메뉴 건너뛰기




Volumn 12, Issue 6, 2012, Pages 683-689

Cholesterol metabolism and resistance to tamoxifen

Author keywords

[No Author keywords available]

Indexed keywords

11 [4 (2 DIMETHYLAMINOETHOXY)PHENYL]ESTRADIOL; AFIMOXIFENE; ALPHA TOCOPHEROL; CHOLESTEROL 5,6 EPOXIDE HYDROLASE; CHOLESTEROL ACYLTRANSFERASE; CLOMIFENE; DOXORUBICIN; HYDROLASE; MUCIN 1; N PYRROLIDINO 2 [4 (BENZYL)PHENOXYETHANAMINE]; RALOXIFENE; TAMOXIFEN; TAMOXIFEN DERIVATIVE; TESMILIFENE; UNCLASSIFIED DRUG;

EID: 84870566249     PISSN: 14714892     EISSN: 14714973     Source Type: Journal    
DOI: 10.1016/j.coph.2012.09.007     Document Type: Review
Times cited : (50)

References (44)
  • 2
    • 33845904405 scopus 로고    scopus 로고
    • Chemoprevention of breast cancer with selective oestrogen-receptor modulators
    • V.C. Jordan Chemoprevention of breast cancer with selective oestrogen-receptor modulators Nat Rev Cancer 7 2007 46 53
    • (2007) Nat Rev Cancer , vol.7 , pp. 46-53
    • Jordan, V.C.1
  • 3
    • 82555185372 scopus 로고    scopus 로고
    • Four decades of discovery in breast cancer research and treatment - An interview with V. Craig Jordan
    • M. Poirot Four decades of discovery in breast cancer research and treatment - an interview with V. Craig Jordan Int J Dev Biol 55 2011 703 712
    • (2011) Int J Dev Biol , vol.55 , pp. 703-712
    • Poirot, M.1
  • 4
    • 79960980007 scopus 로고    scopus 로고
    • Strategies for subtypes - Dealing with the diversity of breast cancer: Highlights of the St Gallen International Expert Consensus on the Primary Therapy of Early Breast Cancer 2011
    • A. Goldhirsch, W.C. Wood, A.S. Coates, R.D. Gelber, B. Thurlimann, and H.J. Senn Strategies for subtypes - dealing with the diversity of breast cancer: highlights of the St Gallen International Expert Consensus on the Primary Therapy of Early Breast Cancer 2011 Ann Oncol 22 2011 1736 1747
    • (2011) Ann Oncol , vol.22 , pp. 1736-1747
    • Goldhirsch, A.1    Wood, W.C.2    Coates, A.S.3    Gelber, R.D.4    Thurlimann, B.5    Senn, H.J.6
  • 6
    • 70450247207 scopus 로고    scopus 로고
    • Mucins in cancer: Function, prognosis and therapy
    • D.W. Kufe Mucins in cancer: function, prognosis and therapy Nat Rev Cancer 9 2009 874 885
    • (2009) Nat Rev Cancer , vol.9 , pp. 874-885
    • Kufe, D.W.1
  • 7
    • 84863612718 scopus 로고    scopus 로고
    • MUC1-C oncoprotein as a target in breast cancer: Activation of signaling pathways and therapeutic approaches
    • D.W. Kufe MUC1-C oncoprotein as a target in breast cancer: activation of signaling pathways and therapeutic approaches Oncogene 2012
    • (2012) Oncogene
    • Kufe, D.W.1
  • 8
    • 65249127544 scopus 로고    scopus 로고
    • MUC1-induced alterations in a lipid metabolic gene network predict response of human breast cancers to tamoxifen treatment
    • S.P. Pitroda, N.N. Khodarev, M.A. Beckett, D.W. Kufe, and R.R. Weichselbaum MUC1-induced alterations in a lipid metabolic gene network predict response of human breast cancers to tamoxifen treatment Proc Natl Acad Sci USA 106 2009 5837 5841
    • (2009) Proc Natl Acad Sci USA , vol.106 , pp. 5837-5841
    • Pitroda, S.P.1    Khodarev, N.N.2    Beckett, M.A.3    Kufe, D.W.4    Weichselbaum, R.R.5
