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Volumn 2013, Issue , 2013, Pages

In vitro permeation of micronized and nanonized alaptide from semisolid formulations

Author keywords

[No Author keywords available]

Indexed keywords

CYCLO(ALANINE (1 AMINO 1 CYCLOPENTANE)CARBONYL); CYCLO(ALANINE-(1-AMINO-1-CYCLOPENTANE)CARBONYL); CYCLOPEPTIDE; NANOPARTICLE; NEUROPEPTIDE;

EID: 84893847515     PISSN: None     EISSN: 1537744X     Source Type: Journal    
DOI: 10.1155/2013/787283     Document Type: Article
Times cited : (11)

References (45)
  • 1
    • 84893833257 scopus 로고    scopus 로고
    • Inventors; Cristalia Produtos Quimicos e Farmaceuticos, Ltd. assignee, "Pharmaceutical compositions of topic use, applied in treatment of skin and/or mucous injuries; use of compositions in treatment of skin and/or mucous injuries and use of compounds in treatment of skin and/or mucous injuries", WO 2002083086 A1, 2002
    • De Souza Russo E. M., Russo V. F. T.,. Inventors; Cristalia Produtos Quimicos e Farmaceuticos, Ltd., assignee, "Pharmaceutical compositions of topic use, applied in treatment of skin and/or mucous injuries; use of compositions in treatment of skin and/or mucous injuries and use of compounds in treatment of skin and/or mucous injuries" WO 2002083086 A1, 2002
    • De Souza Russo, E.M.1    Russo, V.F.T.2
  • 2
    • 84893821959 scopus 로고    scopus 로고
    • Inventors; Japan Science and Technology Corporation, assignee, "Skin tissue regeneration promoters comprising ginsenoside Rb1", EP1295893 A1, 2003
    • Hashimoto K., Nakata K., Sakanaka M., Tanaka J.,. Inventors; Japan Science and Technology Corporation, assignee, "Skin tissue regeneration promoters comprising ginsenoside Rb1" EP1295893 A1, 2003
    • Hashimoto, K.1    Nakata, K.2    Sakanaka, M.3    Tanaka, J.4
  • 3
    • 84875046809 scopus 로고    scopus 로고
    • Topical treatment of the buccal mucosa and wounded skin in rats with a triamcinolone acetonide-loaded hydrogel prepared using an electron beam
    • Choi S. G., Baek E. J., Davaa E., Topical treatment of the buccal mucosa and wounded skin in rats with a triamcinolone acetonide-loaded hydrogel prepared using an electron beam. International Journal of Pharmaceutics 2013 447 102 108
    • (2013) International Journal of Pharmaceutics , vol.447 , pp. 102-108
    • Choi, S.G.1    Baek, E.J.2    Davaa, E.3
  • 5
    • 0026508890 scopus 로고
    • Two-step generation of spirocyclic dipeptides from linear peptide ethyl ester precursors
    • 2-s2.0-0026508890 10.1016/0024-3205(92)90271-P
    • Kasafirek E., Rybak M., Krejci I., Sturc A., Krepela E., Sedo A., Two-step generation of spirocyclic dipeptides from linear peptide ethyl ester precursors. Life Sciences 1992 50 3 187 193 2-s2.0-0026508890 10.1016/0024-3205(92)90271-P
    • (1992) Life Sciences , vol.50 , Issue.3 , pp. 187-193
    • Kasafirek, E.1    Rybak, M.2    Krejci, I.3    Sturc, A.4    Krepela, E.5    Sedo, A.6
  • 6
    • 0015093326 scopus 로고
    • Regulation of formation and proposed structure of the factor inhibiting the release of melanocyte-stimulating hormone
    • 2-s2.0-0015093326
    • Celis M. E., Taleisnik S., Walter R., Regulation of formation and proposed structure of the factor inhibiting the release of melanocyte- stimulating hormone. Proceedings of the National Academy of Sciences of the United States of America 1971 68 7 1428 1433 2-s2.0-0015093326
