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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 13, 2013, Pages 3728-3731

Activity-lipophilicity relationship studies on P-gp ligands designed as simplified tariquidar bulky fragments

(8) Contino, Marialessandra a Zinzi, Laura a Cantore, Mariangela a Perrone, Maria Grazia a Leopoldo, Marcello a Berardi, Francesco a Perrone, Roberto a Colabufo, Nicola Antonio a

a UNIVERSITY OF BARI (Italy)

Author keywords

2 Alkyloxyquinoline; BCRP; Lipophilicity; MRP1; P Glycoprotein; Tariquidar

Indexed keywords

ADENOSINE TRIPHOSPHATASE; ADENOSINE TRIPHOSPHATE; ALKYLOXYQUINOLINE DERIVATIVE; BREAST CANCER RESISTANCE PROTEIN; MULTIDRUG RESISTANCE PROTEIN; QUINOLINE DERIVATIVE; TARIQUIDAR; UNCLASSIFIED DRUG;

ARTICLE; CELL LEVEL; CELL MEMBRANE PERMEABILITY; DRUG ACTIVITY; DRUG SYNTHESIS; LIPOPHILICITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; CELL LINE; DOGS; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; LIGANDS; MOLECULAR STRUCTURE; OXYQUINOLINE; P-GLYCOPROTEIN; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84878832186 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.05.019 Document Type: Article

Times cited : (12)

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