메뉴 건너뛰기




Volumn 43, Issue 4, 2013, Pages 259-266

Drug release testing methods of polymeric particulate drug formulations

Author keywords

In vitro drug release test; Microparticles; Sustained release formulations

Indexed keywords

ANGIOPEPTIN; BUPIVACAINE; BUSERELIN; BUSERELIN ACETATE; DEXAMETHASONE; EXENDIN 4; LEUPRORELIN; MINOCYCLINE; NALTREXONE; OCTREOTIDE; POLYGLACTIN; POLYMER; RISPERIDONE; TRIPTORELIN;

EID: 84880677157     PISSN: 20935552     EISSN: 20936214     Source Type: Journal    
DOI: 10.1007/s40005-013-0072-5     Document Type: Review
Times cited : (42)

References (49)
  • 1
    • 84865378492 scopus 로고    scopus 로고
    • Development of biodegradable in situ implant and microparticle injectable formulations for sustained delivery of haloperidol
    • Ahmed TA, Ibrahim HM, Ibrahim F, Samy AM, Kaseem A, Nutan MT, Hussain MD (2012) Development of biodegradable in situ implant and microparticle injectable formulations for sustained delivery of haloperidol. J Pharm Sci 101: 3753-3762.
    • (2012) J Pharm Sci , vol.101 , pp. 3753-3762
    • Ahmed, T.A.1    Ibrahim, H.M.2    Ibrahim, F.3    Samy, A.M.4    Kaseem, A.5    Nutan, M.T.6    Hussain, M.D.7
  • 2
    • 0343247711 scopus 로고    scopus 로고
    • Biodegradation and biocompatibility of PLA and PLGA microspheres
    • Anderson JM, Shive MS (1997) Biodegradation and biocompatibility of PLA and PLGA microspheres. Adv Drug Deliv Rev 28: 5-24.
    • (1997) Adv Drug Deliv Rev , vol.28 , pp. 5-24
    • Anderson, J.M.1    Shive, M.S.2
  • 3
    • 77952241968 scopus 로고    scopus 로고
    • In vitro release behavior and cytotoxicity of doxorubicin-loaded gold nanoparticles in cancerous cells
    • Asadishad B, Vossoughi M, Alamzadeh I (2010) In vitro release behavior and cytotoxicity of doxorubicin-loaded gold nanoparticles in cancerous cells. Biotechnol Lett 32: 649-654.
    • (2010) Biotechnol Lett , vol.32 , pp. 649-654
    • Asadishad, B.1    Vossoughi, M.2    Alamzadeh, I.3
  • 5
    • 0023557345 scopus 로고
    • The preparation and evaluation of drug-containing poly(dl-lactide) microspheres formed by the solvent evaporation method
    • Bodmeier R, McGinity JW (1987) The preparation and evaluation of drug-containing poly(dl-lactide) microspheres formed by the solvent evaporation method. Pharm Res 4: 465-471.
    • (1987) Pharm Res , vol.4 , pp. 465-471
    • Bodmeier, R.1    McGinity, J.W.2
  • 7
    • 84870313070 scopus 로고    scopus 로고
    • Recent advances in PLGA particulate systems for drug delivery
    • Choi JS, Seo K, Yoo JW (2012) Recent advances in PLGA particulate systems for drug delivery. J Pharm Invest 42: 155-163.
    • (2012) J Pharm Invest , vol.42 , pp. 155-163
    • Choi, J.S.1    Seo, K.2    Yoo, J.W.3
  • 8
    • 0000314961 scopus 로고
    • Design and production of single immunization vaccines using polylactide polyglycolide microsphere systems
    • M. F. Powell and M. J. Newman (Eds.), New York: Plenum
    • Cleland JL (1995) Design and production of single immunization vaccines using polylactide polyglycolide microsphere systems. In: Powell MF, Newman MJ (eds) Vaccine Design. Plenum, New York, pp 439-472.
    • (1995) Vaccine Design , pp. 439-472
    • Cleland, J.L.1
  • 9
    • 0028944513 scopus 로고
    • Testing of "in vitro" dissolution behavior of microparticulate drug delivery systems
    • Conti B, Genta I, Giunchedi P, Modena T (1995) Testing of "in vitro" dissolution behavior of microparticulate drug delivery systems. Drug Dev Ind Pharm 21: 1223-1233.
