The development of potential new fluorine-18 labelled radiotracers for imaging the GABAA receptor

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 3, 2013, Pages 821-826

  Jackson, Alexander ^a   Guilbert, Benedicte B ^a   Plant, Stuart D ^a   Goggi, Julian ^a   Battle, Mark R ^a   Woodcraft, John L ^a   Gaeta, Alessandra ^a   Jones, Clare L ^a   Bouvet, Denis R ^a   Jones, Paul A ^a   O'Shea, Dennis M ^a   Zheng, Penny Hao ^a   Brown, Samantha L ^a   Ewan, Amanda L ^a   Trigg, William ^a  

^a GE HEALTHCARE   (United Kingdom)

Author keywords

Benzodiazepine; FASTlab; Flumazenil; GABAA; GE 194; PET

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; BRETAZENIL; FLUMAZENIL C 11; FLUMAZENIL DERIVATIVE F 18; FLUMAZENIL F 18; FLUORINE 18; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; IN VITRO STUDY; POSITRON EMISSION TOMOGRAPHY; RADIOCHEMISTRY;

FLUMAZENIL; FLUORINE RADIOISOTOPES; HUMANS; POSITRON-EMISSION TOMOGRAPHY; RADIOPHARMACEUTICALS; RECEPTORS, GABA-A; SMALL MOLECULE LIBRARIES;

EID: 84872350543     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.11.066     Document Type: Article

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