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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 1, 2013, Pages 55-61

Studies on synthesis, stability, release and pharmacodynamic profile of a novel diacerein-thymol prodrug

(4) Dhaneshwar, Suneela a Patel, Vriha a Patil, Dipmala a Meena, Gourav a

a BHARATI VIDYAPEETH DEEMED UNIVERSITY (India)

Author keywords

Antioxidant; Co drug; Diacerein; IL 1 beta inhibitor; Osteoarthritis; Oxidative stress; Thymol; Ulcerogenicity

Indexed keywords

DIACEREIN; DIACEREIN THYMOL PRODRUG; PRODRUG; THYMOL; UNCLASSIFIED DRUG;

ALKALINITY; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIINFLAMMATORY ACTIVITY; ARTHRITIS; ARTICLE; COLD STRESS; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG DESIGN; DRUG RELEASE; DRUG SCREENING; DRUG STABILITY; DRUG SYNTHESIS; HISTOPATHOLOGY; HOMOGENATE; LIPOPHILICITY; MALE; NONHUMAN; PHARMACODYNAMICS; RAT; SMALL INTESTINE; SMALL INTESTINE HOMOGENATE; SPECTROSCOPY; SYNOVITIS;

ANIMALS; ANKLE JOINT; ANTHRAQUINONES; ANTI-INFLAMMATORY AGENTS; ARTHRITIS; HALF-LIFE; INTESTINE, SMALL; MALE; PRODRUGS; RATS; RATS, WISTAR; THYMOL;

ANIMALIA; RATTUS;

EID: 84871007351 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.11.016 Document Type: Article

Times cited : (32)

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