-
2
-
-
0036144207
-
Efficacy and safety of amisulpride 50 mg versus paroxetine 20 mg in major depression: A randomized, double-blind, parallel group study
-
Cassano, G. B. and Jori, M. C. (2002) Efficacy and safety of amisulpride 50 mg versus paroxetine 20 mg in major depression: a randomized, double-blind, parallel group study Int. Clin. Psychopharmacol. 17, 27-32 (Pubitemid 34056522)
-
(2002)
International Clinical Psychopharmacology
, vol.17
, Issue.1
, pp. 27-32
-
-
Cassano, G.B.1
Jori, M.C.2
-
3
-
-
0031110985
-
Amilsulpride versus imipramine and placebo in dysthymia and major depression
-
DOI 10.1016/S0165-0327(96)00103-6, PII S0165032796013876
-
Lecrubier, Y., Boyer, P., Turjanski, S., and Rein, W. (1997) Amisulpride versus imipramine and placebo in dysthymia and major depression. Amisulpride Study Group J. Affective Disord. 43, 95-103 (Pubitemid 27221927)
-
(1997)
Journal of Affective Disorders
, vol.43
, Issue.2
, pp. 95-103
-
-
Lecrubier, Y.1
Boyer, P.2
Turjanski, S.3
Rein, W.4
-
4
-
-
67649452096
-
7 antagonist: Relevance for antidepressant actions in vivo
-
7 antagonist: relevance for antidepressant actions in vivo Psychopharmacology (Berlin, Ger.) 205, 119-128
-
(2009)
Psychopharmacology (Berlin, Ger.)
, vol.205
, pp. 119-128
-
-
Abbas, A.I.1
Hedlund, P.B.2
Huang, X.P.3
Tran, T.B.4
Meltzer, H.Y.5
Roth, B.L.6
-
5
-
-
77953753014
-
1A receptor activity
-
1A receptor activity J. Pharmacol. Exp. Ther. 334, 171-181
-
(2010)
J. Pharmacol. Exp. Ther.
, vol.334
, pp. 171-181
-
-
Ishibashi, T.1
Horisawa, T.2
Tokuda, K.3
Ishiyama, T.4
Ogasa, M.5
Tagashira, R.6
Matsumoto, K.7
Nishikawa, H.8
Ueda, Y.9
Toma, S.10
Oki, H.11
Tanno, N.12
Saji, I.13
Ito, A.14
Ohno, Y.15
Nakamura, M.16
-
6
-
-
33748935747
-
7 serotonin receptor
-
DOI 10.1124/mol.106.024612
-
7 serotonin receptor Mol. Pharmacol. 70, 1264-1270 (Pubitemid 44435978)
-
(2006)
Molecular Pharmacology
, vol.70
, Issue.4
, pp. 1264-1270
-
-
Smith, C.1
Rahman, T.2
Toohey, N.3
Mazurkiewicz, J.4
Herrick-Davis, K.5
Teitler, M.6
-
8
-
-
77954218914
-
7 radiotracer for positron emission tomography
-
7 radiotracer for positron emission tomography Bioorg. Med. Chem. Lett. 20, 3730-3733
-
(2010)
Bioorg. Med. Chem. Lett.
, vol.20
, pp. 3730-3733
-
-
Andries, J.1
Lemoine, L.2
Mouchel-Blaisot, A.3
Tang, S.4
Verdurand, M.5
Le, B.D.6
Zimmer, L.7
Billard, T.8
-
11
-
-
84863220845
-
7 receptor imaging
-
7 receptor imaging Bioorg. Med. Chem. 20, 4574-4581
-
(2012)
Bioorg. Med. Chem.
, vol.20
, pp. 4574-4581
-
-
Herth, M.M.1
Hansen, H.D.2
Ettrup, A.3
Dyssegaard, A.4
Lehel, S.5
Kristensen, J.6
Knudsen, G.M.7
-
12
-
-
79151477312
-
7 receptor agents: Structure-activity relationships and potential therapeutic applications in central nervous system disorders
-
7 receptor agents: Structure-activity relationships and potential therapeutic applications in central nervous system disorders Pharmacol. Ther. 129, 120-148
-
(2011)
Pharmacol. Ther.
