메뉴 건너뛰기




Volumn 68, Issue 3, 2014, Pages 401-408

Microwave-assisted synthesis and antibacterial activity of derivatives of 3-[1-(4-fluorobenzyl)-1H-indol-3-yl]-5-(4-fluorobenzylthio)-4H-1,2, 4-triazol-4-amine

Author keywords

antibacterial activity; indole; microwave synthesis; Schiff base; triazole

Indexed keywords


EID: 84890119397     PISSN: 03666352     EISSN: 13369075     Source Type: Journal    
DOI: 10.2478/s11696-013-0461-2     Document Type: Article
Times cited : (12)

References (22)
  • 1
    • 80054909846 scopus 로고    scopus 로고
    • 1,3-Dihydro-2H-indol-2-ones derivatives: Design, synthesis, in vitro antibacterial, antifungal and antitubercular study
    • 10.1016/j.ejmech.2011.09.023 1:CAS:528:DC%2BC3MXhtlKkurzI
    • Akhaja, T. N.; & Raval, J. P. (2011). 1,3-Dihydro-2H-indol-2-ones derivatives: Design, synthesis, in vitro antibacterial, antifungal and antitubercular study. European Journal of Medicinal Chemistry, 46, 5573-5579. DOI: 10.1016/j.ejmech.2011.09.023.
    • (2011) European Journal of Medicinal Chemistry , vol.46 , pp. 5573-5579
    • Akhaja, T.N.1    Raval, J.P.2
  • 2
    • 84859005110 scopus 로고    scopus 로고
    • Design, synthesis, in vitro evaluation of tetrahydropyrimidine-isatin hybrids as potential antibacterial, antifungal and anti-tubercular agents
    • 10.1016/j.cclet.2012.01.040 1:CAS:528:DC%2BC38XksVyqt70%3D
    • Akhaja, T. N.; & Raval, J. P. (2012). Design, synthesis, in vitro evaluation of tetrahydropyrimidine-isatin hybrids as potential antibacterial, antifungal and anti-tubercular agents. Chinese Chemical Letters, 23, 446-449. DOI: 10.1016/j.cclet.2012.01.040.
    • (2012) Chinese Chemical Letters , vol.23 , pp. 446-449
    • Akhaja, T.N.1    Raval, J.P.2
  • 4
    • 73549100860 scopus 로고    scopus 로고
    • Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2,4-disubstituted thiazole ring
    • 10.1016/j.ejmech.2009.11.008 1:CAS:528:DC%2BC3cXos1SgtA%3D%3D
    • Bharti, S. K.; Nath, G.; Tilak, R.; & Singh, S. K. (2010). Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2,4-disubstituted thiazole ring. European Journal of Medicinal Chemistry, 45, 651-660. DOI: 10.1016/j.ejmech.2009.11.008.
    • (2010) European Journal of Medicinal Chemistry , vol.45 , pp. 651-660
    • Bharti, S.K.1    Nath, G.2    Tilak, R.3    Singh, S.K.4
  • 7
    • 70349976957 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activities of novel quinoline derivatives carrying 1,2,4-triazole moiety
    • 10.1016/j.ejmech.2009.06.031 1:CAS:528:DC%2BD1MXht1GgtbvE
    • Eswaran, S.; Adhikari, A. V.; & Shetty, N. S. (2009). Synthesis and antimicrobial activities of novel quinoline derivatives carrying 1,2,4-triazole moiety. European Journal of Medicinal Chemistry, 44, 4637-4647. DOI: 10.1016/j.ejmech.2009.06. 031.
    • (2009) European Journal of Medicinal Chemistry , vol.44 , pp. 4637-4647
    • Eswaran, S.1    Adhikari, A.V.2    Shetty, N.S.3
  • 8
    • 2142806013 scopus 로고    scopus 로고
    • Synthesis, reactions and antimicrobial activity of some new indolyl-1,3,4-oxadiazole, triazole and pyrazole derivatives
    • Farghaly, A. R. A. H. (2004). Synthesis, reactions and antimicrobial activity of some new indolyl-1,3,4-oxadiazole, triazole and pyrazole derivatives. Journal of the Chinese Chemical Society, 51, 147-156.
    • (2004) Journal of the Chinese Chemical Society , vol.51 , pp. 147-156
    • Farghaly, A.R.A.H.1
  • 9
    • 77957968194 scopus 로고    scopus 로고
    • Supranational surveillance of antimicrobial resistance: The legacy of the last decade and proposals for the future
    • 10.1016/j.drup.2010.08.002
    • Giske, C. G.; & Cornaglia, G. (2010). Supranational surveillance of antimicrobial resistance: The legacy of the last decade and proposals for the future. Drug Resistance Updates, 13, 93-98. DOI: 10.1016/j.drup.2010.08.002.
    • (2010) Drug Resistance Updates , vol.13 , pp. 93-98
