Baicalin and scutellarin are proteasome inhibitors that specifically target chymotrypsin-like catalytic activity

Phytotherapy Research

Volumn 27, Issue 9, 2013, Pages 1362-1367

  Wu, Yi Xin ^a   Sato, Eiji ^a   Kimura, Wataru ^a   Miura, Naoyuki ^a  

^a HAMAMATSU UNIVERSITY SCHOOL OF MEDICINE   (Japan)

Author keywords

baicalin; flavonoid; inhibitor; proteasome; scutellarin

Indexed keywords

BAICALIN; CHYMOTRYPSIN; PEPTIDYLGLUTAMYL PEPTIDE; PROTEASOME; PROTEASOME INHIBITOR; SCUTELLARIN; TRYPSIN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CANCER CELL; CATALYSIS; CONTROLLED STUDY; DRUG EFFECT; DRUG TARGETING; ENZYME INHIBITION; ENZYME SUBSTRATE; ENZYME SUBUNIT; HUMAN; HUMAN CELL; HYDROLYSIS; MOUSE; NONHUMAN;

ERIGERON BREVISCAPUS; MUS; SCUTELLARIA BAICALENSIS;

BAICALIN; FLAVONOID; INHIBITOR; PROTEASOME; SCUTELLARIN;

ANIMALS; APIGENIN; APOPTOSIS; CELL LINE, TUMOR; CELL SURVIVAL; CHYMOTRYPSIN; ERIGERON; FEMALE; FLAVONOIDS; GLUCURONATES; HUMANS; LIVER; MICE; MICE, INBRED ICR; PROTEASOME ENDOPEPTIDASE COMPLEX; PROTEASOME INHIBITORS; SCUTELLARIA BAICALENSIS;

EID: 84883741908     PISSN: 0951418X     EISSN: 10991573     Source Type: Journal    
DOI: 10.1002/ptr.4878     Document Type: Article

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