SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 2, 2014, Pages 560-564

Synthesis and biological evaluation of 2-aminothiazole derivatives as antimycobacterial and antiplasmodial agents

(8) Mjambili, Faith a Njoroge, Mathew a Naran, Krupa a De Kock, Carmen b Smith, Peter J b Mizrahi, Valerie a Warner, Digby a Chibale, Kelly a

a UNIVERSITY OF CAPE TOWN (South Africa)

b UNIVERSITY OF CAPE TOWN (South Africa)

Author keywords

2 Amino 4 (2 pyridyl)thiazoles; Antimycobacterial; Antiplasmodial; Hit optimisation; Structure activity relationship

Indexed keywords

2 AMINOTHIAZOLE DERIVATIVE; AMIDE; ANTIMYCOBACTERIAL AGENT; ANTIPROTOZOAL AGENT; CHLOROQUINE; PYRIDINE; THIAZOLE;

ANIMAL CELL; ANTIBACTERIAL ACTIVITY; ANTIPROTOZOAL ACTIVITY; ARTICLE; CONTROLLED STUDY; CYTOTOXICITY; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; HYDROPHOBICITY; IN VITRO STUDY; MAMMAL CELL; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PLASMODIUM FALCIPARUM;

MAMMALIA; MYCOBACTERIUM TUBERCULOSIS; PLASMODIUM FALCIPARUM;

2-AMINO-4-(2-PYRIDYL)THIAZOLES; ANTIMYCOBACTERIAL; ANTIPLASMODIAL; HIT OPTIMISATION; STRUCTURE-ACTIVITY RELATIONSHIP;

ANIMALS; ANTI-BACTERIAL AGENTS; ANTIMALARIALS; CHO CELLS; CRICETINAE; CRICETULUS; DRUG EVALUATION, PRECLINICAL; MYCOBACTERIUM TUBERCULOSIS; PLASMODIUM FALCIPARUM; THIAZOLES;

EID: 84891849170 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.12.022 Document Type: Article

Times cited : (61)

References (16)

1
- 84877100401
- World Health Organisation: Geneva, Switzerland
- WHO Global Tuberculosis Report 2012, World Health Organisation: Geneva, Switzerland, 2012.
- (2012) WHO Global Tuberculosis Report 2012

2
- 84877267006
- A. Zumla, P. Nahid, and S.T. Cole Nat. Rev. Drug Discov. 12 2013 388
- (2013) Nat. Rev. Drug Discov. , vol.12 , pp. 388
- Zumla, A.¹ Nahid, P.² Cole, S.T.³

3
- 70350570382
- K.E.A. Lougheed, D.L. Taylor, S.A. Osborne, J.S. Bryans, and R.S. Buxton Tuberculosis (Edinb). 89 2009 364
- (2009) Tuberculosis (Edinb). , vol.89 , pp. 364
- Lougheed, K.E.A.¹ Taylor, D.L.² Osborne, S.A.³ Bryans, J.S.⁴ Buxton, R.S.⁵

4
- 84883436933
- J.C. Palomino, and A. Martin Curr. Med. Chem 20 2013 3785
- (2013) Curr. Med. Chem , vol.20 , pp. 3785
- Palomino, J.C.¹ Martin, A.²

5
- 84891620068
- World Health Organisation: Geneva, Switzerland
- WHO World Malaria Report 2012, World Health Organisation: Geneva, Switzerland, 2012.
- (2012) WHO World Malaria Report 2012

6
- 44349176702
- M. Schlitzer Arch. Pharm. (Weinheim) 341 2008 149
- (2008) Arch. Pharm. (Weinheim) , vol.341 , pp. 149
- Schlitzer, M.¹

7
- 78649887837
- second; World Health Organisation
- WHO Guidelines for the treatment of malaria; second; World Health Organisation, 2010.
- (2010) WHO Guidelines for the Treatment of Malaria

8
- 84861314006
- N. Siddiqui, S. Kumar, W. Ahsan, and B. Azad Int. J. Drug Dev. Res. 3 2011 55
- (2011) Int. J. Drug Dev. Res. , vol.3 , pp. 55
- Siddiqui, N.¹ Kumar, S.² Ahsan, W.³ Azad, B.⁴

