메뉴 건너뛰기




Volumn 21, Issue 3, 2014, Pages 325-329

Effect of DA-8031, a novel oral compound for premature ejaculation, on male rat sexual behavior

Author keywords

Animals; DA 8031; Premature ejaculation; Sexual behavior

Indexed keywords

AGENTS ACTING ON THE GENITAL SYSTEM; DA 8031; ISOBENZOFURAN DERIVATIVE; SEROTONIN TRANSPORTER; UNCLASSIFIED DRUG;

EID: 84896711891     PISSN: 09198172     EISSN: 14422042     Source Type: Journal    
DOI: 10.1111/iju.12256     Document Type: Article
Times cited : (12)

References (30)
  • 1
    • 0033540646 scopus 로고    scopus 로고
    • Sexual dysfunction in the United States: prevalence and predictors
    • Laumann EO, Paik A, Resen RC. Sexual dysfunction in the United States: prevalence and predictors. JAMA 1999; 281: 537-544.
    • (1999) JAMA , vol.281 , pp. 537-544
    • Laumann, E.O.1    Paik, A.2    Resen, R.C.3
  • 2
    • 14544281524 scopus 로고    scopus 로고
    • Sexual problems among women and men aged 40-80 y: prevalence and correlates identified in the Global Study of Sexual Attitudes and Behaviors
    • Laumann EO, Nicolosi A, Glasser DB etal. Sexual problems among women and men aged 40-80 y: prevalence and correlates identified in the Global Study of Sexual Attitudes and Behaviors. Int. J. Impot. Res. 2005; 17: 39-57.
    • (2005) Int. J. Impot. Res. , vol.17 , pp. 39-57
    • Laumann, E.O.1    Nicolosi, A.2    Glasser, D.B.3
  • 3
    • 33646008605 scopus 로고    scopus 로고
    • Premature ejaculation: the most common male sexual dysfunction
    • Hellstrom WJG, Nehra A, Shabsigh R, Sharlip ID. Premature ejaculation: the most common male sexual dysfunction. J. Sex. Med. 2006; 3 (S1): 1-3.
    • (2006) J. Sex. Med. , vol.3 , Issue.S1 , pp. 1-3
    • Hellstrom, W.J.G.1    Nehra, A.2    Shabsigh, R.3    Sharlip, I.D.4
  • 4
    • 5044248352 scopus 로고    scopus 로고
    • Utility of selective serotonin reuptake inhibitors in premature ejaculation
    • Waldinger MD, Oliver B. Utility of selective serotonin reuptake inhibitors in premature ejaculation. Curr. Opin. Investig. Drugs 2004; 5: 743-747.
    • (2004) Curr. Opin. Investig. Drugs , vol.5 , pp. 743-747
    • Waldinger, M.D.1    Oliver, B.2
  • 5
    • 16344386416 scopus 로고    scopus 로고
    • On-demand SSRI treatment of premature ejaculation: pharmacodynamic limitations for relevant ejaculation delay and consequent solutions
    • Waldinger MD, Schweitzer DH, Olivier B. On-demand SSRI treatment of premature ejaculation: pharmacodynamic limitations for relevant ejaculation delay and consequent solutions. J. Sex. Med. 2005; 2: 121-131.
    • (2005) J. Sex. Med. , vol.2 , pp. 121-131
    • Waldinger, M.D.1    Schweitzer, D.H.2    Olivier, B.3
  • 6
    • 84871872718 scopus 로고    scopus 로고
    • Dapoxetine: a new option in the medical management of premature ejaculation
    • McMahon CG. Dapoxetine: a new option in the medical management of premature ejaculation. Ther. Adv. Urol. 2012; 4: 233-251.
    • (2012) Ther. Adv. Urol. , vol.4 , pp. 233-251
    • McMahon, C.G.1
  • 7
    • 0036893805 scopus 로고    scopus 로고
    • The neurobiological approach to premature ejaculation
    • Waldinger MD. The neurobiological approach to premature ejaculation. J. Urol. 2002; 168: 2359-2367.
