Structural basis of mycobacterial inhibition by Cyclomarin A

Journal of Biological Chemistry

Volumn 288, Issue 43, 2013, Pages 30883-30891

  Vasudevan, Dileep ^a   Rao, Srinivasa P S ^a   Noble, Christian G ^a  

^a NOVARTIS INSTITUTE FOR TROPICAL DISEASES   (Singapore)

Author keywords

[No Author keywords available]

Indexed keywords

COCRYSTAL STRUCTURE; HIGH RESOLUTION; IN-VITRO; MYCOBACTERIAL; N-TERMINAL DOMAINS; PULLDOWN; STRUCTURAL BASIS;

BIOCHEMISTRY; BIOLOGY;

MACHINERY;

CASEINOLYTIC PROTEIN C1; CHAPERONE; CYCLOMARIN A; NATURAL PRODUCT; PHENYLALANINE; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ARTICLE; COMPLEX FORMATION; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG TARGETING; GENE OVEREXPRESSION; IN VITRO STUDY; IN VIVO STUDY; MYCOBACTERIUM BOVIS; MYCOBACTERIUM SMEGMATIS; NONHUMAN; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN DEGRADATION; PROTEIN DOMAIN; STRUCTURE ANALYSIS;

CLPC; CRYSTAL STRUCTURE; CYCLOMARIN; DRUG DISCOVERY; ENZYME INHIBITORS; ENZYMES; NATURAL PRODUCTS;

BACTERIAL PROTEINS; CRYSTALLOGRAPHY, X-RAY; HEAT-SHOCK PROTEINS; MODELS, MOLECULAR; MUTATION; MYCOBACTERIUM TUBERCULOSIS; OLIGOPEPTIDES; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY;

EID: 84886703421     PISSN: 00219258     EISSN: 1083351X     Source Type: Journal    
DOI: 10.1074/jbc.M113.493767     Document Type: Article

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