    • (1971) Proceedings of the National Academy of Sciences of the United States of America , vol.68 , Issue.7 , pp. 1428-1433
    • Celis, M.E.1    Taleisnik, S.2    Walter, R.3
  • 7
    • 9744248711 scopus 로고    scopus 로고
    • Prolyl-leucyl-glycinamide shares some effects with oxytocin but decreases oxytocin levels
    • DOI 10.1016/j.physbeh.2004.08.034, PII S0031938404003865
    • Petersson M., Uvnäs-Moberg K., Prolyl-leucyl-glycinamide shares some effects with oxytocin but decreases oxytocin levels. Physiology and Behavior 2004 83 3 475 481 2-s2.0-9744248711 10.1016/j.physbeh.2004.08.034 (Pubitemid 39586670)
    • (2004) Physiology and Behavior , vol.83 , Issue.3 , pp. 475-481
    • Petersson, M.1    Uvnas-Moberg, K.2
  • 9
    • 84893835509 scopus 로고    scopus 로고
    • Inventors; Faculty of Pharmacy, University of Veterinary and Pharmaceutical Sciences Brno, assignee, "Alaptide: Methods of effecting its solubility, membrane permeation and pharmaceutical compositions for human and veterinary applications", PTC/CZ2012/000074, 2012
    • Jampílek J., Opatrilova R., Rezacova A., Oktabec Z., Dohnal J.,. Inventors; Faculty of Pharmacy, University of Veterinary and Pharmaceutical Sciences Brno, assignee, "Alaptide: Methods of effecting its solubility, membrane permeation and pharmaceutical compositions for human and veterinary applications" PTC/CZ2012/000074, 2012
    • Jampílek, J.1    Opatrilova, R.2    Rezacova, A.3    Oktabec, Z.4    Dohnal, J.5
  • 10
    • 79959231140 scopus 로고    scopus 로고
    • Liquid chromatographic method for enantiopurity control of alaptide using polysaccharide stationary phases
    • 2-s2.0-79959231140 10.1002/jssc.201100135
    • Douša M., Lemr K., Liquid chromatographic method for enantiopurity control of alaptide using polysaccharide stationary phases. Journal of Separation Science 2011 34 12 1402 1406 2-s2.0-79959231140 10.1002/jssc. 201100135
    • (2011) Journal of Separation Science , vol.34 , Issue.12 , pp. 1402-1406
    • Douša, M.1    Lemr, K.2
  • 11
    • 62349116508 scopus 로고    scopus 로고
    • X-ray powder diffraction data for alaptide, 8(S)-methyl-6,9-diazaspiro/4, 5/decane-7,10-dione or cyclo(l-alanyl-1-amino-1-cyclopentan carbonyl), cyclo(l-Ala-Acp)
    • 2-s2.0-69549113358
    • Maixner J., Rohlíček J., Kratochvíl B., Šturc A., X-ray powder diffraction data for alaptide, 8(S)-methyl-6,9-diazaspiro/4,5/ decane-7,10-dione or cyclo(l-alanyl-1-amino-1-cyclopentan carbonyl), cyclo(l-Ala-Acp). Powder Diffraction 2009 24 32 34 2-s2.0-69549113358
    • (2009) Powder Diffraction , vol.24 , pp. 32-34
    • Maixner, J.1    Rohlíček, J.2    Kratochvíl, B.3    Šturc, A.4
  • 15
    • 0024005907 scopus 로고
    • The epidermal keratinocyte
    • 2-s2.0-0024005907
    • Watt F. M., The epidermal keratinocyte. BioEssays 1988 8 5 163 167 2-s2.0-0024005907
    • (1988) BioEssays , vol.8 , Issue.5 , pp. 163-167
    • Watt, F.M.1
  • 16
    • 0022656905 scopus 로고
    • Inhibition of proliferative activity by cyclic dipeptides: Spirocyclic derivatives of 1-aminocyclopentanecarboxylic acid
    • Vanzura J., Kosar K., Kasafirek E., Inhibition of proliferative activity by cyclic dipeptides: spirocyclic derivatives of 1-aminocyclopentanecarboxylic acid. Toxicology Letters 1986 31 3 189 193 2-s2.0-0022656905 (Pubitemid 16098315)
    • (1986) Toxicology Letters , vol.31 , Issue.3 , pp. 189-193