    • (2002) J. Urol. , vol.168 , pp. 2359-2367
    • Waldinger, M.D.1
  • 8
    • 33947309885 scopus 로고    scopus 로고
    • Premature ejaculation: definition and drug treatment
    • Waldinger MD. Premature ejaculation: definition and drug treatment. Drugs 2007; 67: 547-568.
    • (2007) Drugs , vol.67 , pp. 547-568
    • Waldinger, M.D.1
  • 9
    • 3242773768 scopus 로고    scopus 로고
    • AUA guideline on the pharmacological management of premature ejaculation
    • Montague D, Jarow J, Broderick G etal. AUA guideline on the pharmacological management of premature ejaculation. J. Urol. 2004; 172: 290-294.
    • (2004) J. Urol. , vol.172 , pp. 290-294
    • Montague, D.1    Jarow, J.2    Broderick, G.3
  • 10
    • 0344110152 scopus 로고    scopus 로고
    • Pharmacokinetics of selective serotonin reuptake inhibitors
    • Hiemke C, Hartter S. Pharmacokinetics of selective serotonin reuptake inhibitors. Pharmacol. Ther. 2000; 85: 11-28.
    • (2000) Pharmacol. Ther. , vol.85 , pp. 11-28
    • Hiemke, C.1    Hartter, S.2
  • 11
    • 32944463634 scopus 로고    scopus 로고
    • Single- and multiple-dose pharmacokinetics of dapoxetine hydrochloride, a novel agent for the treatment of premature ejaculation
    • Modi NB, Dresser MJ, Simon M, Lin D, Desai D, Gupta S. Single- and multiple-dose pharmacokinetics of dapoxetine hydrochloride, a novel agent for the treatment of premature ejaculation. J. Clin. Pharmacol. 2006; 46: 301-309.
    • (2006) J. Clin. Pharmacol. , vol.46 , pp. 301-309
    • Modi, N.B.1    Dresser, M.J.2    Simon, M.3    Lin, D.4    Desai, D.5    Gupta, S.6
  • 12
    • 77953648907 scopus 로고    scopus 로고
    • Pharmacokinetics of dapoxetine hydrochloride in healthy Chinese, Japanese, and Caucasian men
    • Thyssen A, Sharma O, Tianmei S etal. Pharmacokinetics of dapoxetine hydrochloride in healthy Chinese, Japanese, and Caucasian men. J. Clin. Pharmacol. 2010; 50: 1450-1460.
    • (2010) J. Clin. Pharmacol. , vol.50 , pp. 1450-1460
    • Thyssen, A.1    Sharma, O.2    Tianmei, S.3
  • 13
    • 60249103913 scopus 로고    scopus 로고
    • Dapoxetine for the treatment of premature ejaculation: results from a randomized, double-blind, placebo-controlled phase 3 trial in 22 countries
    • Buvat J, Tesfaye F, Rothman M, Rivas DA, Giuliano F. Dapoxetine for the treatment of premature ejaculation: results from a randomized, double-blind, placebo-controlled phase 3 trial in 22 countries. Eur. Urol. 2009; 55: 957-967.
    • (2009) Eur. Urol. , vol.55 , pp. 957-967
    • Buvat, J.1    Tesfaye, F.2    Rothman, M.3    Rivas, D.A.4    Giuliano, F.5
  • 14
    • 84870414526 scopus 로고    scopus 로고
    • Dapoxetine: an evidence-based review of its effectiveness in treatment of premature ejaculation
    • McCarty E, Dinsmore W. Dapoxetine: an evidence-based review of its effectiveness in treatment of premature ejaculation. Core. Evid. 2012; 7: 1-14.
    • (2012) Core. Evid. , vol.7 , pp. 1-14
    • McCarty, E.1    Dinsmore, W.2
  • 15
    • 79953156439 scopus 로고    scopus 로고
    • Cardiovascular safety profile of dapoxetine during the premarketing evaluation