    • (1995) Drug Dev Ind Pharm , vol.21 , pp. 1223-1233
    • Conti, B.1    Genta, I.2    Giunchedi, P.3    Modena, T.4
  • 10
    • 27744494863 scopus 로고    scopus 로고
    • Development of a dialysis in vitro release method for biodegradable microspheres
    • D'Souza SS, DeLuca PP (2005) Development of a dialysis in vitro release method for biodegradable microspheres. AAPS PharmSciTech 6: E323-E328.
    • (2005) AAPS PharmSciTech , vol.6
    • D'Souza, S.S.1    DeLuca, P.P.2
  • 11
    • 33644984488 scopus 로고    scopus 로고
    • Methods to assess in vitro drug release from injectable polymeric particulate systems
    • D'Souza SS, DeLuca PP (2006) Methods to assess in vitro drug release from injectable polymeric particulate systems. Pharm Res 23: 460-474.
    • (2006) Pharm Res , vol.23 , pp. 460-474
    • D'Souza, S.S.1    DeLuca, P.P.2
  • 12
    • 27844439408 scopus 로고    scopus 로고
    • A model-dependent approach to correlate accelerated with real-time release from biodegradable microspheres
    • D'Souza SS, Faraj JA, DeLuca PP (2005) A model-dependent approach to correlate accelerated with real-time release from biodegradable microspheres. AAPS PharmSciTech 6: E553-E564.
    • (2005) AAPS PharmSciTech , vol.6
    • D'Souza, S.S.1    Faraj, J.A.2    DeLuca, P.P.3
  • 13
    • 0029335538 scopus 로고
    • Biodegradable polymers for protein and peptide drug delivery
    • Gombotz WR, Pettit DK (1995) Biodegradable polymers for protein and peptide drug delivery. Bioconjug Chem 6: 332-351.
    • (1995) Bioconjug Chem , vol.6 , pp. 332-351
    • Gombotz, W.R.1    Pettit, D.K.2
  • 14
    • 52449107294 scopus 로고    scopus 로고
    • Ketotifen-loaded microspheres prepared by spray-drying poly(d,l-lactide) and poly(d,l-lactide-co-glycolide) polymers: characterization and in vivo evaluation
    • Guerrero S, Muñíz E, Teijón C, Olmo R, Teijón JM, Blanco MD (2008) Ketotifen-loaded microspheres prepared by spray-drying poly(d, l-lactide) and poly(d, l-lactide-co-glycolide) polymers: characterization and in vivo evaluation. J Pharm Sci 97: 3153-3169.
    • (2008) J Pharm Sci , vol.97 , pp. 3153-3169
    • Guerrero, S.1    Muñíz, E.2    Teijón, C.3    Olmo, R.4    Teijón, J.M.5    Blanco, M.D.6
  • 16
    • 0036709194 scopus 로고    scopus 로고
    • Effect of drug stability on the analysis of release data from controlled release microspheres
    • Kim H, Burgess DJ (2002) Effect of drug stability on the analysis of release data from controlled release microspheres. J Microencapsul 19: 631-640.
    • (2002) J Microencapsul , vol.19 , pp. 631-640
    • Kim, H.1    Burgess, D.J.2
  • 17
    • 0018763038 scopus 로고
    • Problems of dialysis techniques in the study of macromolecule binding of drugs
    • Kinget R, Bontinck AM, Herbots H (1979) Problems of dialysis techniques in the study of macromolecule binding of drugs. Int J Pharm 3: 65-72.
    • (1979) Int J Pharm , vol.3 , pp. 65-72
    • Kinget, R.1    Bontinck, A.M.2    Herbots, H.3
  • 18
    • 40949133332 scopus 로고    scopus 로고
    • PLGA-based drug delivery systems: importance of the type of drug and device geometry
    • Klose D, Siepmann F, Elkharraz K, Siepmann J (2008) PLGA-based drug delivery systems: importance of the type of drug and device geometry. Int J Pharm 354: 95-103.