    • Vanzura, J.1    Kosar, K.2    Kasafirek, E.3
  • 17
    • 0026042950 scopus 로고
    • Pharmacokinetics and brain entry of alaptide, a novel nootropic agent, in mice, rats and rabbits
    • 2-s2.0-0026042950
    • Lapka R., Pharmacokinetics and brain entry of alaptide, a novel nootropic agent, in mice, rats and rabbits. Journal of Pharmacy and Pharmacology 1991 43 12 874 876 2-s2.0-0026042950
    • (1991) Journal of Pharmacy and Pharmacology , vol.43 , Issue.12 , pp. 874-876
    • Lapka, R.1
  • 18
    • 0023716854 scopus 로고
    • Embryotoxicity of L-prolyl-L-leucyl-glycinamide, cyclo(1-amino- cyclopentanecarbonyl-alanyl) and cyclo(glycyl-leucyl), new potential neuropeptides in chick embryos
    • Kosar K., Vanzura J., Embryotoxicity of L-prolyl-L-leucyl-glycinamide, cyclo(1-amino-cyclopentanecarbonyl-alanyl) and cyclo(glycyl-leucyl), new potential neuropeptides in chick embryos. Pharmazie 1988 43 10 715 716 2-s2.0-0023716854 (Pubitemid 18260308)
    • (1988) Pharmazie , vol.43 , Issue.10 , pp. 715-716
    • Kosar, K.1    Vanzura, J.2
  • 19
    • 84893862412 scopus 로고    scopus 로고
    • Bioveta-Alaptid veterinary ointment.cz
    • Bioveta-Alaptid veterinary ointment.cz, http://www.bioveta.cz/en/ veterinary-division/products/new-products-for-dogs-and-cats/alaptid-veterinary- ointment.html
  • 21
    • 73949137818 scopus 로고    scopus 로고
    • Penetration of nanoparticles and nanomaterials in the skin: Fiction or reality?
    • 2-s2.0-73949137818 10.1002/jps.21817
    • Baroli B., Penetration of nanoparticles and nanomaterials in the skin: fiction or reality? Journal of Pharmaceutical Sciences 2010 99 1 21 50 2-s2.0-73949137818 10.1002/jps.21817
    • (2010) Journal of Pharmaceutical Sciences , vol.99 , Issue.1 , pp. 21-50
    • Baroli, B.1
  • 25
    • 0032568397 scopus 로고    scopus 로고
    • Physicochemical high throughput screening: Parallel artificial membrane permeation assay in the description of passive absorption processes
    • DOI 10.1021/jm970530e
    • Kansy M., Senner F., Gubernator K., Physicochemical high throughput screening: parallel artificial membrane permeation assay in the description of passive absorption processes. Journal of Medicinal Chemistry 1998 41 7 1007 1010 2-s2.0-0032568397 10.1021/jm970530e (Pubitemid 28207375)
    • (1998) Journal of Medicinal Chemistry , vol.41 , Issue.7 , pp. 1007-1010
    • Kansy, M.1    Senner, F.2    Gubernator, K.3
  • 26
    • 33644895433 scopus 로고    scopus 로고
    • PAMPA - A drug absorption in vitro model: 13. Chemical selectivity due to membrane hydrogen bonding: In combo comparisons of HDM-, DOPC-, and DS-PAMPA models
    • 2-s2.0-33644895433 10.1016/j.ejps.2005.12.008
    • Avdeef A., Tsinman O., PAMPA-a drug absorption in vitro model: 13. Chemical selectivity due to membrane hydrogen bonding: in combo comparisons of HDM-, DOPC-, and DS-PAMPA models. European Journal of Pharmaceutical Sciences 2006 28 1-2 43 50 2-s2.0-33644895433 10.1016/j.ejps.2005.12.008
    • (2006) European Journal of Pharmaceutical Sciences , vol.28 , Issue.1-2 , pp. 43-50
    • Avdeef, A.1    Tsinman, O.2
  • 28
    • 0016610679 scopus 로고
    • Percutaneous absorption. on the relevance of in vitro data
    • 2-s2.0-0016610679
    • Franz T. J., Percutaneous absorption. On the relevance of in vitro data. Journal of Investigative Dermatology 1975 64 3 190 195 2-s2.0-0016610679