    • Kowey PR, Mudumbi RV, Aquilina JW, DiBattiste PM. Cardiovascular safety profile of dapoxetine during the premarketing evaluation. Drugs R. D. 2011; 11: 1-11.
    • (2011) Drugs R. D. , vol.11 , pp. 1-11
    • Kowey, P.R.1    Mudumbi, R.V.2    Aquilina, J.W.3    DiBattiste, P.M.4
  • 16
    • 74049146657 scopus 로고    scopus 로고
    • The effects of oral administration of d-modafinil on male rat ejaculatory behavior
    • Marson L, Yu G, Farber NM. The effects of oral administration of d-modafinil on male rat ejaculatory behavior. J. Sex. Med. 2010; 7: 70-78.
    • (2010) J. Sex. Med. , vol.7 , pp. 70-78
    • Marson, L.1    Yu, G.2    Farber, N.M.3
  • 17
    • 84866683764 scopus 로고    scopus 로고
    • Effect of dexmedetomidine on ejaculatory behavior and sexual motivation in intact male rats
    • Snoeren EM, Lehtimäki J, Agmo A. Effect of dexmedetomidine on ejaculatory behavior and sexual motivation in intact male rats. Pharmacol. Biochem. Behav. 2012; 103: 345-352.
    • (2012) Pharmacol. Biochem. Behav. , vol.103 , pp. 345-352
    • Snoeren, E.M.1    Lehtimäki, J.2    Agmo, A.3
  • 18
    • 79953899827 scopus 로고    scopus 로고
    • Candidate molecule for premature ejaculation, DA-8031: in vivo and in vitro characterization of DA-8031
    • Jeon HJ, Kim HS, Lee CH etal. Candidate molecule for premature ejaculation, DA-8031: in vivo and in vitro characterization of DA-8031. Urology 2011; 77: e17-21.
    • (2011) Urology , vol.77
    • Jeon, H.J.1    Kim, H.S.2    Lee, C.H.3
  • 19
    • 84875516548 scopus 로고    scopus 로고
    • Ejaculatory responses are inhibited by a new chemical entity, DA-8031, in pre-clinical rodent models of ejaculation
    • Kang KK, Ahn GJ, Sung HJ, Kim SH, Kim H, Lee S. Ejaculatory responses are inhibited by a new chemical entity, DA-8031, in pre-clinical rodent models of ejaculation. Urology 2013; 81: e13-18.
    • (2013) Urology , vol.81
    • Kang, K.K.1    Ahn, G.J.2    Sung, H.J.3    Kim, S.H.4    Kim, H.5    Lee, S.6
  • 20
    • 0032216268 scopus 로고    scopus 로고
    • An optimized approach for the assessment of sexual behavior in male rats
    • Chahoud I, Faqi AS. An optimized approach for the assessment of sexual behavior in male rats. Reprod. Toxicol. 1998; 12: 667-671.
    • (1998) Reprod. Toxicol. , vol.12 , pp. 667-671
    • Chahoud, I.1    Faqi, A.S.2
  • 21
    • 0345515992 scopus 로고    scopus 로고
    • Male rat sexual behavior
    • Agmo A. Male rat sexual behavior. Brain. Res. Protoc. 1997; 1: 203-209.
    • (1997) Brain. Res. Protoc. , vol.1 , pp. 203-209
    • Agmo, A.1
  • 23
    • 22144434171 scopus 로고    scopus 로고
    • Animal models of premature and retarded ejaculation
    • Waldinger MD, Olivier B. Animal models of premature and retarded ejaculation. World J. Urol. 2005; 23: 115-118.
    • (2005) World J. Urol. , vol.23 , pp. 115-118
    • Waldinger, M.D.1    Olivier, B.2
  • 24
    • 0032971206 scopus 로고    scopus 로고
    • A comparison of the effects of different serotonin reuptake blockers on sexual behaviour of the male rat
    • Mos J, Mollet I, Tolboom JT, Waldinger MD, Olivier B. A comparison of the effects of different serotonin reuptake blockers on sexual behaviour of the male rat. Eur. Neuropsychopharmacol. 1999; 9: 123-135.