    • Giske, C.G.1    Cornaglia, G.2
  • 10
    • 23244455993 scopus 로고    scopus 로고
    • Microwave-assisted cyclocondensation of hydrazine derivatives with alkyl dihalides or ditosylates in aqueous media: Syntheses of pyrazole, pyrazolidine and phthalazine derivatives
    • 10.1016/j.tetlet.2005.07.018 1:CAS:528:DC%2BD2MXntVygu7c%3D
    • Ju, Y. H.; & Varma, R. S. (2005). Microwave-assisted cyclocondensation of hydrazine derivatives with alkyl dihalides or ditosylates in aqueous media: syntheses of pyrazole, pyrazolidine and phthalazine derivatives. Tetrahedron Letters, 46, 6011-6014. DOI: 10.1016/j.tetlet.2005.07. 018.
    • (2005) Tetrahedron Letters , vol.46 , pp. 6011-6014
    • Ju, Y.H.1    Varma, R.S.2
  • 11
    • 77957848201 scopus 로고    scopus 로고
    • Efficient synthesis of novel 1,2,4-triazole fused acyclic and 21-28 membered macrocyclic and/or lariat macrocyclic oxaazathia crown compounds with potential antimicrobial activity
    • 10.1016/j.ejmech.2010.08.046 1:CAS:528:DC%2BC3cXht1KrtrfN
    • Khalil, N. S. A. M. (2010). Efficient synthesis of novel 1,2,4-triazole fused acyclic and 21-28 membered macrocyclic and/or lariat macrocyclic oxaazathia crown compounds with potential antimicrobial activity. European Journal of Medicinal Chemistry, 45, 5265-5277. DOI: 10.1016/j.ejmech.2010.08. 046.
    • (2010) European Journal of Medicinal Chemistry , vol.45 , pp. 5265-5277
    • Khalil, N.S.A.M.1
  • 12
    • 79956213779 scopus 로고    scopus 로고
    • Longterm environmental monitoring of persistent organic pollutants and metals in a chemical/petrochemical area: Human health risks
    • 10.1016/j.envpol.2011.04.007 1:CAS:528:DC%2BC3MXmsVajur4%3D
    • Nadal, M.; Schuhmacher, M.; & Domingo, J. L. (2011). Longterm environmental monitoring of persistent organic pollutants and metals in a chemical/petrochemical area: Human health risks. Environmental Pollution, 159, 1769-1777. DOI: 10.1016/j.envpol.2011.04.007.
    • (2011) Environmental Pollution , vol.159 , pp. 1769-1777
    • Nadal, M.1    Schuhmacher, M.2    Domingo, J.L.3
  • 14
    • 78651379302 scopus 로고    scopus 로고
    • Screening for potential antimicrobial activities of some cationic uracil biocides against wide-spreading bacterial strains
    • 10.1007/s11743-010-1229-0 1:CAS:528:DC%2BC3cXhtFOisLfM
    • Negm, N. A.; Aiad, I. A.; & Tawfik, S. M. (2010). Screening for potential antimicrobial activities of some cationic uracil biocides against wide-spreading bacterial strains. Journal of Surfactants and Detergents, 13, 503-511. DOI: 10.1007/s11743-010-1229-0.
    • (2010) Journal of Surfactants and Detergents , vol.13 , pp. 503-511
    • Negm, N.A.1    Aiad, I.A.2    Tawfik, S.M.3
  • 15
    • 80054782764 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of some novel triazol-3-ones as antimicrobial agents
    • 10.1016/j.bmcl.2011.08.049 1:CAS:528:DC%2BC3MXht12jtrvJ
    • Pardeshi, S.; & Bobade, V. D. (2011). Synthesis and biological evaluation of some novel triazol-3-ones as antimicrobial agents. Bioorganic & Medicinal Chemistry Letters, 21, 6559-6562. DOI: 10.1016/j.bmcl.2011.08. 049.
    • (2011) Bioorganic & Medicinal Chemistry Letters , vol.21 , pp. 6559-6562
    • Pardeshi, S.1    Bobade, V.D.2
  • 16
    • 77954314818 scopus 로고    scopus 로고
    • Synthesis, characterization and antimicrobial studies of 2-(4-methoxy-phenyl)-5-methyl-4-(2-arylsulfanyl-ethyl)-2,4-dihydro-[1,2,4]triaz olo-3-ones and their corresponding sulfones
    • 10.1016/j.ejmech.2010.04.016 1:CAS:528:DC%2BC3cXnsVSqu78%3D
    • Patil, B. S.; Krishnamurthy, G.; Naik, H. S. B.; Latthe, P. R.; & Ghate, M. (2010). Synthesis, characterization and antimicrobial studies of 2-(4-methoxy-phenyl)-5-methyl-4-(2-arylsulfanyl-ethyl)-2,4-dihydro-[1,2,4]triaz olo-3-ones and their corresponding sulfones. European Journal of Medicinal Chemistry, 45, 3329-3334. DOI: 10.1016/j.ejmech.2010.04.016.