    • (2008) Int J Pharm , vol.354 , pp. 95-103
    • Klose, D.1    Siepmann, F.2    Elkharraz, K.3    Siepmann, J.4
  • 19
    • 0037123707 scopus 로고    scopus 로고
    • In vivo release of bupivacaine from subcutaneously administered oily solution. Comparison with in vitro release
    • Larsen DB, Joergensen S, Olsen NV, Hansen SH, Larsen C (2002) In vivo release of bupivacaine from subcutaneously administered oily solution. Comparison with in vitro release. J Control Release 81: 145-154.
    • (2002) J Control Release , vol.81 , pp. 145-154
    • Larsen, D.B.1    Joergensen, S.2    Olsen, N.V.3    Hansen, S.H.4    Larsen, C.5
  • 20
    • 71249151006 scopus 로고    scopus 로고
    • Role of in vitro release models in formulation development and quality control of parenteral depots
    • Larsen C, Larsen SW, Jensen H, Yaghmur A, Ostergaard J (2009) Role of in vitro release models in formulation development and quality control of parenteral depots. Expert Opin Drug Deliv 6: 1283-1295.
    • (2009) Expert Opin Drug Deliv , vol.6 , pp. 1283-1295
    • Larsen, C.1    Larsen, S.W.2    Jensen, H.3    Yaghmur, A.4    Ostergaard, J.5
  • 21
    • 0035800238 scopus 로고    scopus 로고
    • Paclitaxel loaded poly(l-lactic acid) microspheres: properties of microspheres made with low molecular weight polymers
    • Liggins RT, Burt HM (2001) Paclitaxel loaded poly(l-lactic acid) microspheres: properties of microspheres made with low molecular weight polymers. Int J Pharm 222: 19-33.
    • (2001) Int J Pharm , vol.222 , pp. 19-33
    • Liggins, R.T.1    Burt, H.M.2
  • 22
    • 12144253184 scopus 로고    scopus 로고
    • Formulation and characterization of triclosan sub-micron emulsions and nanocapsules
    • Maestrelli F, Mura P, Alonso MJ (2004) Formulation and characterization of triclosan sub-micron emulsions and nanocapsules. J Microencapsul 21: 857-864.
    • (2004) J Microencapsul , vol.21 , pp. 857-864
    • Maestrelli, F.1    Mura, P.2    Alonso, M.J.3
  • 23
    • 77954073585 scopus 로고    scopus 로고
    • Use of in vitro-in vivo correlation (IVIVC) to facilitate the development of polymer-based controlled release injectable formulation
    • Mitra A, Wu Y (2010) Use of in vitro-in vivo correlation (IVIVC) to facilitate the development of polymer-based controlled release injectable formulation. Recent Pat Drug Deliv Formul 4: 94-104.
    • (2010) Recent Pat Drug Deliv Formul , vol.4 , pp. 94-104
    • Mitra, A.1    Wu, Y.2
  • 24
    • 38349154138 scopus 로고    scopus 로고
    • Nano/micro technologies for delivering macromolecular therapeutics using poly(d,l-lactide-co-glycolide) and its derivatives
    • Mundargi RC, Babu VR, Rangaswamy V, Patel P, Aminabhavi TM (2008) Nano/micro technologies for delivering macromolecular therapeutics using poly(d, l-lactide-co-glycolide) and its derivatives. J Control Release 125: 193-209.
    • (2008) J Control Release , vol.125 , pp. 193-209
    • Mundargi, R.C.1    Babu, V.R.2    Rangaswamy, V.3    Patel, P.4    Aminabhavi, T.M.5
  • 25
    • 4344596313 scopus 로고    scopus 로고
    • Identification of chemically modified peptide from poly(d,l-lactide-co-glycolide) microspheres under in vitro release conditions
    • Murty SB, Goodman J, Thanoo BC, DeLuca PP (2003) Identification of chemically modified peptide from poly(d, l-lactide-co-glycolide) microspheres under in vitro release conditions. AAPS PharmSciTech 4: E50.
    • (2003) AAPS PharmSciTech , vol.4
    • Murty, S.B.1    Goodman, J.2    Thanoo, B.C.3    DeLuca, P.P.4
  • 26
    • 19344375338 scopus 로고    scopus 로고
    • Impurity formation studies with peptide-loaded polymeric microspheres Part II. In vitro evaluation
    • Murty SB, Na DH, Thanoo BC, DeLuca PP (2005) Impurity formation studies with peptide-loaded polymeric microspheres Part II. In vitro evaluation. Int J Pharm 297: 62-72.
