SCOPUS 정보 검색 플랫폼

Volumn 5, Issue 1, 2014, Pages 41-46

Novel pyrazolo[1,5-a]pyridines as PI3K inhibitors: Variation of the central linker group

(19) Kendall, Jackie D a,b Marshall, Andrew J a Giddens, Anna C a Tsang, Kit Yee a,d Boyd, Maruta a Frédérick, Raphaël a,e Lill, Claire L c Lee, Woo Jeong c Kolekar, Sharada c Chao, Mindy c Malik, Alisha c Yu, Shuqiao c Chaussade, Claire b,c,f Buchanan, Christina M b,c Rewcastle, Gordon W a,b Baguley, Bruce C a,b Flanagan, Jack U a,b Denny, William A a,b Shepherd, Peter R b,c

a UNIVERSITY OF AUCKLAND (New Zealand)

b MAURICE WILKINS CENTRE FOR MOLECULAR BIODISCOVERY (New Zealand)

c UNIVERSITY OF AUCKLAND (New Zealand)

d Hong Kong Science Park (Hong Kong)

e UNIVERSITÉ CATHOLIQUE DE LOUVAIN (Belgium)

f UNIVERSITY HOSPITAL OF NICE (France)

Author keywords

[No Author keywords available]

Indexed keywords

2 METHYL 5 NITROPHENYL; 5 BROMOPYRAZOLO[1,5 A]PYRIDINE; 5 CYANOPYRAZOLO[1,5 A]PYRIDINE; BENZENE DERIVATIVE; ENZYME INHIBITOR; HYDRAZIDE; PHOSPHATIDYLINOSITOL 3 KINASE INHIBITOR; PYRAZOLO[1,5 A]PYRIDINE; SULFONOHYDRAZIDE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BINDING SITE; COMPUTER PROGRAM; CONTROLLED STUDY; DRUG EFFECT; DRUG POTENCY; DRUG STRUCTURE; ENZYME INHIBITION; HYDROGEN BOND; IC 50; LIPOPHILICITY; MOLECULAR DYNAMICS; MOLECULAR MODEL; PRIORITY JOURNAL;

EID: 84890813322 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c3md00221g Document Type: Article

Times cited : (17)

References (20)

1
- 77953719346
- S. Shuttleworth F. Silva C. Tomassi A. Cecil T. Hill H. Rogers P. Townsend Prog. Med. Chem. 2009 48 81 131
- (2009) Prog. Med. Chem. , vol.48 , pp. 81-131
- Shuttleworth, S.¹ Silva, F.² Tomassi, C.³ Cecil, A.⁴ Hill, T.⁵ Rogers, H.⁶ Townsend, P.⁷

2
- 79953038262
- M. C. Hollander G. M. Blumenthal P. A. Dennis Nat. Rev. Cancer 2011 11 289 301
- (2011) Nat. Rev. Cancer , vol.11 , pp. 289-301
- Hollander, M.C.¹ Blumenthal, G.M.² Dennis, P.A.³

3
- 62649095679
- C. Chaussade K. Cho C. Mawson G. W. Rewcastle P. R. Shepherd Biochem. Biophys. Res. Commun. 2009 381 577 581
- (2009) Biochem. Biophys. Res. Commun. , vol.381 , pp. 577-581
- Chaussade, C.¹ Cho, K.² Mawson, C.³ Rewcastle, G.W.⁴ Shepherd, P.R.⁵

4
- 77952243758
- J. M. Cleary G. I. Shapiro Curr. Oncol. Rep. 2010 12 87 94
- (2010) Curr. Oncol. Rep. , vol.12 , pp. 87-94
- Cleary, J.M.¹ Shapiro, G.I.²

5
- 68249093818
- P. Liu H. Cheng T. M. Roberts J. J. Zhao Nat. Rev. Drug Discovery 2009 8 627 644
- (2009) Nat. Rev. Drug Discovery , vol.8 , pp. 627-644
- Liu, P.¹ Cheng, H.² Roberts, T.M.³ Zhao, J.J.⁴

