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Volumn 2, Issue 12, 2011, Pages 1244-1253

A modular strategy to prepare multivalent inhibitors of prostate-specific membrane antigen (PSMA)

Author keywords

Bivalent urea inhibitor; Molecular imaging; Multivalency; Naaladase; Prostate specific membrane antigen (PSMA); SPECT imaging

Indexed keywords

DIAGNOSTIC AGENT; GLUTAMATE CARBOXYPEPTIDASE II; GLUTAMATE CARBOXYPEPTIDASE II, HUMAN; MEMBRANE ANTIGEN; RADIOPHARMACEUTICAL AGENT;

EID: 84862883597     PISSN: None     EISSN: 19492553     Source Type: Journal    
DOI: 10.18632/oncotarget.415     Document Type: Article
Times cited : (49)

References (37)
  • 2
    • 3843113671 scopus 로고    scopus 로고
    • Tumor target prostate specific membrane antigen (PSMA) and its regulation in prostate cancer
    • Ghosh A and Heston WD. Tumor target prostate specific membrane antigen (PSMA) and its regulation in prostate cancer. J Cell Biochem. 2004; 91:528-539.
    • (2004) J Cell Biochem , vol.91 , pp. 528-539
    • Ghosh, A.1    Heston, W.D.2
  • 4
    • 35048823742 scopus 로고    scopus 로고
    • Clinical trials of cancer therapies targeting prostate-specific membrane antigen
    • Olson WC, Heston WD and Rajasekaran AK. Clinical trials of cancer therapies targeting prostate-specific membrane antigen. Rev Recent Clin Trials. 2007; 2:182-190.
    • (2007) Rev Recent Clin Trials , vol.2 , pp. 182-190
    • Olson, W.C.1    Heston, W.D.2    Rajasekaran, A.K.3
  • 6
    • 79959328548 scopus 로고    scopus 로고
    • Noninvasive measurement of androgen receptor signaling with a positron-emitting radiopharmaceutical that targets prostate-specific membrane antigen
    • Evans MJ, Smith-Jones PM, Wongvipat J, Navarro V, Kim S, Bander NH, Larson SM and Sawyers CL. Noninvasive measurement of androgen receptor signaling with a positron-emitting radiopharmaceutical that targets prostate-specific membrane antigen. Proc Natl Acad Sci U S A. 2011; 108:9578-9582.
    • (2011) Proc Natl Acad Sci U S A , vol.108 , pp. 9578-9582
    • Evans, M.J.1    Smith-Jones, P.M.2    Wongvipat, J.3    Navarro, V.4    Kim, S.5    Bander, N.H.6    Larson, S.M.7    Sawyers, C.L.8
  • 7
    • 79960301987 scopus 로고    scopus 로고
    • 123I-MIP-1072, a small-molecule inhibitor of prostate-specific membrane antigen, is effective at monitoring tumor response to taxane therapy
    • Hillier SM, Kern AM, Maresca KP, Marquis JC, Eckelman WC, Joyal JL and Babich JW. 123I-MIP-1072, a small-molecule inhibitor of prostate-specific membrane antigen, is effective at monitoring tumor response to taxane therapy. J Nucl Med. 2011; 52:1087-1093.
    • (2011) J Nucl Med , vol.52 , pp. 1087-1093
    • Hillier, S.M.1    Kern, A.M.2    Maresca, K.P.3    Marquis, J.C.4    Eckelman, W.C.5    Joyal, J.L.6    Babich, J.W.7
  • 15
    • 46749087806 scopus 로고    scopus 로고
    • Characterization of a targeted nanoparticle functionalized with a urea-based inhibitor of prostate-specific membrane antigen (PSMA)
    • Chandran SS, Banerjee SR, Mease RC, Pomper MG and Denmeade SR. Characterization of a targeted nanoparticle functionalized with a urea-based inhibitor of prostate-specific membrane antigen (PSMA). Cancer Biol Ther. 2008; 7:974-982.
    • (2008) Cancer Biol Ther , vol.7 , pp. 974-982
    • Chandran, S.S.1    Banerjee, S.R.2    Mease, R.C.3    Pomper, M.G.4    Denmeade, S.R.5
  • 17
    • 1242330435 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of a (99m)Tc-labelled cyclic RGD peptide for imaging the alphavbeta3 expression
    • Haubner R, Bruchertseifer F, Bock M, Kessler H, Schwaiger M and Wester HJ. Synthesis and biological evaluation of a (99m)Tc-labelled cyclic RGD peptide for imaging the alphavbeta3 expression. Nuklearmedizin. 2004; 43:26-32.
    • (2004) Nuklearmedizin , vol.43 , pp. 26-32
    • Haubner, R.1    Bruchertseifer, F.2    Bock, M.3    Kessler, H.4    Schwaiger, M.5    Wester, H.J.6
