SCOPUS 정보 검색 플랫폼

Volumn 12, Issue 6, 2014, Pages 965-978

Design, synthesis and binding properties of a fluorescent α9β1/α4β1 integrin antagonist and its application as an in vivo probe for bone marrow haemopoietic stem cells

(10) Cao, Benjamin a Hutt, Oliver E a Zhang, Zhen a Li, Songhui a Heazlewood, Shen Y a Williams, Brenda a Smith, Jessica A a Haylock, David N a,b Savage, G Paul a Nilsson, Susan K a,b

a CSIRO (Australia)

b MONASH UNIVERSITY (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

BINDING ENERGY; BONE; CHEMICAL ACTIVATION; COPPER COMPOUNDS; CYTOLOGY; FLUORESCENCE; GLYCOPROTEINS; KETONES; MOLECULES; PROBES; PROTEINS;

AZIDE-ALKYNE CYCLOADDITION; BINDING AFFINITIES; BINDING PROPERTIES; BIOCHEMICAL PROPERTIES; BIOLOGICAL PROCESS; FLUORESCENT PROBES; PROTEIN INTERACTION; SMALL MOLECULE INHIBITOR;

STEM CELLS;

DIPEPTIDE; DRUG DERIVATIVE; FLUORESCENT DYE; INTEGRIN; INTEGRIN ALPHA 9 BETA 1; PROLINE; R BC154; R-BC154; RHODAMINE; VERY LATE ACTIVATION ANTIGEN 4;

ARTICLE; BINDING SITE; BONE MARROW CELL; CHEMISTRY; CONFORMATION; CYTOLOGY; DOSE RESPONSE; DRUG ANTAGONISM; DRUG DESIGN; DRUG EFFECT; FLUORESCENCE; HUMAN; STRUCTURE ACTIVITY RELATION; SYNTHESIS; TUMOR CELL LINE;

BINDING SITES; BONE MARROW CELLS; CELL LINE, TUMOR; DIPEPTIDES; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; FLUORESCENCE; FLUORESCENT DYES; HUMANS; INTEGRIN ALPHA4BETA1; INTEGRINS; MOLECULAR CONFORMATION; PROLINE; RHODAMINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84892576496 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/c3ob42332h Document Type: Article

Times cited : (10)

References (42)

1
- 0026770377
- R. O. Hynes Cell 1992 69 11 25
- (1992) Cell , vol.69 , pp. 11-25
- Hynes, R.O.¹

2
- 0028987936
- E. A. Clark J. S. Brugge Science 1995 268 233 239
- (1995) Science , vol.268 , pp. 233-239
- Clark, E.A.¹ Brugge, J.S.²

3
- 77957363101
- D. Cox M. Brennan N. Moran Nat. Rev. Drug. Discovery 2010 9 804 820
- (2010) Nat. Rev. Drug. Discovery , vol.9 , pp. 804-820
- Cox, D.¹ Brennan, M.² Moran, N.³

4
- 33750453714
- J. D. Humphries A. Byron M. J. Humphries J. Cell Sci. 2006 119 3901 3903
- (2006) J. Cell Sci. , vol.119 , pp. 3901-3903
- Humphries, J.D.¹ Byron, A.² Humphries, M.J.³

5
- 0031802697
- K. J. Bayless G. A. Meininger J. M. Scholtz G. E. Davis J. Cell Sci. 1998 111 1165 1174
- (1998) J. Cell Sci. , vol.111 , pp. 1165-1174
- Bayless, K.J.¹ Meininger, G.A.² Scholtz, J.M.³ Davis, G.E.⁴

6
- 0028173015
- R. R. Lobb M. E. Hemler J. Clin. Invest. 1994 94 1722 1728
- (1994) J. Clin. Invest. , vol.94 , pp. 1722-1728
- Lobb, R.R.¹ Hemler, M.E.²

7
- 0032797233
- R. R. Lobb S. P. Adams Expert Opin. Invest. Drugs 1999 8 935 945
- (1999) Expert Opin. Invest. Drugs , vol.8 , pp. 935-945
- Lobb, R.R.¹ Adams, S.P.²

8
- 80255122951
- M. Millard S. Odde N. Neamati Theranostics 2011 1 154 188
- (2011) Theranostics , vol.1 , pp. 154-188
- Millard, M.¹ Odde, S.² Neamati, N.³

