메뉴 건너뛰기




Volumn 136, Issue 5, 2012, Pages 808-814

Activity of 5-chloro-pyrazinamide in mice infected with Mycobacterium tuberculosis or Mycobacterium bovis

Author keywords

Experimental chemotherapy; Mouse; Pyrazinamide; Tuberculosis

Indexed keywords

5 CHLORO PYRAZINAMIDE; ISONIAZID; PYRAZINAMIDE; RIFAMPICIN; UNCLASSIFIED DRUG;

EID: 84872087742     PISSN: 09715916     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (16)

References (20)
  • 1
    • 51149085652 scopus 로고    scopus 로고
    • Enhancement of the antituberculosis activity of weak acids by inhibitors of energy metabolism but not by anaerobiosis suggests that weak acids act differently from the front-line tuberculosis drug pyrazinamide
    • Gu P, Constantino L, Zhang Y. Enhancement of the antituberculosis activity of weak acids by inhibitors of energy metabolism but not by anaerobiosis suggests that weak acids act differently from the front-line tuberculosis drug pyrazinamide. J Med Microbiol 2008; 57: 1129-34.
    • (2008) J Med Microbiol , vol.57 , pp. 1129-1134
    • Gu, P.1    Constantino, L.2    Zhang, Y.3
  • 2
    • 4344678279 scopus 로고    scopus 로고
    • Anaerobic incubation conditions enhance pyrazinamide activity against Mycobacterium tuberculosis
    • Wade MM, Zhang Y. Anaerobic incubation conditions enhance pyrazinamide activity against Mycobacterium tuberculosis. J Med Microbiol 2004; 53: 769-73.
    • (2004) J Med Microbiol , vol.53 , pp. 769-773
    • Wade, M.M.1    Zhang, Y.2
  • 3
    • 0023707358 scopus 로고
    • The role of pyrazinamide in tuberculosis chemotherapy
    • Steele MA, Des Prez RM. The role of pyrazinamide in tuberculosis chemotherapy. Chest 1988; 94: 845-50.
    • (1988) Chest , vol.94 , pp. 845-850
    • Steele, M.A.1    des Prez, R.M.2
  • 4
    • 0011358622 scopus 로고
    • Nicotinamidase in mycobacteria: A method for distinguishing bovine type tubercle bacilli from other mycobacteria
    • Konno K, Nagayama H, Oka S. Nicotinamidase in mycobacteria: a method for distinguishing bovine type tubercle bacilli from other mycobacteria. Nature 1959; 184: 1743-4.
    • (1959) Nature , vol.184 , pp. 1743-1744
    • Konno, K.1    Nagayama, H.2    Oka, S.3
  • 5
    • 0037252098 scopus 로고    scopus 로고
    • The curious characteristics of pyrazinamide: A review
    • Zhang Y, Mitchison D. The curious characteristics of pyrazinamide: a review. Int J Tuberc Lung Dis 2003; 7: 6-21.
    • (2003) Int J Tuberc Lung Dis , vol.7 , pp. 6-21
    • Zhang, Y.1    Mitchison, D.2
  • 6
    • 0242437861 scopus 로고    scopus 로고
    • Mode of action of pyrazinamide: Disruption of Mycobacterium tuberculosis membrane transport and energetics by pyrazinoic acid
    • Zhang Y, Wade MM, Scorpio A, Zhang H, Sun Z. Mode of action of pyrazinamide: disruption of Mycobacterium tuberculosis membrane transport and energetics by pyrazinoic acid. J Antimicrob Chemother 2003; 52: 790-5.
    • (2003) J Antimicrob Chemother , vol.52 , pp. 790-795
    • Zhang, Y.1    Wade, M.M.2    Scorpio, A.3    Zhang, H.4    Sun, Z.5
  • 7
    • 0033834868 scopus 로고    scopus 로고
    • Pyrazinamide inhibits the eukaryotic-like fatty acid synthetase I (FASI) of Mycobacterium tuberculosis
    • Zimhony O, Cox JS, Welch JT, Vilchèze C, Jacobs WR, Jr. Pyrazinamide inhibits the eukaryotic-like fatty acid synthetase I (FASI) of Mycobacterium tuberculosis. Nat Med 2000; 6: 1043-7.
    • (2000) Nat Med , vol.6 , pp. 1043-1047
    • Zimhony, O.1    Cox, J.S.2    Welch, J.T.3    Vilchèze, C.4    Jacobs Jr., W.R.5
  • 8
    • 0014062867 scopus 로고
    • Pyrazinamide susceptibility and amidase activity of tubercle bacilli
    • Konno K, Feldmann FM, McDermott W. Pyrazinamide susceptibility and amidase activity of tubercle bacilli. Am Rev Respir Dis 1967; 95: 461-9.
    • (1967) Am Rev Respir Dis , vol.95 , pp. 461-469