9
- 80051940406
- K.K. Roy, S. Singh, S.K. Sharma, R. Srivastava, V. Chaturvedi, and A.K. Saxena Bioorg. Med. Chem. Lett. 21 2011 5589
- (2011) Bioorg. Med. Chem. Lett. , vol.21 , pp. 5589
- Roy, K.K.¹ Singh, S.² Sharma, S.K.³ Srivastava, R.⁴ Chaturvedi, V.⁵ Saxena, A.K.⁶

10
- 77949489030
- G. Turan-Zitouni, Z.A. Kaplancikli, and A. Ozdemir Eur. J. Med. Chem. 45 2010 2085
- (2010) Eur. J. Med. Chem. , vol.45 , pp. 2085
- Turan-Zitouni, G.¹ Kaplancikli, Z.A.² Ozdemir, A.³

11
- 84865707796
- A. Cohen, P. Verhaeghe, M.D. Crozet, S. Hutter, P. Rathelot, P. Vanelle, and N. Azas Eur. J. Med. Chem. 55 2012 315
- (2012) Eur. J. Med. Chem. , vol.55 , pp. 315
- Cohen, A.¹ Verhaeghe, P.² Crozet, M.D.³ Hutter, S.⁴ Rathelot, P.⁵ Vanelle, P.⁶ Azas, N.⁷

12
- 80455140504
- D. González Cabrera, F. Douelle, T.-S. Feng, A.T. Nchinda, Y. Younis, K.L. White, Q. Wu, E. Ryan, J.N. Burrows, D. Waterson, M.J. Witty, S. Wittlin, S.A. Charman, K. Chibale, and D. Gonz J. Med. Chem. 54 2011 7713
- (2011) J. Med. Chem. , vol.54 , pp. 7713
- González Cabrera, D.¹ Douelle, F.² Feng, T.-S.³ Nchinda, A.T.⁴ Younis, Y.⁵ White, K.L.⁶ Wu, Q.⁷ Ryan, E.⁸ Burrows, J.N.⁹ Waterson, D.¹⁰ Witty, M.J.¹¹ Wittlin, S.¹² Charman, S.A.¹³ Chibale, K.¹⁴ Gonz, D.¹⁵

13
- 70350765485
- S. Ananthan, E.R. Faaleolea, R.C. Goldman, J.V. Hobrath, C.D. Kwong, B.E. Laughon, J.a. Maddry, A. Mehta, L. Rasmussen, R.C. Reynolds, J.a. Secrist, N. Shindo, D.N. Showe, E. Sosa, W.J. Suling, and E.L. White Tuberculosis (Edinb) 89 2009 334
- (2009) Tuberculosis (Edinb) , vol.89 , pp. 334
- Ananthan, S.¹ Faaleolea, E.R.² Goldman, R.C.³ Hobrath, J.V.⁴ Kwong, C.D.⁵ Laughon, B.E.⁶ Maddry, J.A.⁷ Mehta, A.⁸ Rasmussen, L.⁹ Reynolds, R.C.¹⁰ Secrist, J.A.¹¹ Shindo, N.¹² Showe, D.N.¹³ Sosa, E.¹⁴ Suling, W.J.¹⁵ White, E.L.¹⁶

14
- 84885177568
- A. Meisnner, H.I. Boschoff, M. Vasan, B.P. Duckworth, C.E. Barry III, and C.C. Aldrich Biorg. Med. Chem. 21 2013 6385
- (2013) Biorg. Med. Chem. , vol.21 , pp. 6385
- Meisnner, A.¹ Boschoff, H.I.² Vasan, M.³ Duckworth, B.P.⁴ Barry III, C.E.⁵ Aldrich, C.C.⁶

15
- 0035289779
- C.A. Lipinski, F. Lombardo, B.W. Dominy, and P.J. Feeney Adv. Drug Delivery Rev. 46 2001 3
- (2001) Adv. Drug Delivery Rev. , vol.46 , pp. 3
- Lipinski, C.A.¹ Lombardo, F.² Dominy, B.W.³ Feeney, P.J.⁴

16
- 2642513322
- L. Di, E.H. Kerns, N. Gao, S.Q. Li, Y. Huang, J.L. Bourassa, and D.M. Huryn J. Pharm. Sci. 93 2004 1537
- (2004) J. Pharm. Sci. , vol.93 , pp. 1537
- Di, L.¹ Kerns, E.H.² Gao, N.³ Li, S.Q.⁴ Huang, Y.⁵ Bourassa, J.L.⁶ Huryn, D.M.⁷

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.