  • 18
    • 35948945504 scopus 로고    scopus 로고
    • Adventures in multivalency, the Harry S. Fischer memorial lecture CMR 2005; Evian France
    • Tweedle MF. Adventures in multivalency, the Harry S. Fischer memorial lecture CMR 2005; Evian, France. Contrast Media Mol Imaging. 2006; 1:2-9.
    • (2006) Contrast Media Mol Imaging , vol.1 , pp. 2-9
    • Tweedle, M.F.1
  • 19
    • 80054935311 scopus 로고    scopus 로고
    • Design, synthesis, and biological studies of efficient multivalent melanotropin ligands: tools toward melanoma diagnosis and treatment
    • Brabez N, Lynch RM, Xu L, Gillies RJ, Chassaing G, Lavielle S and Hruby VJ. Design, synthesis, and biological studies of efficient multivalent melanotropin ligands: tools toward melanoma diagnosis and treatment. J Med Chem. 2011; 54:7375-7384.
    • (2011) J Med Chem , vol.54 , pp. 7375-7384
    • Brabez, N.1    Lynch, R.M.2    Xu, L.3    Gillies, R.J.4    Chassaing, G.5    Lavielle, S.6    Hruby, V.J.7
  • 20
    • 70349922812 scopus 로고    scopus 로고
    • Imparting multivalency to a bifunctional chelator: a scaffold design for targeted PET imaging probes
    • Liu W, Hao G, Long MA, Anthony T, Hsieh JT and Sun X. Imparting multivalency to a bifunctional chelator: a scaffold design for targeted PET imaging probes. Angew Chem Int Ed Engl. 2009; 48:7346-7349.
    • (2009) Angew Chem Int Ed Engl , vol.48 , pp. 7346-7349
    • Liu, W.1    Hao, G.2    Long, M.A.3    Anthony, T.4    Hsieh, J.T.5    Sun, X.6
  • 22
    • 60549097550 scopus 로고    scopus 로고
    • Multivalent scaffolds for affinity maturation of small molecule cell surface binders and their application to prostate tumor targeting
    • Humblet V, Misra P, Bhushan KR, Nasr K, Ko YS, Tsukamoto T, Pannier N, Frangioni JV and Maison W. Multivalent scaffolds for affinity maturation of small molecule cell surface binders and their application to prostate tumor targeting. J Med Chem. 2009; 52:544-550.
    • (2009) J Med Chem , vol.52 , pp. 544-550
    • Humblet, V.1    Misra, P.2    Bhushan, K.R.3    Nasr, K.4    Ko, Y.S.5    Tsukamoto, T.6    Pannier, N.7    Frangioni, J.V.8    Maison, W.9
  • 23
    • 36749014055 scopus 로고
    • 1,3-Dipolar Cycloadditions. Past and Future
    • Huisgen R. 1,3-Dipolar Cycloadditions. Past and Future. Angew Chem Int Ed. 1963; 2:565-598.
    • (1963) Angew Chem Int Ed , vol.2 , pp. 565-598
    • Huisgen, R.1
  • 24
    • 0037099395 scopus 로고    scopus 로고
    • A stepwise huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes
    • Rostovtsev VV, Green LG, Fokin VV and Sharpless KB. A stepwise huisgen cycloaddition process: copper(I)- catalyzed regioselective "ligation" of azides and terminal alkynes. Angewandte Chemie (International ed.) 2002; 41:2596-2599.
    • (2002) Angewandte Chemie (International ed. ) , vol.41 , pp. 2596-2599
    • Rostovtsev, V.V.1    Green, L.G.2    Fokin, V.V.3    Sharpless, K.B.4
  • 25
    • 33644700192 scopus 로고    scopus 로고
    • NAAG peptidase inhibitors and their potential for diagnosis and therapy
    • Zhou J, Neale JH, Pomper MG and Kozikowski AP. NAAG peptidase inhibitors and their potential for diagnosis and therapy. Nat Rev Drug Discov. 2005; 4:1015-1026.
    • (2005) Nat Rev Drug Discov , vol.4 , pp. 1015-1026
    • Zhou, J.1    Neale, J.H.2    Pomper, M.G.3    Kozikowski, A.P.4
  • 26
    • 0033168844 scopus 로고    scopus 로고
    • Five different anti-prostate-specific membrane antigen (PSMA) antibodies confirm PSMA expression in tumor-associated neovasculature
    • Chang SS, Reuter VE, Heston WD, Bander NH, Grauer LS and Gaudin PB. Five different anti-prostate-specific membrane antigen (PSMA) antibodies confirm PSMA expression in tumor-associated neovasculature. Cancer Res. 1999; 59:3192-3198.
    • (1999) Cancer Res , vol.59 , pp. 3192-3198
