Chemical tagging of a drug target using 5-sulfonyl tetrazole

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 6, 2013, Pages 1608-1611

  Otsuki, Satsuki ^a   Nishimura, Shinichi ^a   Takabatake, Hisae ^a   Nakajima, Kozue ^a   Takasu, Yasuaki ^a   Yagura, Toru ^a   Sakai, Yuki ^a   Hattori, Akira ^a   Kakeya, Hideaki ^a  

^a KYOTO UNIVERSITY   (Japan)

Author keywords

5 Sulfonyl tetrazole; Bioactive small molecule; Chemical tagging; Receptor protein; Target identification

Indexed keywords

5 SULFONYL TETRAZOLE; CYCLOPHILIN A; CYCLOSPORIN A; LIGAND; RECEPTOR PROTEIN; TETRAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; ATOM; BINDING AFFINITY; CHEMICAL REACTION; CHEMICAL STRUCTURE; CHEMICAL TAGGING; CYCLOADDITION; DRUG TARGETING; MOLECULAR PROBE; NUCLEOPHILICITY; OXIDATION; SIGNAL TRANSDUCTION; SUBSTITUTION REACTION; SYNTHESIS;

CYCLOPHILIN A; CYCLOSPORINE; LIGANDS; PROTEIN BINDING; TETRAZOLES;

EID: 84874654262     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.01.092     Document Type: Article

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