    • (2005) Int J Pharm , vol.297 , pp. 62-72
    • Murty, S.B.1    Na, D.H.2    Thanoo, B.C.3    DeLuca, P.P.4
  • 27
    • 34548279009 scopus 로고    scopus 로고
    • In vitro release study of mono-PEGylated growth hormone-releasing peptide-6 from PLGA microspheres
    • Park EJ, Na DH, Lee KC (2007) In vitro release study of mono-PEGylated growth hormone-releasing peptide-6 from PLGA microspheres. Int J Pharm 343: 281-283.
    • (2007) Int J Pharm , vol.343 , pp. 281-283
    • Park, E.J.1    Na, D.H.2    Lee, K.C.3
  • 28
    • 15544385237 scopus 로고    scopus 로고
    • Biodegradable polymers for microencapsulation of drugs
    • Park JH, Ye M, Park K (2005) Biodegradable polymers for microencapsulation of drugs. Molecules 10: 146-161.
    • (2005) Molecules , vol.10 , pp. 146-161
    • Park, J.H.1    Ye, M.2    Park, K.3
  • 29
    • 84878998624 scopus 로고    scopus 로고
    • Long-acting injectable formulations of antipsychotic drugs for the treatment of schizophrenia
    • doi:10.1007/s12272-013-0105-7
    • Park EJ, Amatya S, Kim MS, Park JH, Seol E, Lee H, Shin YH, Na DH (2013) Long-acting injectable formulations of antipsychotic drugs for the treatment of schizophrenia. Arch Pharm Res. doi: 10. 1007/s12272-013-0105-7.
    • (2013) Arch Pharm Res
    • Park, E.J.1    Amatya, S.2    Kim, M.S.3    Park, J.H.4    Seol, E.5    Lee, H.6    Shin, Y.H.7    Na, D.H.8
  • 30
    • 0041666519 scopus 로고    scopus 로고
    • Assessment of drug salt release from solutions, suspensions and in situ suspensions using a rotating dialysis cell
    • Parshad H, Frydenvang K, Liljefors T, Cornett C, Larsen C (2003) Assessment of drug salt release from solutions, suspensions and in situ suspensions using a rotating dialysis cell. Eur J Pharm Sci 19: 263-272.
    • (2003) Eur J Pharm Sci , vol.19 , pp. 263-272
    • Parshad, H.1    Frydenvang, K.2    Liljefors, T.3    Cornett, C.4    Larsen, C.5
  • 31
    • 79955015946 scopus 로고    scopus 로고
    • USP apparatus 4 method for in vitro release testing of protein loaded microspheres
    • Rawat A, Burgess DJ (2011) USP apparatus 4 method for in vitro release testing of protein loaded microspheres. Int J Pharm 409: 178-184.
    • (2011) Int J Pharm , vol.409 , pp. 178-184
    • Rawat, A.1    Burgess, D.J.2
  • 32
    • 80054702104 scopus 로고    scopus 로고
    • Validation of USP apparatus 4 method for microsphere in vitro release testing using Risperdal Consta
    • Rawat A, Stippler E, Shah VP, Burgess DJ (2011) Validation of USP apparatus 4 method for microsphere in vitro release testing using Risperdal Consta. Int J Pharm 420: 198-205.
    • (2011) Int J Pharm , vol.420 , pp. 198-205
    • Rawat, A.1    Stippler, E.2    Shah, V.P.3    Burgess, D.J.4
  • 33
    • 84864134224 scopus 로고    scopus 로고
    • Comparison of in vitro-in vivo release of Risperdal Consta microspheres
    • Rawat A, Bhardwaj U, Burgess DJ (2012) Comparison of in vitro-in vivo release of Risperdal Consta microspheres. Int J Pharm 434: 115-121.
    • (2012) Int J Pharm , vol.434 , pp. 115-121
    • Rawat, A.1    Bhardwaj, U.2    Burgess, D.J.3
  • 34
    • 84855872350 scopus 로고    scopus 로고
    • Effect of agitation regimen on the in vitro release of leuprolide from poly(lactic-co-glycolic) acid microparticles
    • Schoubben A, Blasi P, Deluca PP (2012) Effect of agitation regimen on the in vitro release of leuprolide from poly(lactic-co-glycolic) acid microparticles. J Pharm Sci 101: 1212-1220.