, vol.129
, pp. 120-148
-
-
Leopoldo, M.1
Lacivita, E.2
Berardi, F.3
Perrone, R.4
Hedlund, P.B.5
-
13
-
-
43049113873
-
7 receptor antagonists
-
DOI 10.1021/jm070279v
-
7 receptor antagonists J. Med. Chem. 51, 2522-2532 (Pubitemid 351628514)
-
(2008)
Journal of Medicinal Chemistry
, vol.51
, Issue.8
, pp. 2522-2532
-
-
Volk, B.1
Barkoczy, J.2
Hegedus, E.3
Udvari, S.4
Gacsalyi, I.5
Mezei, T.6
Pallagi, K.7
Kompagne, H.8
Levay, G.9
Egyed, A.10
Harsing Jr., L.G.11
Spedding, M.12
Simig, G.13
-
14
-
-
80053927380
-
7 receptor antagonist activity
-
7 receptor antagonist activity J. Med. Chem. 54, 6657-6669
-
(2011)
J. Med. Chem.
, vol.54
, pp. 6657-6669
-
-
Volk, B.1
Gacsalyi, I.2
Pallagi, K.3
Poszavacz, L.4
Gyonos, I.5
Szabo, E.6
Bako, T.7
Spedding, M.8
Simig, G.9
Szenasi, G.10
-
15
-
-
17044459906
-
3H]WAY-100635
-
DOI 10.1016/S0006-8993(96)01131-6, PII S0006899396011316
-
11C]WAY 100635 Brain Res. 745, 96-108 (Pubitemid 27055749)
-
(1997)
Brain Research
, vol.745
, Issue.1-2
, pp. 96-108
-
-
Hall, H.1
Lundkvist, C.2
Halldin, C.3
Farde, L.4
Pike, V.W.5
McCarron, J.A.6
Fletcher, A.7
Cliffe, I.A.8
Barf, T.9
Wikstrom, H.10
Sedvall, G.11
-
16
-
-
4444323618
-
3H]SB-269970
-
DOI 10.1016/j.neulet.2004.06.025, PII S0304394004007608
-
3H]SB-269970 Neurosci. Lett. 367, 313-316 (Pubitemid 39178603)
-
(2004)
Neuroscience Letters
, vol.367
, Issue.3
, pp. 313-316
-
-
Varnas, K.1
Thomas, D.R.2
Tupala, E.3
Tiihonen, J.4
Hall, H.5
-
17
-
-
0242354956
-
New one-pot synthesis of 3-alkyl- and 3-(ω-hydroxyalkyl)oxindoles from isatins
-
Volk, B. and Simig, G. (2003) New one-pot synthesis of 3-alkyl- and 3-(ω-hydroxyalkyl)oxindoles from isatins Eur. J. Org. Chem. 3991-3996
-
(2003)
Eur. J. Org. Chem.
, pp. 3991-3996
-
-
Volk, B.1
Simig, G.2
-
18
-
-
0002953363
-
Formation of N-substituted and C-substituted derivatives during alkylation of indol-2(3 H)-one
-
Gruda, I. (1972) Formation of N-substituted and C-substituted derivatives during alkylation of indol-2(3 H)-one Can. J. Chem. 50, 18-23
-
(1972)
Can. J. Chem.
, vol.50
, pp. 18-23
-
-
Gruda, I.1
-
19
-
-
0021191466
-
SYNTHESEWEGE ZU 3-SUBSTITUIERTEN INDOL-2-ONEN
-
Reisch, J., Muller, M., and Labitzke, H. (1984) Synthetic pathways for 3-substituted indol-2-ones Arch. Pharm. 317, 639-646 (Pubitemid 14077640)
-
(1984)
Archiv der Pharmazie
, vol.317
, Issue.7
, pp. 639-646
-
-
Reisch, J.1
Muller, M.2
Labitzke, H.3
-
20
-
-
0002651083
-
Regioselective C-3 alkylations of oxindole dianion
-
Kende, A. S. and Hodges, J. C. (1982) Regioselective C-3 alkylations of oxindole dianion Synth. Commun. 12, 1-10
-
(1982)
Synth. Commun.