    • (1975) Journal of Investigative Dermatology , vol.64 , Issue.3 , pp. 190-195
    • Franz, T.J.1
  • 29
    • 84864851442 scopus 로고    scopus 로고
    • Azone analogues: Classification, design, and transdermal penetration principles
    • Jampilek J., Brychtova K., Azone analogues: classification, design, and transdermal penetration principles. Medical Research Review 2012 32 907 947
    • (2012) Medical Research Review , vol.32 , pp. 907-947
    • Jampilek, J.1    Brychtova, K.2
  • 30
    • 84888396706 scopus 로고    scopus 로고
    • Transdermal application of drugs and techniques affecting skin barrier
    • Jampilek J., Transdermal application of drugs and techniques affecting skin barrier. Journal of Bioequivalence & Bioavailability 2013 5 233 235
    • (2013) Journal of Bioequivalence & Bioavailability , vol.5 , pp. 233-235
    • Jampilek, J.1
  • 32
    • 33746921312 scopus 로고    scopus 로고
    • Pig ear skin ex vivo as a model for in vivo dermatopharmacokinetic studies in man
    • DOI 10.1007/s11095-006-9011-8
    • Herkenne C., Naik A., Kalia Y. N., Hadgraft J., Guy R. H., Pig ear skin ex vivo as a model for in vivo dermatopharmacokinetic studies in man. Pharmaceutical Research 2006 23 8 1850 1856 2-s2.0-33746921312 10.1007/s11095-006-9011-8 (Pubitemid 44200549)
    • (2006) Pharmaceutical Research , vol.23 , Issue.8 , pp. 1850-1856
    • Herkenne, C.1    Naik, A.2    Kalia, Y.N.3    Hadgraft, J.4    Guy, R.H.5
  • 33
    • 0018228183 scopus 로고
    • The skin of domestic mammals as a model for the human skin, with special reference to the domestic pig
    • 2-s2.0-0018228183
    • Meyer W., Schwarz R., Neurand K., The skin of domestic mammals as a model for the human skin, with special reference to the domestic pig. Current Problems in Dermatology 1978 7 39 52 2-s2.0-0018228183
    • (1978) Current Problems in Dermatology , vol.7 , pp. 39-52
    • Meyer, W.1    Schwarz, R.2    Neurand, K.3
  • 34
    • 0035806281 scopus 로고    scopus 로고
    • Topical transport of hydrophilic compounds using water-in-oil nanoemulsions
    • DOI 10.1016/S0378-5173(01)00671-8, PII S0378517301006718
    • Wu H., Ramachandran C., Weiner N. D., Roessler B. J., Topical transport of hydrophilic compounds using water-in-oil nanoemulsions. International Journal of Pharmaceutics 2001 220 1-2 63 75 2-s2.0-0035806281 10.1016/S0378-5173(01) 00671-8 (Pubitemid 32476842)
    • (2001) International Journal of Pharmaceutics , vol.220 , Issue.1-2 , pp. 63-75
    • Wu, H.1    Ramachandran, C.2    Weiner, N.D.3    Roessler, B.J.4
  • 35
    • 79959990575 scopus 로고    scopus 로고
    • Penetration enhancing effect of polysorbate 20 and 80 on the in vitro percutaneous absorption of L-ascorbic acid
    • 2-s2.0-79959990575 10.4314/tjpr.v10i3.1
    • Akhtar N., Rehman M. U., Khan H. M. S., Rasool F., Saeed T., Murtaza G., Penetration enhancing effect of polysorbate 20 and 80 on the in vitro percutaneous absorption of L-ascorbic acid. Tropical Journal of Pharmaceutical Research 2011 10 3 281 288 2-s2.0-79959990575 10.4314/tjpr.v10i3.1
    • (2011) Tropical Journal of Pharmaceutical Research , vol.10 , Issue.3 , pp. 281-288
    • Akhtar, N.1    Rehman, M.U.2    Khan, H.M.S.3    Rasool, F.4    Saeed, T.5    Murtaza, G.6
  • 36
    • 27744519546 scopus 로고    scopus 로고
    • The effect of pH and organic ester penetration enhancers on skin permeation kinetics of terbutaline sulfate from pseudolatex-type transdermal delivery systems through mouse and human cadaver skins