    • (1999) Eur. Neuropsychopharmacol. , vol.9 , pp. 123-135
    • Mos, J.1    Mollet, I.2    Tolboom, J.T.3    Waldinger, M.D.4    Olivier, B.5
  • 25
    • 33947161531 scopus 로고    scopus 로고
    • Acute and chronic dosing of Lepidium meyenii (Maca) on male rat sexual behavior
    • Lentz A, Gravitt K, Carson CC, Marson L. Acute and chronic dosing of Lepidium meyenii (Maca) on male rat sexual behavior. J. Sex. Med. 2007; 4: 332-339.
    • (2007) J. Sex. Med. , vol.4 , pp. 332-339
    • Lentz, A.1    Gravitt, K.2    Carson, C.C.3    Marson, L.4
  • 26
    • 74049084296 scopus 로고    scopus 로고
    • Actions of dapoxetine on ejaculation and sexual behavior in rats
    • Gengo P, Marson L, Gravitt K. Actions of dapoxetine on ejaculation and sexual behavior in rats. J. Sex. Med. 2006; 3 (S3): 200.
    • (2006) J. Sex. Med. , vol.3 , Issue.S3 , pp. 200
    • Gengo, P.1    Marson, L.2    Gravitt, K.3
  • 27
    • 23944456497 scopus 로고    scopus 로고
    • Effects of chronic selective serotonin reuptake inhibitors on 8-OH-DPAT induced facilitation of ejaculation in rats: comparison of fluvoxamine and paroxetine
    • de Jong TR, Pattij T, Veening JG, Waldinger MD, Cools AR, Olivier B. Effects of chronic selective serotonin reuptake inhibitors on 8-OH-DPAT induced facilitation of ejaculation in rats: comparison of fluvoxamine and paroxetine. Psychopharmacology (Berl) 2005; 179: 509-515.
    • (2005) Psychopharmacology (Berl) , vol.179 , pp. 509-515
    • de Jong, T.R.1    Pattij, T.2    Veening, J.G.3    Waldinger, M.D.4    Cools, A.R.5    Olivier, B.6
  • 28
    • 0036119053 scopus 로고    scopus 로고
    • The selective serotonin re-uptake inhibitors fluvoxamine and paroxetine differ in sexual inhibitory effects after chronic treatment
    • Waldinger MD, van De Plas A, Pattij T etal. The selective serotonin re-uptake inhibitors fluvoxamine and paroxetine differ in sexual inhibitory effects after chronic treatment. Psychopharmacology (Berl) 2002; 160: 283-289.
    • (2002) Psychopharmacology (Berl) , vol.160 , pp. 283-289
    • Waldinger, M.D.1    van De Plas, A.2    Pattij, T.3
  • 29
    • 64149109693 scopus 로고    scopus 로고
    • Delay of ejaculation induced by SB-277011, a selective dopamine d3 receptor antagonist, in the rat
    • Clement P, Pozzato C, Heidbreder C, Alexandre L, Giuliano F, Melotto S. Delay of ejaculation induced by SB-277011, a selective dopamine d3 receptor antagonist, in the rat. J. Sex. Med. 2009; 6: 980-988.
    • (2009) J. Sex. Med. , vol.6 , pp. 980-988
    • Clement, P.1    Pozzato, C.2    Heidbreder, C.3    Alexandre, L.4    Giuliano, F.5    Melotto, S.6
  • 30
    • 23944456378 scopus 로고    scopus 로고
    • Individual differences in male rat ejaculatory behaviour: searching for models to study ejaculation disorders
    • Pattij T, de Jong TR, Uitterdijk A etal. Individual differences in male rat ejaculatory behaviour: searching for models to study ejaculation disorders. Eur. J. Neurosci. 2005; 22: 724-734.
    • (2005) Eur. J. Neurosci. , vol.22 , pp. 724-734
    • Pattij, T.1    de Jong, T.R.2    Uitterdijk, A.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.