Identification and characterization of novel human glucose-6-phosphate dehydrogenase inhibitors

Journal of Biomolecular Screening

Volumn 18, Issue 3, 2013, Pages 286-297

  Preuss, Janina ^a,b,c   Richardson, Adam D ^b   Pinkerton, Anthony ^b   Hedrick, Michael ^b   Sergienko, Eduard ^b   Rahlfs, Stefan ^c   Becker, Katja ^c   Bode, Lars ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b BURNHAM INSTITUTE   (United States)

^c JUSTUS LIEBIG UNIVERSITY   (Germany)

Author keywords

glucose 6 phosphate dehydrogenase; high throughput screening; MCF10; pentose phosphate pathway; redox metabolism

Indexed keywords

6 AMINONICOTINAMIDE; GLUCOSE 6 PHOSPHATE DEHYDROGENASE; OXIDOREDUCTASE INHIBITOR; PRASTERONE;

ARTICLE; BREAST CARCINOMA; CANCER CELL CULTURE; CELL VIABILITY; CONTROLLED STUDY; DRUG DETERMINATION; DRUG PENETRATION; DRUG POTENCY; DRUG PURIFICATION; DRUG SCREENING; DRUG SOLUBILITY; ENZYME INHIBITION; FALSE POSITIVE RESULT; GENE OVEREXPRESSION; HIGH THROUGHPUT SCREENING; IC 50; PRIORITY JOURNAL;

6-AMINONICOTINAMIDE; CELL LINE, TUMOR; DEHYDROEPIANDROSTERONE; ENZYME INHIBITORS; GLUCOSEPHOSPHATE DEHYDROGENASE; HIGH-THROUGHPUT SCREENING ASSAYS; HUMANS; INHIBITORY CONCENTRATION 50; SMALL MOLECULE LIBRARIES;

EID: 84873615866     PISSN: 10870571     EISSN: 1552454X     Source Type: Journal    
DOI: 10.1177/1087057112462131     Document Type: Article

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