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Tetrahedron Letters

Volumn 54, Issue 21, 2013, Pages 2612-2614

Simple approach to the synthesis of 3-fluoro pyrazolo[1,5-a]pyrimidine analogues

(4) Bel Abed, Hassen a Mammoliti, Oscar b Van Lommen, Guy b Herdewijn, Piet a

a REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

b GALAPAGOS NV (Belgium)

Author keywords

Cyclization; Heterocycle; Pyrazole; Pyrazolo 1,5 a pyrimidine

Indexed keywords

3 AMINO 4 FLUORO PYRAZOLE; 3 FLUORO PYRAZOLO[1,5-A]PYRIMIDINE DERIVATIVE; ACETONITRILE DERIVATIVE; BENZENECARBONYL CHLORIDE; CHLORIDE; PYRAZOLE DERIVATIVE; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS;

EID: 84876409858 PISSN: 00404039 EISSN: 18733581 Source Type: Journal
DOI: 10.1016/j.tetlet.2013.03.015 Document Type: Article

Times cited : (23)

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