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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 5, 2013, Pages 1557-1563

Synthesis and SAR of 99mTc/Re-labeled small molecule prostate specific membrane antigen inhibitors with novel polar chelates

(7) Lu, Genliang a Maresca, Kevin P a Hillier, Shawn M a Zimmerman, Craig N a Eckelman, William C a Joyal, John L a Babich, John W a

a Clinical Research (United States)

Author keywords

Inhibitor; Polar chelates; PSMA; Rhenium; Structure activity relationships; Technetium

Indexed keywords

AMINO ACID; CHELATE; GLUTAMIC ACID; LYSINE; PROSTATE SPECIFIC MEMBRANE ANTIGEN; RHENIUM TECHNETIUM TC 99M; UREA; CHELATING AGENT; KALLIKREIN; KALLIKREIN-RELATED PEPTIDASE 3, HUMAN; LIGAND; PROSTATE SPECIFIC ANTIGEN; RADIOPHARMACEUTICAL AGENT; RHENIUM; TECHNETIUM COMPLEX; KALLIKREIN RELATED PEPTIDASE 3, HUMAN;

ARTICLE; BINDING AFFINITY; CELL STRAIN LNCAP; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; IN VITRO STUDY; PHARMACOPHORE; STRUCTURE ACTIVITY RELATION; ANTAGONISTS AND INHIBITORS; CHEMISTRY; MALE; METABOLISM; PROSTATE TUMOR; SCINTISCANNING; SYNTHESIS; TISSUE DISTRIBUTION; TUMOR CELL LINE; DRUG ANTAGONISM;

CELL LINE, TUMOR; CHELATING AGENTS; HUMANS; KALLIKREINS; LIGANDS; MALE; ORGANOTECHNETIUM COMPOUNDS; PROSTATE-SPECIFIC ANTIGEN; PROSTATIC NEOPLASMS; RADIOPHARMACEUTICALS; RHENIUM; STRUCTURE-ACTIVITY RELATIONSHIP; TISSUE DISTRIBUTION;

EID: 84873729101 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.09.014 Document Type: Article

Times cited : (77)

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