, vol.12
, pp. 1-10
-
-
Kende, A.S.1
Hodges, J.C.2
-
21
-
-
65249134003
-
Iridium catalysed C-3 alkylation of oxindole with alcohols under solvent free thermal or microwave conditions
-
Grigg, R., Whitney, S., Sridharan, V., Keep, A., and Derrick, A. (2009) Iridium catalysed C-3 alkylation of oxindole with alcohols under solvent free thermal or microwave conditions Tetrahedron 65, 4375-4383
-
(2009)
Tetrahedron
, vol.65
, pp. 4375-4383
-
-
Grigg, R.1
Whitney, S.2
Sridharan, V.3
Keep, A.4
Derrick, A.5
-
22
-
-
0036230837
-
Raney nickel-induced 3-alkylation of oxindole with alcohols and diols
-
Volk, B., Mezei, T., and Simig, G. (2002) Raney nickel-induced 3-alkylation of oxindole with alcohols and diols Synthesis-Stuttgart 595-597 (Pubitemid 34303972)
-
(2002)
Synthesis
, Issue.5
, pp. 595-597
-
-
Volk, B.1
Mezei, T.2
Simig, G.3
-
24
-
-
33749250382
-
Novel potent neuropeptide Y Y5 receptor antagonists: Synthesis and structure-activity relationships of phenylpiperazine derivatives
-
DOI 10.1016/j.bmc.2006.07.023, PII S0968089606005761
-
Takahashi, T., Sakuraba, A., Hirohashi, T., Shibata, T., Hirose, M., Haga, Y., Nonoshita, K., Kanno, T., Ito, J., Iwaasa, H., Kanatani, A., Fukami, T., and Sato, N. (2006) Novel potent neuropeptide YY5 receptor antagonists: Synthesis and structure-activity relationships of phenylpiperazine derivatives Bioorg. Med. Chem. 14, 7501-7511 (Pubitemid 44486804)
-
(2006)
Bioorganic and Medicinal Chemistry
, vol.14
, Issue.22
, pp. 7501-7511
-
-
Takahashi, T.1
Sakuraba, A.2
Hirohashi, T.3
Shibata, T.4
Hirose, M.5
Haga, Y.6
Nonoshita, K.7
Kanno, T.8
Ito, J.9
Iwaasa, H.10
Kanatani, A.11
Fukami, T.12
Sato, N.13
-
25
-
-
0001412263
-
Determination of lipophilicity by gradient elution high-performance liquid chromatography
-
Krass, J. D., Jastorff, B., and Genieser, H. G. (1997) Determination of lipophilicity by gradient elution high-performance liquid chromatography Anal. Chem. 69, 2575-2581 (Pubitemid 127482932)
-
(1997)
Analytical Chemistry
, vol.69
, Issue.13
, pp. 2575-2581
-
-
Krass, J.D.1
Jastorff, B.2
Genieser, H.-G.3
-
26
-
-
15644370083
-
Effect of plasma protein binding-on in vivo activity and brain penetration of glycine/NMDA receptor antagonists
-
DOI 10.1021/jm970417o
-
Rowley, M., Kulagowski, J. J., Watt, A. P., Rathbone, D., Stevenson, G. I., Carling, R. W., Baker, R., Marshall, G. R., Kemp, J. A., Foster, A. C., Grimwood, S., Hargreaves, R., Hurley, C., Saywell, K. L., Tricklebank, M. D., and Leeson, P. D. (1997) Effect of plasma protein binding on in vivo activity and brain penetration of glycine/NMDA receptor antagonists J. Med. Chem. 40, 4053-4068 (Pubitemid 28008400)
-
(1997)
Journal of Medicinal Chemistry
, vol.40
, Issue.25
, pp. 4053-4068
-
-
Rowley, M.1
Kulagowski, J.J.2
Watt, A.P.3
Rathbone, D.4
Stevenson, G.I.5
Carling, R.W.6
Baker, R.7
Marshall, G.R.8
Kemp, J.A.9
Foster, A.C.10
Grimwood, S.11
Hargreaves, R.12
Hurley, C.13
Saywell, K.L.14
Tricklebank, M.D.15
Leeson, P.D.16
-
27
-
-
79956273216
-
11C] methylation
-
11C]methylation Org Biomol. Chem. 9, 4287-4294
-
(2011)
Org Biomol. Chem.
, vol.9
, pp. 4287-4294
-
-
Koyama, H.1
Siqin2
Zhang, Z.3
Sumi, K.4
Hatta, Y.5
Nagata, H.6
Doi, H.7
Suzuki, M.8
-
28
-
-
0037204696
-
11C-carbamoyl compounds
-
DOI 10.1021/jo016307d
-
Kihlberg, T., Karimi, F., and Langstrom, B. (2002) [C-11]Carbon monoxide in selenium-mediated synthesis of C-11-carbamoyl compounds J. Org. Chem. 67, 3687-3692 (Pubitemid 34563979)
-
(2002)
Journal of Organic Chemistry
, vol.67
, Issue.11
, pp. 3687-3692
-
-
Kihlberg, T.1
Karimi, F.2
Langstrom, B.3
-
29
-
-
35348886690
-
18F-labelled aromatic amino acids
-
DOI 10.1016/j.apradiso.2007.06.002, PII S0969804307001790
-
18F- benzaldehydes for modelling syntheses of F-18-labelled aromatic amino acids Appl. Radiat. Isot. 65, 1227-1231 (Pubitemid 47575941)
-
(2007)
Applied Radiation and Isotopes
, vol.65
, Issue.11
, pp. 1227-1231
-
-
Shen, B.1
Loffler, D.2
Zeller, K.-P.3
Ubele, M.4
Reischl, G.5
Machulla, H.-J.6
-
30
-
-
44849112165
-
Molecular imaging with PET
-
DOI 10.1021/cr0782426
-
Ametamey, S. M., Honer, M., and Schubiger, P. A. (2008) Molecular imaging with PET Chem. Rev. 108, 1501-1516 (Pubitemid 351796395)
-
(2008)
Chemical Reviews
, vol.108
, Issue.5
, pp. 1501-1516
-
-
Ametamey, S.M.1
Honer, M.2
Schubiger, P.A.3
-
31
-
-
39449099398
-
11C labelled radiotracers synthesis
-
DOI 10.2174/092986708783497292
-
Allard, M., Fouquet, E., James, D., and Szlosek-Pinaud, M. (2008) State of art in C-11 labelled radiotracers synthesis Curr. Med. Chem. 15, 235-277 (Pubitemid 351265134)
-
(2008)
Current Medicinal Chemistry
, vol.15
, Issue.3
, pp. 235-277
-
-
Allard, M.1
Fouquet, E.2
James, D.3
Szlosek-Pinaud, M.4
-
32
-
-
0000547341
-
Nucleophilic aromatic-substitution of activated cationic groups by F-18-labeled fluoride - A useful route to no-carrier-added (NCA) F-18-labeled aryl fluorides
-
Angelini, G., Speranza, M., Wolf, A. P., and Shiue, C. Y. (1985) Nucleophilic aromatic-substitution of activated cationic groups by F-18-labeled fluoride-a useful route to no-carrier-added (NCA) F-18-labeled aryl fluorides J. Fluorine Chem. 27, 177-191
-
(1985)
