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Volumn 57, Issue 9, 2008, Pages 1129-1134

Enhancement of the antituberculosis activity of weak acids by inhibitors of energy metabolism but not by anaerobiosis suggests that weak acids act differently from the front-line tuberculosis drug pyrazinamide

Author keywords

[No Author keywords available]

Indexed keywords

4 DODECYLOXYLBENZOIC ACID; BENZAMIDE DERIVATIVE; BENZOIC ACID ESTER DERIVATIVE; DICYCLOHEXYLCARBODIIMIDE; PROPYLHYDROXYBENZOIC ACID; PYRAZINAMIDE; PYRAZINOIC ACID; SODIUM AZIDE; UNCLASSIFIED DRUG;

EID: 51149085652     PISSN: 00222615     EISSN: None     Source Type: Journal    
DOI: 10.1099/jmm.0.2008/000786-0     Document Type: Article
Times cited : (17)

References (16)
  • 2
    • 0026662342 scopus 로고
    • The microsomal demethylation of N,N-dimethylbenzamides. Substituent and kinetic deuterium isotope effects
    • Constantino, L., Rosa, E. & Iley, J. (1992). The microsomal demethylation of N,N-dimethylbenzamides. Substituent and kinetic deuterium isotope effects. Biochem Pharmacol 44, 651-658.
    • (1992) Biochem Pharmacol , vol.44 , pp. 651-658
    • Constantino, L.1    Rosa, E.2    Iley, J.3
  • 3
    • 0038182191 scopus 로고    scopus 로고
    • The TB epidemic from 1992 to 2002
    • Raviglione, M. C. (2003). The TB epidemic from 1992 to 2002. Tuberculosis (Edinb) 83, 4-14.
    • (2003) Tuberculosis (Edinb) , vol.83 , pp. 4-14
    • Raviglione, M.C.1
  • 4
    • 0014608748 scopus 로고
    • Linear free-energy relationship between alcohol pKa and solvolysis rates of esters where substituent variation is in the alkyl portion of the ester
    • Robinson, J. R. & Matheson, L. E. (1969). Linear free-energy relationship between alcohol pKa and solvolysis rates of esters where substituent variation is in the alkyl portion of the ester. J Org Chem 34, 3630-3633.
    • (1969) J Org Chem , vol.34 , pp. 3630-3633
    • Robinson, J.R.1    Matheson, L.E.2
  • 5
    • 0037018901 scopus 로고    scopus 로고
    • Escherichia coli genes involved in resistance to pyrazinoic acid, the active component of the tuberculosis drug pyrazinamide
    • Schaller, A., Guo, M., Gisanrin, O. & Zhang, Y. (2002). Escherichia coli genes involved in resistance to pyrazinoic acid, the active component of the tuberculosis drug pyrazinamide. FEMS Microbiol Lett 211, 265-270.
    • (2002) FEMS Microbiol Lett , vol.211 , pp. 265-270
    • Schaller, A.1    Guo, M.2    Gisanrin, O.3    Zhang, Y.4
  • 6
    • 0033052157 scopus 로고    scopus 로고
    • Reduced pyrazinamidase activity and the natural resistance of Mycobacterium kansasii to the antituberculosis drug pyrazinamide
    • Sun, Z. & Zhang, Y. (1999a). Reduced pyrazinamidase activity and the natural resistance of Mycobacterium kansasii to the antituberculosis drug pyrazinamide. Antimicrob Agents Chemother 43, 537-542.
    • (1999) Antimicrob Agents Chemother , vol.43 , pp. 537-542
    • Sun, Z.1    Zhang, Y.2
  • 7
    • 0032833154 scopus 로고    scopus 로고
    • Antituberculosis activity of certain antifungal and antihelmintic drugs
    • Sun, Z. & Zhang, Y. (1999b). Antituberculosis activity of certain antifungal and antihelmintic drugs. Tuber Lung Dis 79, 319-320.
    • (1999) Tuber Lung Dis , vol.79 , pp. 319-320
    • Sun, Z.1    Zhang, Y.2
  • 8
    • 7444253306 scopus 로고    scopus 로고
    • Prodrug research: Futile or fertile?
    • Testa, B. (2004). Prodrug research: futile or fertile? Biochem Pharmacol 68, 2097-2106.
    • (2004) Biochem Pharmacol , vol.68 , pp. 2097-2106
    • Testa, B.1
  • 9