    • (2012) J Pharm Sci , vol.101 , pp. 1212-1220
    • Schoubben, A.1    Blasi, P.2    Deluca, P.P.3
  • 35
    • 0030734317 scopus 로고    scopus 로고
    • Rotating dialysis cell as in vitro release method for oily parenteral depot solutions
    • Schultz K, Møllgaard B, Frokjaer S, Larsen C (1997) Rotating dialysis cell as in vitro release method for oily parenteral depot solutions. Int J Pharm 157: 163-169.
    • (1997) Int J Pharm , vol.157 , pp. 163-169
    • Schultz, K.1    Møllgaard, B.2    Frokjaer, S.3    Larsen, C.4
  • 36
    • 84655170026 scopus 로고    scopus 로고
    • Accelerated in vitro release testing of implantable PLGA microsphere/PVA hydrogel composite coatings
    • Shen J, Burgess DJ (2012) Accelerated in vitro release testing of implantable PLGA microsphere/PVA hydrogel composite coatings. Int J Pharm 422: 341-348.
    • (2012) Int J Pharm , vol.422 , pp. 341-348
    • Shen, J.1    Burgess, D.J.2
  • 37
    • 0342546477 scopus 로고    scopus 로고
    • Diclofenac sodium incorporated PLGA (50:50) microspheres: formulation considerations and in vitro/in vivo evaluation
    • Tunçay M, Caliş S, Kaş HS, Ercan MT, Peksoy I, Hincal AA (2000) Diclofenac sodium incorporated PLGA (50: 50) microspheres: formulation considerations and in vitro/in vivo evaluation. Int J Pharm 195: 179-188.
    • (2000) Int J Pharm , vol.195 , pp. 179-188
    • Tunçay, M.1    Caliş, S.2    Kaş, H.S.3    Ercan, M.T.4    Peksoy, I.5    Hincal, A.A.6
  • 38
    • 0035857705 scopus 로고    scopus 로고
    • Gelatin microspheres crosslinked with d,l-glyceraldehyde as a potential drug delivery system: preparation, characterisation, in vitro and in vivo studies
    • Vandelli MA, Rivasi F, Guerra P, Forni F, Arletti R (2001) Gelatin microspheres crosslinked with d, l-glyceraldehyde as a potential drug delivery system: preparation, characterisation, in vitro and in vivo studies. Int J Pharm 215: 175-184.
    • (2001) Int J Pharm , vol.215 , pp. 175-184
    • Vandelli, M.A.1    Rivasi, F.2    Guerra, P.3    Forni, F.4    Arletti, R.5
  • 39
    • 42649113729 scopus 로고    scopus 로고
    • In situ fiber optic method for long-term in vitro release testing of microspheres
    • Voisine JM, Zolnik BS, Burgess DJ (2008) In situ fiber optic method for long-term in vitro release testing of microspheres. Int J Pharm 356: 206-211.
    • (2008) Int J Pharm , vol.356 , pp. 206-211
    • Voisine, J.M.1    Zolnik, B.S.2    Burgess, D.J.3
  • 40
    • 0028157782 scopus 로고
    • Piroxicam release from spray-dried biodegradable microspheres
    • Wagenaar BW, Müller BW (1994) Piroxicam release from spray-dried biodegradable microspheres. Biomaterials 15: 49-54.
    • (1994) Biomaterials , vol.15 , pp. 49-54
    • Wagenaar, B.W.1    Müller, B.W.2
  • 41
    • 0037151323 scopus 로고    scopus 로고
    • Characterization of the initial burst release of a model peptide from poly(d,l-lactide-co-glycolide) microspheres
    • Wang J, Wang BM, Schwendeman SP (2002) Characterization of the initial burst release of a model peptide from poly(d, l-lactide-co-glycolide) microspheres. J Control Release 82: 289-307.
