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Volumn 75, Issue , 2014, Pages 96-105

Discovery of 2-methoxy-3-phenylsulfonamino-5-(quinazolin-6-yl or quinolin-6-yl)benzamides as novel PI3K inhibitors and anticancer agents by bioisostere

(10) Shao, Teng a Wang, Juan b Chen, Jian Gang a Wang, Xiao Meng a Li, Huan a Li, Yi Ping a Li, Yan a Yang, Guang De a Mei, Qi Bing b Zhang, San Qi a

a XI'AN JIAOTONG UNIVERSITY (China)

b SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (China)

Author keywords

Anticancer effect; Antiproliferative activity; Benzamide; Bioisostere; PI3K inhibitor; Quinazoline

Indexed keywords

ANTICANCER EFFECT; ANTIPROLIFERATIVE ACTIVITY; BENZAMIDE; BIOISOSTERE; PI3K INHIBITOR; QUINAZOLINE;

ANIMALS; ANTINEOPLASTIC AGENTS; BENZAMIDES; CELL LINE, TUMOR; CELL PROLIFERATION; HUMANS; MALE; MICE; MICE, INBRED BALB C; MICE, NUDE; NEOPLASMS; PHOSPHATIDYLINOSITOL 3-KINASES; QUINAZOLINES; SIGNAL TRANSDUCTION; TOR SERINE-THREONINE KINASES;

EID: 84893947635 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2014.01.053 Document Type: Article

Times cited : (43)

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