6
- 79960794613
- S. Jamieson J. U. Flanagan S. Kolekar C. Buchanan J. D. Kendall W.-J. Lee G. W. Rewcastle W. A. Denny R. Singh J. Dickson B. C. Baguley P. R. Shepherd Biochem. J. 2011 438 53 62
- (2011) Biochem. J. , vol.438 , pp. 53-62
- Jamieson, S.¹ Flanagan, J.U.² Kolekar, S.³ Buchanan, C.⁴ Kendall, J.D.⁵ Lee, W.-J.⁶ Rewcastle, G.W.⁷ Denny, W.A.⁸ Singh, R.⁹ Dickson, J.¹⁰ Baguley, B.C.¹¹ Shepherd, P.R.¹²

7
- 84865060816
- P. Wu Y. Hu Med. Chem. Commun. 2012 3 1337 1355
- (2012) Med. Chem. Commun. , vol.3 , pp. 1337-1355
- Wu, P.¹ Hu, Y.²

8
- 84876731682
- B. Markman J. J. Tao M. Scaltriti Curr. Pharm. Des. 2013 19 895 906
- (2013) Curr. Pharm. Des. , vol.19 , pp. 895-906
- Markman, B.¹ Tao, J.J.² Scaltriti, M.³

9
- 84855202660
- J. D. Kendall P. D. O'Connor A. J. Marshall R. Frédérick E. S. Marshall C. L. Lill W.-J. Lee S. Kolekar M. Chao A. Malik S. Yu C. Chaussade C. Buchanan G. W. Rewcastle B. C. Baguley J. U. Flanagan S. M. F. Jamieson W. A. Denny P. R. Shepherd Bioorg. Med. Chem. 2012 20 69 85
- (2012) Bioorg. Med. Chem. , vol.20 , pp. 69-85
- Kendall, J.D.¹ O'Connor, P.D.² Marshall, A.J.³ Frédérick, R.⁴ Marshall, E.S.⁵ Lill, C.L.⁶ Lee, W.-J.⁷ Kolekar, S.⁸ Chao, M.⁹ Malik, A.¹⁰ Yu, S.¹¹ Chaussade, C.¹² Buchanan, C.¹³ Rewcastle, G.W.¹⁴ Baguley, B.C.¹⁵ Flanagan, J.U.¹⁶ Jamieson, S.M.F.¹⁷ Denny, W.A.¹⁸ Shepherd, P.R.¹⁹

10
- 84855202236
- J. D. Kendall A. C. Giddens K. Y. Tsang R. Frédérick E. S. Marshall R. Singh C. L. Lill W.-J. Lee S. Kolekar M. Chao A. Malik S. Yu C. Chaussade C. Buchanan G. W. Rewcastle B. C. Baguley J. U. Flanagan S. M. F. Jamieson W. A. Denny P. R. Shepherd Bioorg. Med. Chem. 2012 20 58 68
- (2012) Bioorg. Med. Chem. , vol.20 , pp. 58-68
- Kendall, J.D.¹ Giddens, A.C.² Tsang, K.Y.³ Frédérick, R.⁴ Marshall, E.S.⁵ Singh, R.⁶ Lill, C.L.⁷ Lee, W.-J.⁸ Kolekar, S.⁹ Chao, M.¹⁰ Malik, A.¹¹ Yu, S.¹² Chaussade, C.¹³ Buchanan, C.¹⁴ Rewcastle, G.W.¹⁵ Baguley, B.C.¹⁶ Flanagan, J.U.¹⁷ Jamieson, S.M.F.¹⁸ Denny, W.A.¹⁹ Shepherd, P.R.²⁰ more..

11
- 0020325715
- S. D. Nelson J. Med. Chem. 1982 25 753 765
- (1982) J. Med. Chem. , vol.25 , pp. 753-765
- Nelson, S.D.¹

12
- 33750953816
- M. Hayakawa H. Kaizawa K.-i. Kawaguchi N. Ishikawa T. Koizumi T. Ohishi M. Yamano M. Okada M. Ohta S.-i. Tsukamoto F. I. Raynaud M. D. Waterfield P. Parker P. Workman Bioorg. Med. Chem. 2007 15 403 412
- (2007) Bioorg. Med. Chem. , vol.15 , pp. 403-412
- Hayakawa, M.¹ Kaizawa, H.² Kawaguchi, K.-I.³ Ishikawa, N.⁴ Koizumi, T.⁵ Ohishi, T.⁶ Yamano, M.⁷ Okada, M.⁸ Ohta, M.⁹ Tsukamoto, S.-I.¹⁰ Raynaud, F.I.¹¹ Waterfield, M.D.¹² Parker, P.¹³ Workman, P.¹⁴