9
- 0033583322
- Y. Taooka J. Chen T. Yednock D. Sheppard J. Cell Biol. 1999 145 413 420
- (1999) J. Cell Biol. , vol.145 , pp. 413-420
- Taooka, Y.¹ Chen, J.² Yednock, T.³ Sheppard, D.⁴

10
- 0033579511
- Y. Yokosaki N. Matsuura T. Sasaki I. Murakami H. Schneider S. Higashiyama Y. Saitoh M. Yamakido Y. Taooka D. Sheppard J. Biol. Chem. 1999 274 36328 36334
- (1999) J. Biol. Chem. , vol.274 , pp. 36328-36334
- Yokosaki, Y.¹ Matsuura, N.² Sasaki, T.³ Murakami, I.⁴ Schneider, H.⁵ Higashiyama, S.⁶ Saitoh, Y.⁷ Yamakido, M.⁸ Taooka, Y.⁹ Sheppard, D.¹⁰

11
- 0034604565
- H. Takahashi T. Isobe S. Horibe J. Takagi Y. Yokosaki D. Sheppard Y. Saito J. Biol. Chem. 2000 275 23589 23595
- (2000) J. Biol. Chem. , vol.275 , pp. 23589-23595
- Takahashi, H.¹ Isobe, T.² Horibe, S.³ Takagi, J.⁴ Yokosaki, Y.⁵ Sheppard, D.⁶ Saito, Y.⁷

12
- 18444398629
- R. B. Pepinsky R. A. Mumford L. L. Chen D. Leone S. E. Amo G. Van Riper A. Whitty B. Dolinski R. R. Lobb D. C. Dean L. L. Chang C. E. Raab Q. Si W. K. Hagmann R. B. Lingham Biochemistry 2002 41 7125 7141
- (2002) Biochemistry , vol.41 , pp. 7125-7141
- Pepinsky, R.B.¹ Mumford, R.A.² Chen, L.L.³ Leone, D.⁴ Amo, S.E.⁵ Van Riper, G.⁶ Whitty, A.⁷ Dolinski, B.⁸ Lobb, R.R.⁹ Dean, D.C.¹⁰ Chang, L.L.¹¹ Raab, C.E.¹² Si, Q.¹³ Hagmann, W.K.¹⁴ Lingham, R.B.¹⁵

13
- 34447502532
- N. E. Vlahakis B. A. Young A. Atakilit A. E. Hawkridge R. B. Issaka N. Boudreau D. Sheppard J. Biol. Chem. 2007 282 15187 15196
- (2007) J. Biol. Chem. , vol.282 , pp. 15187-15196
- Vlahakis, N.E.¹ Young, B.A.² Atakilit, A.³ Hawkridge, A.E.⁴ Issaka, R.B.⁵ Boudreau, N.⁶ Sheppard, D.⁷

14
- 84862840437
- E. M. Walsh R. Kim L. Del Valle M. Weaver J. Sheffield P. Lazarovici C. Marcinkiewicz Neuro-Oncology 2012 14 890 901
- (2012) Neuro-Oncology , vol.14 , pp. 890-901
- Walsh, E.M.¹ Kim, R.² Del Valle, L.³ Weaver, M.⁴ Sheffield, J.⁵ Lazarovici, P.⁶ Marcinkiewicz, C.⁷

15
- 58149332702
- P. Singh C. Chen S. Pal-Ghosh M. A. Stepp D. Sheppard L. Van De Water J. Invest. Dermatol. 2009 129 217 228
- (2009) J. Invest. Dermatol. , vol.129 , pp. 217-228
- Singh, P.¹ Chen, C.² Pal-Ghosh, S.³ Stepp, M.A.⁴ Sheppard, D.⁵ Van De Water, L.⁶

16
- 34248376549
- I. Staniszewska S. Zaveri L. Del Valle I. Oliva V. L. Rothman S. E. Croul D. D. Roberts D. F. Mosher G. P. Tuszynski C. Marcinkiewicz Circ. Res. 2007 100 1308 1316
- (2007) Circ. Res. , vol.100 , pp. 1308-1316
- Staniszewska, I.¹ Zaveri, S.² Del Valle, L.³ Oliva, I.⁴ Rothman, V.L.⁵ Croul, S.E.⁶ Roberts, D.D.⁷ Mosher, D.F.⁸ Tuszynski, G.P.⁹ Marcinkiewicz, C.¹⁰