    • Konno, K.1    Feldmann, F.M.2    McDermott, W.3
  • 10
    • 0029954860 scopus 로고    scopus 로고
    • Mutations in pncA a gene encoding pyrazinamidase/nicotin-amidase cause resistance to the antituberculosis drug pyrazinamide in M. tuberculosis
    • Scorpio A, Zhang Y. Mutations in pncA a gene encoding pyrazinamidase/nicotin-amidase cause resistance to the antituberculosis drug pyrazinamide in M. tuberculosis. Nature Med 1996; 2: 662-7.
    • (1996) Nature Med , vol.2 , pp. 662-667
    • Scorpio, A.1    Zhang, Y.2
  • 11
    • 0008160534 scopus 로고
    • Antimycobacterial drugs
    • Peterson PK, Verhoef J, editors, New York: Elsevier
    • Gangadharam PRJ, Iseman MD. Antimycobacterial drugs. In: Peterson PK, Verhoef J, editors. The antimicrobial agents annual. New York: Elsevier; 1986. p. 17-40.
    • (1986) The Antimicrobial Agents Annual , pp. 17-40
    • Gangadharam, P.R.J.1    Iseman, M.D.2
  • 12
    • 0028804965 scopus 로고
    • Pyrazinoic acid esters with broad spectrum in vitro antimycobacterial activity
    • Cynamon MH, Gimi R, Gyenes F, Sharpe CA, Bergmann KR, Han HJ, et al. Pyrazinoic acid esters with broad spectrum in vitro antimycobacterial activity. J Med Chem 1995; 38: 3902-7.
    • (1995) J Med Chem , vol.38 , pp. 3902-3907
    • Cynamon, M.H.1    Gimi, R.2    Gyenes, F.3    Sharpe, C.A.4    Bergmann, K.R.5    Han, H.J.6
  • 13
    • 0026696665 scopus 로고
    • Antimycobacterial activity of a series of pyrazinoic acid esters
    • Cynamon MH, Klemens SP, Chou TS. Antimycobacterial activity of a series of pyrazinoic acid esters. J Med Chem 1992; 35: 1212-5.
    • (1992) J Med Chem , vol.35 , pp. 1212-1215
    • Cynamon, M.H.1    Klemens, S.P.2    Chou, T.S.3
  • 16
    • 65649089528 scopus 로고    scopus 로고
    • Promising antituberculosis activity of the oxazolidinone PNU-100480 relative to that of linezolid in a murine model
    • Williams KN, Stover CK, Zhu T, Zhu T, Ogden A, Tasneen R, et al. Promising antituberculosis activity of the oxazolidinone PNU-100480 relative to that of linezolid in a murine model. Antimicrob Agents Chemother 2009; 53: 1314-9.
    • (2009) Antimicrob Agents Chemother , vol.53 , pp. 1314-1319
    • Williams, K.N.1    Stover, C.K.2    Zhu, T.3    Zhu, T.4    Ogden, A.5    Tasneen, R.6
  • 18
    • 70349318577 scopus 로고    scopus 로고
    • Paradoxical effect of isoniazid on the activity of rifampin-pyrazinamide combination in a mouse model of tuberculosis
    • Almeida D, Nuermberger EL, Tasneen R, Rosenthal I, Tyagi S, Williams K, et al. Paradoxical effect of isoniazid on the activity of rifampin-pyrazinamide combination in a mouse model of tuberculosis. Antimicrob Agents Chemother 2009; 53: 4178-84.
    • (2009) Antimicrob Agents Chemother , vol.53 , pp. 4178-4184
    • Almeida, D.1    Nuermberger, E.L.2    Tasneen, R.3    Rosenthal, I.4    Tyagi, S.5    Williams, K.6
  • 19
    • 0018046759 scopus 로고
    • The sterilizing value of rifampicin and pyrazinamide in experimental short-course chemotherapy
    • Grosset J. The sterilizing value of rifampicin and pyrazinamide in experimental short-course chemotherapy. Bull Int Union Tuberc 1978; 53: 5-12.
    • (1978) Bull Int Union Tuberc , vol.53 , pp. 5-12
    • Grosset, J.1
  • 20
    • 0026583530 scopus 로고
    • Antagonism between isoniazid and the combination pyrazinamide-rifampin against tuberculosis infection in mice
    • Grosset J, Truffot-Pernot C, Lacroix C, Ji B. Antagonism between isoniazid and the combination pyrazinamide-rifampin against tuberculosis infection in mice. Antimicrob Agents Chemother 1992; 36: 548-51.
    • (1992) Antimicrob Agents Chemother , vol.36 , pp. 548-551
    • Grosset, J.1    Truffot-Pernot, C.2    Lacroix, C.3    Ji, B.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.