. Lin, C.K. Larive, and M.Z. Southard A mechanistic study of griseofulvin dissolution into surfactant solutions under laminar flow conditions Journal of Pharmaceutical Sciences 86 1997 1132 1137 (Pubitemid 27430918)
13. M. Schaefer-Korting, H.C. Korting, and E. Mutschler Human plasma and skin blister fluid levels of griseofulvin following a single oral dose European Journal of Clinical Pharmacology 29 1985 109 113 (Pubitemid 15232086)
14. H.J. Schwebel, P. van Hoogevest, M.L.S. Leigh, and M. Kuentz The apparent solubilizing capacity of simulated intestinal fluids for poorly water-soluble drugs Pharmaceutical Development and Technology 16 2011 278 286
15. S. Shanmugam, R. Baskaran, P. Balakrishnan, P. Thapa, C.S. Yong, and B.K. Yoo Solid self-nanoemulsifying drug delivery system (S-SNEDDS) containing phospatidylcholine for enhanced bioavailability of highly lipophilic bioactive carotenoid lutein European Journal of Pharmaceutics and Biopharmaceutics 79 2011 250 257
16. The Directorate for the Quality of Medicines & Healthcare of the Council of Europe, 2012. European Pharmacopoeia, 7th ed. Council of Europe, Strasbourg Cedex.
17. M. Thommes, D.R. Ely, M.T. Carvajal, and R. Pinal Improvement of the dissolution rate of poorly soluble drugs by solid crystal suspensions Molecular Pharmaceutics 8 2011 727 735
18. 31P NMR, electron microscopy and permeability studies Biochimica et Biophysica Acta (BBA) - Biomembranes 649 1981 211 220
19. C.-Y. Wu, and L.Z. Benet Predicting drug disposition via application of BCS: transport/absorption/elimination interplay and development of a biopharmaceutics drug disposition classification system Pharmaceutical Research 22 2005 11 23 (Pubitemid 40558141)
20. N.M. Zaki, P. Artursson, and C.A.S. Bergström A modified physiological BCS for prediction of intestinal absorption in drug discovery Molecular Pharmacology 7 2010 1478 1487