    • (2010) European Journal of Medicinal Chemistry , vol.45 , pp. 3329-3334
    • Patil, B.S.1    Krishnamurthy, G.2    Naik, H.S.B.3    Latthe, P.R.4    Ghate, M.5
  • 17
    • 80054788099 scopus 로고    scopus 로고
    • Iodine-catalyzed conjugate addition of indoles onto en-1,4-dione: A novel synthesis of 3-(1-(1H-indol-3-yl)-2-oxo-2-phenylethyl)indolin-2-ones as antibacterial and antifungal agents
    • 10.1016/j.bmcl.2011.08.075 1:CAS:528:DC%2BC3MXht12jtrrK
    • Reddy, B. V. S.; Rajeswari, N.; Sarangapani, M.; Reddy, G. R.; Madan, C.; Kumar, K. P.; & Rao, M. S. (2011). Iodine-catalyzed conjugate addition of indoles onto en-1,4-dione: A novel synthesis of 3-(1-(1H-indol-3-yl)-2-oxo-2- phenylethyl)indolin-2-ones as antibacterial and antifungal agents. Bioorganic & Medicinal Chemistry Letters, 21, 6510-6514. DOI: 10.1016/j.bmcl.2011.08. 075.
    • (2011) Bioorganic & Medicinal Chemistry Letters , vol.21 , pp. 6510-6514
    • Reddy, B.V.S.1    Rajeswari, N.2    Sarangapani, M.3    Reddy, G.R.4    Madan, C.5    Kumar, K.P.6    Rao, M.S.7
  • 18
    • 79951827384 scopus 로고    scopus 로고
    • Synthesis of new Schiff bases derived from dimers of 4-amino-3-(1- naphthyl)-5-thiomethyl-1,2,4-triazole using microwave irradiation
    • 10.3184/174751911X12964930076647 1:CAS:528:DC%2BC3MXivVOisro%3D
    • Shi, Y.; Peng, Y. L.; Zhao, Z. G.; Li, G. H.; & Li, H. R. (2011). Synthesis of new Schiff bases derived from dimers of 4-amino-3-(1-naphthyl)-5- thiomethyl-1,2,4-triazole using microwave irradiation. Journal of Chemical Research, 35, 15-17. DOI: 10.3184/174751911x12964930076647.
    • (2011) Journal of Chemical Research , vol.35 , pp. 15-17
    • Shi, Y.1    Peng, Y.L.2    Zhao, Z.G.3    Li, G.H.4    Li, H.R.5
  • 19
    • 84860321828 scopus 로고    scopus 로고
    • Cobalt, nickel, copper and zinc complexes with 1,3-diphenyl-1H-pyrazole- 4-carboxaldehyde Schiff bases: Antimicrobial, spectroscopic, thermal and fluorescence studies
    • 10.1016/j.ejmech.2012.02.053 1:CAS:528:DC%2BC38XmtlSks74%3D
    • Singh, K.; Kumar, Y.; Puri, P.; Kumar, M.; & Sharma, C. (2012). Cobalt, nickel, copper and zinc complexes with 1,3-diphenyl-1H-pyrazole-4- carboxaldehyde Schiff bases: Antimicrobial, spectroscopic, thermal and fluorescence studies. European Journal of Medicinal Chemistry, 52, 313-321. DOI: 10.1016/j.ejmech.2012.02.053.
    • (2012) European Journal of Medicinal Chemistry , vol.52 , pp. 313-321
    • Singh, K.1    Kumar, Y.2    Puri, P.3    Kumar, M.4    Sharma, C.5
  • 20
    • 80052578837 scopus 로고    scopus 로고
    • Synthesis, antibacterial activities and molecular docking studies of Schiff bases derived from N-(2/4-benzaldehyde-amino) phenyl-N-phenylthiourea
    • 10.1016/j.bmc.2011.06.077 1:CAS:528:DC%2BC3MXhtFKhsrzE
    • Zhang, H. J.; Qin, X.; Liu, K.; Zhu, D. D.; Wang, X. M.; & Zhu, H. L. (2011). Synthesis, antibacterial activities and molecular docking studies of Schiff bases derived from N-(2/4-benzaldehyde-amino) phenyl-N-phenylthiourea. Bioorganic & Medicinal Chemistry, 19, 5708-5715. DOI: 10.1016/j.bmc.2011.06. 077.
    • (2011) Bioorganic & Medicinal Chemistry , vol.19 , pp. 5708-5715
    • Zhang, H.J.1    Qin, X.2    Liu, K.3    Zhu, D.D.4    Wang, X.M.5    Zhu, H.L.6
  • 21
    • 77958077980 scopus 로고    scopus 로고
    • Microwave-assisted synthesis of new steroidal thiosemicarbazones derived from methyl 3-oxocholanate under solventfree conditions
    • 10.3184/030823410X12798092457988 1:CAS:528:DC%2BC3cXhtlWls7rP
    • Zhao, Z. G.; Liu, X. L.; Liu, L. L.; & Li, G. H. (2010). Microwave-assisted synthesis of new steroidal thiosemicarbazones derived from methyl 3-oxocholanate under solventfree conditions. Journal of Chemical Research, 34, 455-458. DOI: 10.3184/030823410x12798092457988.
    • (2010) Journal of Chemical Research , vol.34 , pp. 455-458
    • Zhao, Z.G.1    Liu, X.L.2    Liu, L.L.3    Li, G.H.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.