Amiloride derivatives are effective blockers of insect odorant receptors

Chemical Senses

Volumn 38, Issue 3, 2013, Pages 231-236

  Róllecke, Katharina ^a   Werner, Markus ^a   Ziemba, Paul M ^a   Neuhaus, Eva M ^b   Hatt, Hanns ^a   Gisselmann, Günter ^a  

^a RUHR UNIVERSITY BOCHUM   (Germany)

^b CHARITÉ UNIVERSITÄTSMEDIZIN BERLIN   (Germany)

Author keywords

Bombyx mori; Chemosensation; Drosophila melanogaster; Olfaction; Voltage clamp; Xenopus laevis oocytes

Indexed keywords

1 [2 (4 METHOXYPHENYL) 2 [3 (4 METHOXYPHENYL)PROPOXY]ETHYL] 1H IMIDAZOLE; 5 (N ISOBUTYL N METHYL)AMILORIDE; 5 (N,N DIMETHYL)AMILORIDE; 5 (N,N HEXAMETHYLENE)AMILORIDE; AMILORIDE; AMILORIDE DERIVATIVE; DIETHYLTOLUAMIDE; ION CHANNEL; ORCO CHANNEL SUBUNIT; ORCO RECEPTOR; PENTYL ACETATE; RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BOMBYX MORI; CHEMICAL STRUCTURE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DROSOPHILA MELANOGASTER; FEMALE; IC 50; INHIBITION KINETICS; ION CURRENT; NONHUMAN; ODORANT RECEPTOR 1; ODORANT RECEPTOR 47A; ODORANT RECEPTOR 49B; OLFACTORY RECEPTOR; OOCYTE; PRIORITY JOURNAL; RECEPTOR BLOCKING; SIGNAL TRANSDUCTION; VOLTAGE CLAMP; XENOPUS LAEVIS;

AMILORIDE; ANIMALS; BOMBYX; DROSOPHILA MELANOGASTER; ELECTRODES; OOCYTES; PATCH-CLAMP TECHNIQUES; PENTANOLS; RECEPTORS, ODORANT; XENOPUS LAEVIS;

EID: 84874053272     PISSN: 0379864X     EISSN: 14643553     Source Type: Journal    
DOI: 10.1093/chemse/bjs140     Document Type: Article

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