17
- 0026779726
- J. Teixido M. E. Hemler J. S. Greenberger P. Anklesaria J. Clin. Invest. 1992 90 358 367
- (1992) J. Clin. Invest. , vol.90 , pp. 358-367
- Teixido, J.¹ Hemler, M.E.² Greenberger, J.S.³ Anklesaria, P.⁴

18
- 67651071765
- J. Grassinger D. N. Haylock M. J. Storan G. O. Haines B. Williams G. A. Whitty A. R. Vinson C. L. Be S. H. Li E. S. Sorensen P. P. L. Tam D. T. Denhardt D. Sheppard P. F. Choong S. K. Nilsson Blood 2009 114 49 59
- (2009) Blood , vol.114 , pp. 49-59
- Grassinger, J.¹ Haylock, D.N.² Storan, M.J.³ Haines, G.O.⁴ Williams, B.⁵ Whitty, G.A.⁶ Vinson, A.R.⁷ Be, C.L.⁸ Li, S.H.⁹ Sorensen, E.S.¹⁰ Tam, P.P.L.¹¹ Denhardt, D.T.¹² Sheppard, D.¹³ Choong, P.F.¹⁴ Nilsson, S.K.¹⁵

19
- 70449393572
- T. D. Schreiber C. Steinl M. Essl H. Abele K. Geiger C. A. Muller W. K. Aicher G. Klein Haematol.-Hematol. J. 2009 94 1493 1501
- (2009) Haematol.-Hematol. J. , vol.94 , pp. 1493-1501
- Schreiber, T.D.¹ Steinl, C.² Essl, M.³ Abele, H.⁴ Geiger, K.⁵ Muller, C.A.⁶ Aicher, W.K.⁷ Klein, G.⁸

20
- 70349348954
- P. Ramirez M. P. Rettig G. L. Uy E. Deych M. S. Holt J. K. Ritchey J. F. DiPersio Blood 2009 114 1340 1343
- (2009) Blood , vol.114 , pp. 1340-1343
- Ramirez, P.¹ Rettig, M.P.² Uy, G.L.³ Deych, E.⁴ Holt, M.S.⁵ Ritchey, J.K.⁶ Dipersio, J.F.⁷

21
- 35848946625
- S. Choi G. Vilaire C. Marcinkiewicz J. D. Winkler J. S. Bennett W. F. DeGrado J. Med. Chem. 2007 50 5457 5462
- (2007) J. Med. Chem. , vol.50 , pp. 5457-5462
- Choi, S.¹ Vilaire, G.² Marcinkiewicz, C.³ Winkler, J.D.⁴ Bennett, J.S.⁵ Degrado, W.F.⁶

22
- 58849165421
- M. W. Miller S. Basra D. W. Kulp P. C. Billings S. Choi M. P. Beavers O. J. T. McCartye Z. Y. Zou M. L. Kahn J. S. Bennett W. F. DeGrado Proc. Natl. Acad. Sci. U. S. A. 2009 106 719 724
- (2009) Proc. Natl. Acad. Sci. U. S. A. , vol.106 , pp. 719-724
- Miller, M.W.¹ Basra, S.² Kulp, D.W.³ Billings, P.C.⁴ Choi, S.⁵ Beavers, M.P.⁶ McCartye, O.J.T.⁷ Zou, Z.Y.⁸ Kahn, M.L.⁹ Bennett, J.S.¹⁰ Degrado, W.F.¹¹

23
- 80052951717
- O. E. Hutt S. Saubern D. A. Winkler Bioorg. Med. Chem. 2011 19 5903 5911
- (2011) Bioorg. Med. Chem. , vol.19 , pp. 5903-5911
- Hutt, O.E.¹ Saubern, S.² Winkler, D.A.³

24
- 23644434240
- S. Venkatraman J. Lim M. Cramer M. F. Gardner J. James K. Alves R. B. Lingham R. A. Mumford B. Munoz Bioorg. Med. Chem. Lett. 2005 15 4053 4056
- (2005) Bioorg. Med. Chem. Lett. , vol.15 , pp. 4053-4056
- Venkatraman, S.¹ Lim, J.² Cramer, M.³ Gardner, M.F.⁴ James, J.⁵ Alves, K.⁶ Lingham, R.B.⁷ Mumford, R.A.⁸ Munoz, B.⁹