13
- 75349106113
- A. Berndt S. Miller O. Williams D. D. Le B. T. Houseman J. I. Pacold F. Gorrec W.-C. Hon Y. Liu C. Rommel P. Gaillard T. Rückle M. K. Schwarz K. M. Shokat J. P. Shaw R. L. Williams Nat. Chem. Biol. 2010 6 117 124
- (2010) Nat. Chem. Biol. , vol.6 , pp. 117-124
- Berndt, A.¹ Miller, S.² Williams, O.³ Le, D.D.⁴ Houseman, B.T.⁵ Pacold, J.I.⁶ Gorrec, F.⁷ Hon, W.-C.⁸ Liu, Y.⁹ Rommel, C.¹⁰ Gaillard, P.¹¹ Rückle, T.¹² Schwarz, M.K.¹³ Shokat, K.M.¹⁴ Shaw, J.P.¹⁵ Williams, R.L.¹⁶

14
- 0031024171
- C. A. Lipinski F. Lombardo B. W. Dominy P. J. Feeney Adv. Drug Delivery Rev. 1997 23 3 25
- (1997) Adv. Drug Delivery Rev. , vol.23 , pp. 3-25
- Lipinski, C.A.¹ Lombardo, F.² Dominy, B.W.³ Feeney, P.J.⁴

15
- 31544478015
- B. Kaboudin D. Elhamifar Synthesis 2006 224 226
- (2006) Synthesis , pp. 224-226
- Kaboudin, B.¹ Elhamifar, D.²

16
- 0005818844
- M. Yokoyama H. Hatanaka Synthesis 1985 891 892
- (1985) Synthesis , pp. 891-892
- Yokoyama, M.¹ Hatanaka, H.²

17
- 84993896467
- C. R. Rasmussen F. J. Villani L. E. Weaner B. E. Reynolds A. R. Hood L. R. Hecker S. O. Nortey A. Hanslin M. J. Costanzo E. T. Powell A. J. Molinari Synthesis 1988 456 459
- (1988) Synthesis , pp. 456-459
- Rasmussen, C.R.¹ Villani, F.J.² Weaner, L.E.³ Reynolds, B.E.⁴ Hood, A.R.⁵ Hecker, L.R.⁶ Nortey, S.O.⁷ Hanslin, A.⁸ Costanzo, M.J.⁹ Powell, E.T.¹⁰ Molinari, A.J.¹¹

18
- 65249135408
- S. Mahboobi S. Dove A. Sellmer M. Winkler E. Eichhorn H. Pongratz T. Ciossek T. Baer T. Maier T. Beckers J. Med. Chem. 2009 52 2265 2279
- (2009) J. Med. Chem. , vol.52 , pp. 2265-2279
- Mahboobi, S.¹ Dove, S.² Sellmer, A.³ Winkler, M.⁴ Eichhorn, E.⁵ Pongratz, H.⁶ Ciossek, T.⁷ Baer, T.⁸ Maier, T.⁹ Beckers, T.¹⁰

19
- 34250202514
- H. Prokopcová C. O. Kappe J. Org. Chem. 2007 72 4440 4448
- (2007) J. Org. Chem. , vol.72 , pp. 4440-4448
- Prokopcová, H.¹ Kappe, C.O.²

20
- 34250704713
- C. Chaussade G. W. Rewcastle J. D. Kendall W. A. Denny K. Cho L. M. Gronning M. L. Chong S. H. Anagnostou S. P. Jackson N. Daniele P. R. Shepherd Biochem. J. 2007 404 449 458
- (2007) Biochem. J. , vol.404 , pp. 449-458
- Chaussade, C.¹ Rewcastle, G.W.² Kendall, J.D.³ Denny, W.A.⁴ Cho, K.⁵ Gronning, L.M.⁶ Chong, M.L.⁷ Anagnostou, S.H.⁸ Jackson, S.P.⁹ Daniele, N.¹⁰ Shepherd, P.R.¹¹

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