J. Fluorine Chem.
, vol.27
, pp. 177-191
-
-
Angelini, G.1
Speranza, M.2
Wolf, A.P.3
Shiue, C.Y.4
-
34
-
-
0023743170
-
Sigma-receptors in post-mortem human brains
-
Weissman, A. D., Su, T. P., Hedreen, J. C., and London, E. D. (1988) Sigma-receptors in post-mortem human brains J. Pharmacol. Exp. Ther. 247, 29-33
-
(1988)
J. Pharmacol. Exp. Ther.
, vol.247
, pp. 29-33
-
-
Weissman, A.D.1
Su, T.P.2
Hedreen, J.C.3
London, E.D.4
-
35
-
-
3042776615
-
Autoradiographic distribution of serotonin transporters and receptor subtypes in human brain
-
DOI 10.1002/hbm.20035
-
Varnas, K., Halldin, C., and Hall, H. (2004) Autoradiographic distribution of serotonin transporters and receptor subtypes in human brain Human Brain Mapping 22, 246-260 (Pubitemid 38891003)
-
(2004)
Human Brain Mapping
, vol.22
, Issue.3
, pp. 246-260
-
-
Varnas, K.1
Halldin, C.2
Hall, H.3
-
36
-
-
4444323618
-
3H]SB-269970
-
DOI 10.1016/j.neulet.2004.06.025, PII S0304394004007608
-
3H]SB-269970 Neurosci. Lett. 367, 313-316 (Pubitemid 39178603)
-
(2004)
Neuroscience Letters
, vol.367
, Issue.3
, pp. 313-316
-
-
Varnas, K.1
Thomas, D.R.2
Tupala, E.3
Tiihonen, J.4
Hall, H.5
-
37
-
-
17044459906
-
3H]WAY-100635
-
DOI 10.1016/S0006-8993(96)01131-6, PII S0006899396011316
-
11C]WAY-100635 Brain Res. 745, 96-108 (Pubitemid 27055749)
-
(1997)
Brain Research
, vol.745
, Issue.1-2
, pp. 96-108
-
-
Hall, H.1
Lundkvist, C.2
Halldin, C.3
Farde, L.4
Pike, V.W.5
McCarron, J.A.6
Fletcher, A.7
Cliffe, I.A.8
Barf, T.9
Wikstrom, H.10
Sedvall, G.11
-
38
-
-
0024999832
-
1-noradrenergic receptors in the human brain postmortem. Effect of suicide
-
Grossisseroff, R., Dillon, K. A., Fieldust, S. J., and Biegon, A. (1990) Autoradiographic analysis of alpha-1-noradrenergic receptors in the human brain postmortem-Effect of suicide Arch. Gen. Psychiatry 47, 1049-1053 (Pubitemid 20377515)
-
(1990)
Archives of General Psychiatry
, vol.47
, Issue.11
, pp. 1049-1053
-
-
Gross-Isseroff, R.1
Dillon, K.A.2
Fieldust, S.J.3
Biegon, A.4
-
39
-
-
0036006699
-
7 receptors in rodent, pig and primate brain tissues
-
DOI 10.1016/S0028-3908(01)00151-4, PII S0028390801001514
-
7 receptors in rodent, pig and primate brain tissues Neuropharmacology 42, 74-81 (Pubitemid 34062823)
-
(2002)
Neuropharmacology
, vol.42
, Issue.1
, pp. 74-81
-
-
Thomas, D.R.1
Atkinson, P.J.2
Hastie, P.G.3
Roberts, J.C.4
Middlemiss, D.N.5
Price, G.W.6
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