    • 4344678279 scopus 로고    scopus 로고
    • Anaerobic incubation conditions enhance pyrazinamide activity against Mycobacterium tuberculosis
    • Wade, M. M. & Zhang, Y. (2004). Anaerobic incubation conditions enhance pyrazinamide activity against Mycobacterium tuberculosis. J Med Microbiol 53, 769-773.
    • (2004) J Med Microbiol , vol.53 , pp. 769-773
    • Wade, M.M.1    Zhang, Y.2
  • 10
    • 34250213044 scopus 로고    scopus 로고
    • Effects of weak acids, UV and proton motive force inhibitors on pyrazinamide activity against Mycobacterium tuberculosis in vitro
    • Wade, M. M. & Zhang, Y. (2006). Effects of weak acids, UV and proton motive force inhibitors on pyrazinamide activity against Mycobacterium tuberculosis in vitro. J Antimicrob Chemother 58, 936-941.
    • (2006) J Antimicrob Chemother , vol.58 , pp. 936-941
    • Wade, M.M.1    Zhang, Y.2
  • 11
    • 2942530484 scopus 로고    scopus 로고
    • Accurate mapping of mutations of pyrazinamide-resistant Mycobacterium tuberculosis strains with a scanning-frame oligonucleotide microarray
    • Wade, M. M., Volokhov, D., Peredelchuk, M., Chizhikov, V. & Zhang, Y. (2004). Accurate mapping of mutations of pyrazinamide-resistant Mycobacterium tuberculosis strains with a scanning-frame oligonucleotide microarray. Diagn Microbiol Infect Dis 49, 89-97.
    • (2004) Diagn Microbiol Infect Dis , vol.49 , pp. 89-97
    • Wade, M.M.1    Volokhov, D.2    Peredelchuk, M.3    Chizhikov, V.4    Zhang, Y.5
  • 12
    • 13844319812 scopus 로고    scopus 로고
    • The magic bullets and tuberculosis drug targets
    • Zhang, Y. (2005). The magic bullets and tuberculosis drug targets. Annu Rev Pharmacol Toxicol 45, 529-564.
    • (2005) Annu Rev Pharmacol Toxicol , vol.45 , pp. 529-564
    • Zhang, Y.1
  • 13
    • 0037252098 scopus 로고    scopus 로고
    • The curious characteristics of pyrazinamide: A review
    • Zhang, Y. & Mitchison, D. (2003). The curious characteristics of pyrazinamide: a review. Int J Tuberc Lung Dis 7, 6-21.
    • (2003) Int J Tuberc Lung Dis , vol.7 , pp. 6-21
    • Zhang, Y.1    Mitchison, D.2
  • 14
    • 0032936728 scopus 로고    scopus 로고
    • Role of acid pH and deficient efflux of pyrazinoic acid in unique susceptibility of Mycobacterium tuberculosis to pyrazinamide
    • Zhang, Y., Scorpio, A., Nikaido, H. & Sun, Z. (1999). Role of acid pH and deficient efflux of pyrazinoic acid in unique susceptibility of Mycobacterium tuberculosis to pyrazinamide. J Bacteriol 181, 2044-2049.
    • (1999) J Bacteriol , vol.181 , pp. 2044-2049
    • Zhang, Y.1    Scorpio, A.2    Nikaido, H.3    Sun, Z.4
  • 15
    • 0242437861 scopus 로고    scopus 로고
    • Mode of action of pyrazinamide: Disruption of Mycobacterium tuberculosis membrane transport and energetics by pyrazinoic acid
    • Zhang, Y., Wade, M. M., Scorpio, A., Zhang, H. & Sun, Z. (2003a). Mode of action of pyrazinamide: disruption of Mycobacterium tuberculosis membrane transport and energetics by pyrazinoic acid. J Antimicrob Chemother 52, 790-795.
    • (2003) J Antimicrob Chemother , vol.52 , pp. 790-795
    • Zhang, Y.1    Wade, M.M.2    Scorpio, A.3    Zhang, H.4    Sun, Z.5
  • 16
    • 0037587282 scopus 로고    scopus 로고
    • Susceptibility of Mycobacterium tuberculosis to weak acids
    • Zhang, Y., Zhang, H. & Sun, Z. (2003b). Susceptibility of Mycobacterium tuberculosis to weak acids. J Antimicrob Chemother 52, 56-60.
    • (2003) J Antimicrob Chemother , vol.52 , pp. 56-60
    • Zhang, Y.1    Zhang, H.2    Sun, Z.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.