    • DOI 10.1208/pt060225, 25
    • Panigrahi L., Pattnaik S., Ghosal S. K., The effect of pH and organic ester penetration enhancers on skin permeation kinetics of terbutaline sulfate from pseudolatex-type transdermal delivery systems through mouse and human cadaver skins. AAPS PharmSciTech 2005 6 2 E167 E173 2-s2.0-27744519546 10.1208/pt060225 (Pubitemid 41631756)
    • (2005) AAPS PharmSciTech , vol.6 , Issue.2
    • Panigrahi, L.1    Pattnaik, S.2    Ghosal, S.K.3
  • 37
    • 84879582787 scopus 로고    scopus 로고
    • Effect of microemulsions on transdermal delivery of citalopram: Optimization studies using mixture design and response surface methodology
    • Huang C. T., Tsai M. J., Lin Y. H., Effect of microemulsions on transdermal delivery of citalopram: optimization studies using mixture design and response surface methodology. International Journal of Nanomedicine 2013 2013 2295 2304
    • (2013) International Journal of Nanomedicine , vol.2013 , pp. 2295-2304
    • Huang, C.T.1    Tsai, M.J.2    Lin, Y.H.3
  • 38
    • 0035834177 scopus 로고    scopus 로고
    • Transdermal delivery of ketoprofen using microemulsions
    • DOI 10.1016/S0378-5173(01)00827-4, PII S0378517301008274
    • Rhee Y.-S., Choi J.-G., Park E.-S., Chi S.-C., Transdermal delivery of ketoprofen using microemulsions. International Journal of Pharmaceutics 2001 228 1-2 161 170 2-s2.0-0035834177 10.1016/S0378-5173(01)00827-4 (Pubitemid 32905375)
    • (2001) International Journal of Pharmaceutics , vol.228 , Issue.1-2 , pp. 161-170
    • Rhee, Y.-S.1    Choi, J.-G.2    Park, E.-S.3    Chi, S.-C.4
  • 39
    • 29844432699 scopus 로고    scopus 로고
    • A review of the effect of occlusive dressings on lamellar bodies in the stratum corneum and relevance to transdermal absorption
    • 2-s2.0-33746792072
    • Kennish L., Reidenberg B., A review of the effect of occlusive dressings on lamellar bodies in the stratum corneum and relevance to transdermal absorption. Dermatology Online Journal 2005 11 3 7 2-s2.0-33746792072
    • (2005) Dermatology Online Journal , vol.11 , Issue.3 , pp. 7
    • Kennish, L.1    Reidenberg, B.2
  • 41
    • 85123316636 scopus 로고    scopus 로고
    • Nanomaterials and nanoparticles: Sources and toxicity
    • Buzea C., Pacheco I. I., Robbie K., Nanomaterials and nanoparticles: sources and toxicity. Biointerphases 2007 2 MR17 MR71
    • (2007) Biointerphases , vol.2
    • Buzea, C.1    Pacheco, I.I.2    Robbie, K.3
  • 43
    • 73949087550 scopus 로고    scopus 로고
    • Effect of surface properties on nanoparticle-cell interactions
    • 2-s2.0-73949087550 10.1002/smll.200901158
    • Verma A., Stellacci F., Effect of surface properties on nanoparticle-cell interactions. Small 2010 6 1 12 21 2-s2.0-73949087550 10.1002/smll.200901158
    • (2010) Small , vol.6 , Issue.1 , pp. 12-21
    • Verma, A.1    Stellacci, F.2
  • 45
    • 0028898732 scopus 로고
    • Quantitative structure-activity relationships for skin permeability
    • 2-s2.0-0028898732 10.1016/0887-2333(94)00190-6
    • Barratt M. D., Quantitative structure-activity relationships for skin permeability. Toxicology in Vitro 1995 9 1 27 37 2-s2.0-0028898732 10.1016/0887-2333(94)00190-6
    • (1995) Toxicology in Vitro , vol.9 , Issue.1 , pp. 27-37
    • Barratt, M.D.1


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