Screening and evaluation of small organic molecules as ClpB inhibitors and potential antimicrobials

Journal of Medicinal Chemistry

Volumn 56, Issue 18, 2013, Pages 7177-7189

  Martin, Ianire ^a   Underhaug, Jarl ^b   Celaya, Garbiñe ^a   Moro, Fernando ^a   Teigen, Knut ^b   Martinez, Aurora ^b   Muga, Arturo ^a  

^a UNIVERSITY OF THE BASQUE COUNTRY UPV EHU   (Spain)

^b UNIVERSITY OF BERGEN   (Norway)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE TRIPHOSPHATASE; ANTIINFECTIVE AGENT; CHAPERONE; PROTEIN CLPB; PROTEIN CLPB INHIBITOR; PROTEIN INHIBITOR; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; BACTERIAL GROWTH; CONTROLLED STUDY; DRUG DETERMINATION; DRUG PROTEIN BINDING; DRUG SCREENING; ENZYME ACTIVITY; GENE DELETION; GRAM NEGATIVE BACTERIUM; HIGH THROUGHPUT SCREENING; HUMAN; HUMAN CELL; NONHUMAN; OXIDATIVE STRESS; PROTEIN CONFORMATION;

ADENOSINE TRIPHOSPHATASES; ANIMALS; ANTI-INFECTIVE AGENTS; BACTERIAL PROTEINS; CHO CELLS; CRICETINAE; CRICETULUS; DRUG EVALUATION, PRECLINICAL; ESCHERICHIA COLI; GENE DELETION; HEAT-SHOCK PROTEINS; HELA CELLS; HIGH-THROUGHPUT SCREENING ASSAYS; HUMANS; LIGANDS; ORGANIC CHEMICALS; OXIDATIVE STRESS; TEMPERATURE;

EID: 84884992591     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm400499k     Document Type: Article

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