    • (2002) J Control Release , vol.82 , pp. 289-307
    • Wang, J.1    Wang, B.M.2    Schwendeman, S.P.3
  • 42
    • 0142195953 scopus 로고    scopus 로고
    • The release profiles and bioactivity of parathyroid hormone from poly(lactic-co-glycolic acid) microspheres
    • Wei G, Pettway GJ, McCauley LK, Ma PX (2004) The release profiles and bioactivity of parathyroid hormone from poly(lactic-co-glycolic acid) microspheres. Biomaterials 25: 345-352.
    • (2004) Biomaterials , vol.25 , pp. 345-352
    • Wei, G.1    Pettway, G.J.2    McCauley, L.K.3    Ma, P.X.4
  • 43
    • 55649104973 scopus 로고    scopus 로고
    • Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles
    • Wischke C, Schwendeman SP (2008) Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles. Int J Pharm 364: 298-327.
    • (2008) Int J Pharm , vol.364 , pp. 298-327
    • Wischke, C.1    Schwendeman, S.P.2
  • 44
    • 67749133574 scopus 로고    scopus 로고
    • Preparation of monodisperse biodegradable polymer microparticles using a microfluidic flow-focusing device for controlled drug delivery
    • Xu Q, Hashimoto M, Dang TT, Hoare T, Kohane DS, Whitesides GM, Langer R, Anderson DG (2009) Preparation of monodisperse biodegradable polymer microparticles using a microfluidic flow-focusing device for controlled drug delivery. Small 5: 1575-1581.
    • (2009) Small , vol.5 , pp. 1575-1581
    • Xu, Q.1    Hashimoto, M.2    Dang, T.T.3    Hoare, T.4    Kohane, D.S.5    Whitesides, G.M.6    Langer, R.7    Anderson, D.G.8
  • 45
    • 84862795685 scopus 로고    scopus 로고
    • A two-stage reverse dialysis in vitro dissolution testing method for passive targeted liposomes
    • Xu X, Khan MA, Burgess DJ (2012) A two-stage reverse dialysis in vitro dissolution testing method for passive targeted liposomes. Int J Pharm 426: 211-218.
    • (2012) Int J Pharm , vol.426 , pp. 211-218
    • Xu, X.1    Khan, M.A.2    Burgess, D.J.3
  • 46
    • 0034601882 scopus 로고    scopus 로고
    • Effect of preparation temperature on the characteristics and release profiles of PLGA microspheres containing protein fabricated by double-emulsion solvent extraction/evaporation method
    • Yang YY, Chia HH, Chung TS (2000) Effect of preparation temperature on the characteristics and release profiles of PLGA microspheres containing protein fabricated by double-emulsion solvent extraction/evaporation method. J Control Release 69: 81-96.
    • (2000) J Control Release , vol.69 , pp. 81-96
    • Yang, Y.Y.1    Chia, H.H.2    Chung, T.S.3
  • 47
    • 0035806317 scopus 로고    scopus 로고
    • Controlled release of nalbuphine propionate from biodegradable microspheres: in vitro and in vivo studies
    • Yen SY, Sung KC, Wang JJ, Yoa-Pu Hu O (2001) Controlled release of nalbuphine propionate from biodegradable microspheres: in vitro and in vivo studies. Int J Pharm 220: 91-99.
    • (2001) Int J Pharm , vol.220 , pp. 91-99
    • Yen, S.Y.1    Sung, K.C.2    Wang, J.J.3    Yoa-Pu Hu, O.4
  • 48
    • 41249098853 scopus 로고    scopus 로고
    • Evaluation of in vivo-in vitro release of dexamethasone from PLGA microspheres
    • Zolnik BS, Burgess DJ (2008) Evaluation of in vivo-in vitro release of dexamethasone from PLGA microspheres. J Control Release 127: 137-145.
    • (2008) J Control Release , vol.127 , pp. 137-145
    • Zolnik, B.S.1    Burgess, D.J.2
  • 49
    • 33646676075 scopus 로고    scopus 로고
    • Elevated temperature accelerated release testing of PLGA microspheres
    • Zolnik BS, Leary PE, Burgess DJ (2006) Elevated temperature accelerated release testing of PLGA microspheres. J Control Release 112: 293-300.
    • (2006) J Control Release , vol.112 , pp. 293-300
    • Zolnik, B.S.1    Leary, P.E.2    Burgess, D.J.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.