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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 24, 2013, Pages 6923-6927

Oxime-based inhibitors of glucose transporter 1 displaying antiproliferative effects in cancer cells

(10) Tuccinardi, Tiziano a Granchi, Carlotta a Iegre, Jessica a Paterni, Ilaria a Bertini, Simone a MacChia, Marco a Martinelli, Adriano a Qian, Yanrong b Chen, Xiaozhuo b Minutolo, Filippo a

a UNIVERSITY OF PISA (Italy)

b OHIO UNIVERSITY (United States)

Author keywords

Cancer; Glucose transporter; Glycolysis; Modeling; Warburg effect

Indexed keywords

ANTINEOPLASTIC AGENT; GLUCOSE; GLUCOSE TRANSPORTER 1; GLUCOSE TRANSPORTER 1 INHIBITOR; HYDROXYL GROUP; OXIME DERIVATIVE; PHLORETIN; UNCLASSIFIED DRUG; WZB 117;

ANTIPROLIFERATIVE ACTIVITY; ARTICLE; CELL VIABILITY; CONTROLLED STUDY; DRUG BINDING SITE; GLUCOSE TRANSPORT; HUMAN; HUMAN CELL; IN VITRO STUDY; LUNG CANCER; MOLECULAR DYNAMICS;

CANCER; GLUCOSE TRANSPORTER; GLYCOLYSIS; MODELING; WARBURG EFFECT;

BINDING SITES; CELL LINE, TUMOR; CELL PROLIFERATION; ESCHERICHIA COLI; ESCHERICHIA COLI PROTEINS; GLUCOSE TRANSPORTER TYPE 1; HUMANS; IMMUNOGLOBULIN G; MELPHALAN; MOLECULAR DOCKING SIMULATION; OXIMES; PROTEIN STRUCTURE, TERTIARY; SYMPORTERS;

EID: 84888869702 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.09.037 Document Type: Article

Times cited : (43)

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