25
- 19944434038
- R. B. Pepinsky W. C. Lee M. Cornebise A. Gill K. Wortham L. L. Chen D. R. Leone K. Giza B. M. Dolinski S. Perper C. Nickerson-Nutter D. Lepage A. Chakraborty E. T. Whalley R. C. Petter S. P. Adams R. R. Lobb D. M. Scott J. Pharmacol. Exp. Ther. 2005 312 742 750
- (2005) J. Pharmacol. Exp. Ther. , vol.312 , pp. 742-750
- Pepinsky, R.B.¹ Lee, W.C.² Cornebise, M.³ Gill, A.⁴ Wortham, K.⁵ Chen, L.L.⁶ Leone, D.R.⁷ Giza, K.⁸ Dolinski, B.M.⁹ Perper, S.¹⁰ Nickerson-Nutter, C.¹¹ Lepage, D.¹² Chakraborty, A.¹³ Whalley, E.T.¹⁴ Petter, R.C.¹⁵ Adams, S.P.¹⁶ Lobb, R.R.¹⁷ Scott, D.M.¹⁸

26
- 66749172274
- L. S. Lin T. Lanza J. P. Jewell P. Liu C. Jones G. R. Kieczykowski K. Treonze Q. Si S. Manior G. Koo X. C. Tong J. Y. Wang A. Schuelke J. Pivnichny R. Wang C. Raab S. Vincent P. Davies M. MacCoss R. A. Mumford W. K. Hagmann J. Med. Chem. 2009 52 3449 3452
- (2009) J. Med. Chem. , vol.52 , pp. 3449-3452
- Lin, L.S.¹ Lanza, T.² Jewell, J.P.³ Liu, P.⁴ Jones, C.⁵ Kieczykowski, G.R.⁶ Treonze, K.⁷ Si, Q.⁸ Manior, S.⁹ Koo, G.¹⁰ Tong, X.C.¹¹ Wang, J.Y.¹² Schuelke, A.¹³ Pivnichny, J.¹⁴ Wang, R.¹⁵ Raab, C.¹⁶ Vincent, S.¹⁷ Davies, P.¹⁸ Maccoss, M.¹⁹ Mumford, R.A.²⁰ Hagmann, W.K.²¹ more..

27
- 81255143135
- J. A. Smith G. P. Savage O. E. Hutt Aust. J. Chem. 2011 64 1509 1514
- (2011) Aust. J. Chem. , vol.64 , pp. 1509-1514
- Smith, J.A.¹ Savage, G.P.² Hutt, O.E.³

28
- 84857584455
- C. E. Jakobsche P. J. McEnaney A. X. Zhang D. A. Spiegel ACS Chem. Biol. 2012 7 315 320
- (2012) ACS Chem. Biol. , vol.7 , pp. 315-320
- Jakobsche, C.E.¹ McEnaney, P.J.² Zhang, A.X.³ Spiegel, D.A.⁴

29
- 74049161233
- T. S. Reger J. Zunic N. Stock B. W. Wang N. D. Smith B. Munoz M. D. Green M. F. Gardner J. P. James W. C. Chen K. Alves Q. Si K. M. Treonze R. B. Lingham R. A. Mumford Bioorg. Med. Chem. Lett. 2010 20 1173 1176
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 1173-1176
- Reger, T.S.¹ Zunic, J.² Stock, N.³ Wang, B.W.⁴ Smith, N.D.⁵ Munoz, B.⁶ Green, M.D.⁷ Gardner, M.F.⁸ James, J.P.⁹ Chen, W.C.¹⁰ Alves, K.¹¹ Si, Q.¹² Treonze, K.M.¹³ Lingham, R.B.¹⁴ Mumford, R.A.¹⁵

30
- 0037012920
- C. W. Tornoe C. Christensen M. Meldal J. Org. Chem. 2002 67 3057 3064
- (2002) J. Org. Chem. , vol.67 , pp. 3057-3064
- Tornoe, C.W.¹ Christensen, C.² Meldal, M.³