    • Chang, S.S.1    Reuter, V.E.2    Heston, W.D.3    Bander, N.H.4    Grauer, L.S.5    Gaudin, P.B.6
  • 27
  • 28
    • 67249157547 scopus 로고    scopus 로고
    • Prostate-specific membrane antigen targeted imaging and therapy of prostate cancer using a PSMA inhibitor as a homing ligand
    • Kularatne SA, Wang K, Santhapuram HK and Low PS. Prostate-specific membrane antigen targeted imaging and therapy of prostate cancer using a PSMA inhibitor as a homing ligand. Mol Pharmacol. 2009; 6:780-789.
    • (2009) Mol Pharmacol , vol.6 , pp. 780-789
    • Kularatne, S.A.1    Wang, K.2    Santhapuram, H.K.3    Low, P.S.4
  • 29
    • 67249105432 scopus 로고    scopus 로고
    • Design, synthesis, and preclinical evaluation of prostate-specific membrane antigen targeted (99m)Tc-radioimaging agents
    • Kularatne SA, Zhou Z, Yang J, Post CB and Low PS. Design, synthesis, and preclinical evaluation of prostate-specific membrane antigen targeted (99m)Tc-radioimaging agents. Mol Pharmacol. 2009; 6:790-800.
    • (2009) Mol Pharmacol , vol.6 , pp. 790-800
    • Kularatne, S.A.1    Zhou, Z.2    Yang, J.3    Post, C.B.4    Low, P.S.5
  • 32
    • 84868332957 scopus 로고    scopus 로고
    • Preclinical evaluation of 86Y-Labeled inhibitors of prostate specific membrane antigen
    • (19th International Symposium on Radiopharmaceutical Sciences meeting abstract)
    • Banerjee SR, Pullambhatla M, Byun Y, Nimmagadda S, Baidoo KE, Brechbiel MW, Mease RC and Pomper MG. Preclinical evaluation of 86Y-Labeled inhibitors of prostate specific membrane antigen. J Label Compd Radiopharm (19th International Symposium on Radiopharmaceutical Sciences meeting abstract) 2011; 54:S65.
    • (2011) J Label Compd Radiopharm , vol.54
    • Banerjee, S.R.1    Pullambhatla, M.2    Byun, Y.3    Nimmagadda, S.4    Baidoo, K.E.5    Brechbiel, M.W.6    Mease, R.C.7    Pomper, M.G.8
  • 33
    • 13244251095 scopus 로고    scopus 로고
    • New directions in the coordination chemistry of 99mTc: a reflection on technetium core structures and a strategy for new chelate design
    • Banerjee SR, Maresca KP, Francesconi L, Valliant J, Babich JW and Zubieta J. New directions in the coordination chemistry of 99mTc: a reflection on technetium core structures and a strategy for new chelate design. Nucl Med Biol. 2005; 32:1-20.
    • (2005) Nucl Med Biol , vol.32 , pp. 1-20
    • Banerjee, S.R.1    Maresca, K.P.2    Francesconi, L.3    Valliant, J.4    Babich, J.W.5    Zubieta, J.6
  • 34
    • 85039679471 scopus 로고    scopus 로고
    • 99mTc-labeled inhibitors of prostate-specific membrane antigen (PSMA) for imaging prostate cancer
    • (SNM Annual Meeting Abstract)
    • Ray S, Pullambhatla M, Falk A, Byun Y, Foss C, Nimmagadda S, Fox J, Mease R and Pomper M. 99mTc-labeled inhibitors of prostate-specific membrane antigen (PSMA) for imaging prostate cancer. J Nucl Med. (SNM Annual Meeting Abstract). 2011; 52 (Supplement 1): 293.
    • (2011) J Nucl Med , vol.52 , Issue.SUPPL. 1 , pp. 293
    • Ray, S.1    Pullambhatla, M.2    Falk, A.3    Byun, Y.4    Foss, C.5    Nimmagadda, S.6    Fox, J.7    Mease, R.8    Pomper, M.9
  • 35
    • 0014772602 scopus 로고
    • Color test for detection of free terminal amino groups in the solid-phase synthesis of peptides
    • Kaiser E, Colescott RL, Bossinger CD and Cook PI. Color test for detection of free terminal amino groups in the solid-phase synthesis of peptides. Anal Biochem. 1970; 34:595- 598.
    • (1970) Anal Biochem , vol.34 , pp. 595-598
    • Kaiser, E.1    Colescott, R.L.2    Bossinger, C.D.3    Cook, P.I.4
  • 36
    • 0015861774 scopus 로고
    • Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
    • Cheng Y and Prusoff WH. Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction. Biochem Pharmacol. 1973; 22:3099-3108.
    • (1973) Biochem Pharmacol , vol.22 , pp. 3099-3108
    • Cheng, Y.1    Prusoff, W.H.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.