SCOPUS 정보 검색 플랫폼

Volumn 11, Issue 19, 2013, Pages 3103-3107

Synthesis and evaluation of 3-amino/guanidine substituted phenyl oxazoles as a novel class of LSD1 inhibitors with anti-proliferative properties

(10) Dulla, Balakrishna a,b Kirla, Krishna Tulasi c Rathore, Vandana c Deora, Girdhar Singh b Kavela, Sridhar d Maddika, Subbareddy d Chatti, Kiranam c Reiser, Oliver a Iqbal, Javed b Pal, Manojit b

a UNIVERSITY OF REGENSBURG (Germany)

b INSTITUTE OF LIFE SCIENCES (India)

c UNIVERSITY OF HYDERABAD (India)

d Center for DNA Fingerprinting and Diagnostics (India)

Author keywords

[No Author keywords available]

Indexed keywords

ANTI-PROLIFERATIVE; BREAST CANCER CELLS; CANCER CELLS; EPIGENETIC MECHANISMS; FUNCTIONALIZED; IN-VITRO; OXAZOLES; ZEBRAFISH EMBRYOS;

CHEMISTRY; POSITIVE IONS;

CELLS;

ANTINEOPLASTIC AGENT; ENZYME INHIBITOR; GUANIDINE; HISTONE DEMETHYLASE; KDM1A PROTEIN, HUMAN; OXAZOLE DERIVATIVE;

ANIMAL; APOPTOSIS; ARTICLE; CELL PROLIFERATION; CELL SURVIVAL; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG ANTAGONISM; DRUG EFFECT; DRUG SCREENING; HUMAN; METABOLISM; MOLECULAR DYNAMICS; STRUCTURE ACTIVITY RELATION; SYNTHESIS; TUMOR CELL LINE; ZEBRA FISH;

ANIMALS; ANTINEOPLASTIC AGENTS; APOPTOSIS; CELL LINE, TUMOR; CELL PROLIFERATION; CELL SURVIVAL; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SCREENING ASSAYS, ANTITUMOR; ENZYME INHIBITORS; GUANIDINE; HISTONE DEMETHYLASES; HUMANS; MOLECULAR DYNAMICS SIMULATION; MOLECULAR STRUCTURE; OXAZOLES; STRUCTURE-ACTIVITY RELATIONSHIP; ZEBRAFISH;

DANIO RERIO;

EID: 84876931561 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/c3ob40217g Document Type: Article

Times cited : (49)

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