31
- 0037099395
- V. V. Rostovtsev L. G. Green V. V. Fokin K. B. Sharpless Angew. Chem., Int. Ed. 2002 41 2596 2599
- (2002) Angew. Chem., Int. Ed. , vol.41 , pp. 2596-2599
- Rostovtsev, V.V.¹ Green, L.G.² Fokin, V.V.³ Sharpless, K.B.⁴

32
- 80255122805
- T. C. Liu J. R. Nedrow-Byers M. R. Hopkins C. E. Berkman Bioorg. Med. Chem. Lett. 2011 21 7013 7016
- (2011) Bioorg. Med. Chem. Lett. , vol.21 , pp. 7013-7016
- Liu, T.C.¹ Nedrow-Byers, J.R.² Hopkins, M.R.³ Berkman, C.E.⁴

33
- 55249094052
- K. E. Beatty D. A. Tirrel Bioorg. Med. Chem. Lett. 2008 18 5995 5999
- (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 5995-5999
- Beatty, K.E.¹ Tirrel, D.A.²

34
- 79958779833
- A. H. Broderick S. M. Azarin M. E. Buck S. P. Palecek D. M. Lynn Biomacromolecules 2011 12 1998 2007
- (2011) Biomacromolecules , vol.12 , pp. 1998-2007
- Broderick, A.H.¹ Azarin, S.M.² Buck, M.E.³ Palecek, S.P.⁴ Lynn, D.M.⁵

35
- 84869091676
- G. Delaittre A. M. Greiner T. Pauloehrl M. Bastmeyer C. Barner-Kowollik Soft Matter 2012 8 7323 7347
- (2012) Soft Matter , vol.8 , pp. 7323-7347
- Delaittre, G.¹ Greiner, A.M.² Pauloehrl, T.³ Bastmeyer, M.⁴ Barner-Kowollik, C.⁵

36
- 0029969086
- A. P. Mould J. Cell Sci. 1996 109 2613 2618
- (1996) J. Cell Sci. , vol.109 , pp. 2613-2618
- Mould, A.P.¹

37
- 0034698147
- E. F. Plow T. K. Haas L. Zhang J. Loftus J. W. Smith J. Biol. Chem. 2000 275 21785 21788
- (2000) J. Biol. Chem. , vol.275 , pp. 21785-21788
- Plow, E.F.¹ Haas, T.K.² Zhang, L.³ Loftus, J.⁴ Smith, J.W.⁵

38
- 78049378252
- J. Grassinger D. N. Haylock B. Williams G. H. Olsen S. K. Nilsson Blood 2010 116 3185 3196
- (2010) Blood , vol.116 , pp. 3185-3196
- Grassinger, J.¹ Haylock, D.N.² Williams, B.³ Olsen, G.H.⁴ Nilsson, S.K.⁵

39
- 5244370033
- A. B. Pangborn M. A. Giardello R. H. Grubbs R. K. Rosen F. J. Timmers Organometallics 1996 15 1518 1520
- (1996) Organometallics , vol.15 , pp. 1518-1520
- Pangborn, A.B.¹ Giardello, M.A.² Grubbs, R.H.³ Rosen, R.K.⁴ Timmers, F.J.⁵

40
- 0009833614
- R. H. Andreatta V. Nair A. V. Roberston Aust. J. Chem. 1967 20 2701 2713
- (1967) Aust. J. Chem. , vol.20 , pp. 2701-2713
- Andreatta, R.H.¹ Nair, V.² Roberston, A.V.³

41
- 34147097546
- D. N. Haylock B. Williams H. M. Johnston M. C. P. Liu K. E. Rutherford G. A. Whitty P. J. Simmons I. Bertoncello S. K. Nilsson Stem Cells 2007 25 1062 1069
- (2007) Stem Cells , vol.25 , pp. 1062-1069
- Haylock, D.N.¹ Williams, B.² Johnston, H.M.³ Liu, M.C.P.⁴ Rutherford, K.E.⁵ Whitty, G.A.⁶ Simmons, P.J.⁷ Bertoncello, I.⁸ Nilsson, S.K.⁹

42
- 84859212810
- J. Grassinger B. Williams G. H. Olsen D. N. Haylock S. K. Nilsson Cytokine 2012 58 218 225
- (2012) Cytokine , vol.58 , pp. 218-225
- Grassinger, J.¹ Williams, B.² Olsen, G.H.³ Haylock, D.N.⁴ Nilsson, S.K.⁵

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.