Synthesis of 2H-1,3-benzoxazin-4(3H)-one derivatives containing indole moiety: Their in vitro evaluation against PDE4B

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 4, 2014, Pages 1166-1171

  Rao, Raja Mohan ^a   Luther, Bethala Jawahar ^b   Rani, Chekuri Sharmila ^c   Suresh, Namburi ^c   Kapavarapu, Ravikumar ^d   Parsa, Kishore V L ^a   Rao, Mandava V Basaveswara ^c   Pal, Manojit ^a  

^a INSTITUTE OF LIFE SCIENCES   (India)

^b ACHARYA NAGARJUNA UNIVERSITY   (India)

^c KRISHNA UNIVERSITY   (India)

^d UNIVERSITY OF COIMBRA   (Portugal)

Author keywords

2H 1,3 Benzoxazin 4(3H) one; Benzofuran; Indole; Pd C; PDE4

Indexed keywords

2H-1,3-BENZOXAZIN-4(3H)-ONE; BENZOFURAN; INDOLE; PD/C; PDE4;

CYCLIC NUCLEOTIDE PHOSPHODIESTERASES, TYPE 4; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; HEK293 CELLS; HUMANS; INDOLES; MODELS, MOLECULAR; MOLECULAR STRUCTURE; OXAZINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84893807720     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.12.117     Document Type: Article

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