  • 9
    • 79954996475 scopus 로고    scopus 로고
    • Mucin 1 C-terminal subunit oncoprotein is a target for small-molecule inhibitors
    • Y. Zhou, H. Rajabi, and D. Kufe Mucin 1 C-terminal subunit oncoprotein is a target for small-molecule inhibitors Mol Pharmacol 79 2011 886 893
    • (2011) Mol Pharmacol , vol.79 , pp. 886-893
    • Zhou, Y.1    Rajabi, H.2    Kufe, D.3
  • 11
    • 6444219756 scopus 로고    scopus 로고
    • Multiple targeting by the antitumor drug tamoxifen: A structure-activity study
    • P. de Medina, G. Favre, and Poirot M Multiple targeting by the antitumor drug tamoxifen: a structure-activity study Curr Med Chem Anticancer Agents 4 2004 491 508
    • (2004) Curr Med Chem Anticancer Agents , vol.4 , pp. 491-508
    • De Medina, P.1    Favre, G.2    Poirot, M.3
  • 13
    • 23744440323 scopus 로고    scopus 로고
    • Cholesteryl esters in malignancy
    • M.R. Tosi, and V. Tugnoli Cholesteryl esters in malignancy Clin Chim Acta 359 2005 27 45
    • (2005) Clin Chim Acta , vol.359 , pp. 27-45
    • Tosi, M.R.1    Tugnoli, V.2
  • 15
    • 77954401004 scopus 로고    scopus 로고
    • Acyl-coenzyme A: Cholesterol acyltransferase inhibitor Avasimibe affect survival and proliferation of glioma tumor cell lines
    • S. Bemlih, M.D. Poirier, and M.D. El Andaloussi Acyl-coenzyme A: cholesterol acyltransferase inhibitor Avasimibe affect survival and proliferation of glioma tumor cell lines Cancer Biol Ther 9 2010 1025 1032
    • (2010) Cancer Biol Ther , vol.9 , pp. 1025-1032
    • Bemlih, S.1    Poirier, M.D.2    El Andaloussi, M.D.3
  • 16
    • 77955555025 scopus 로고    scopus 로고
    • High ACAT1 expression in estrogen receptor negative basal-like breast cancer cells is associated with LDL-induced proliferation
    • C.J. Antalis, T. Arnold, T. Rasool, B. Lee, K.K. Buhman, and R.A. Siddiqui High ACAT1 expression in estrogen receptor negative basal-like breast cancer cells is associated with LDL-induced proliferation Breast Cancer Res Treat 122 2010 661 670
    • (2010) Breast Cancer Res Treat , vol.122 , pp. 661-670
    • Antalis, C.J.1    Arnold, T.2    Rasool, T.3    Lee, B.4    Buhman, K.K.5    Siddiqui, R.A.6
  • 17
    • 70350370454 scopus 로고    scopus 로고
    • Signaling through cholesterol esterification: A new pathway for the cholecystokinin 2 receptor involved in cell growth and invasion
    • M.R. Paillasse, P. de Medina, G. Amouroux, L. Mhamdi, M. Poirot, and S. Silvente-Poirot Signaling through cholesterol esterification: a new pathway for the cholecystokinin 2 receptor involved in cell growth and invasion J Lipid Res 50 2009 2203 2211
    • (2009) J Lipid Res , vol.50 , pp. 2203-2211
    • Paillasse, M.R.1    De Medina, P.2    Amouroux, G.3    Mhamdi, L.4    Poirot, M.5    Silvente-Poirot, S.6
  • 18
    • 82355173416 scopus 로고    scopus 로고
    • Migration of MDA-MB-231 breast cancer cells depends on the availability of exogenous lipids and cholesterol esterification
    • C.J. Antalis, A. Uchida, K.K. Buhman, and R.A. Siddiqui Migration of MDA-MB-231 breast cancer cells depends on the availability of exogenous lipids and cholesterol esterification Clin Exp Metastasis 28 2011 733 741
    • (2011) Clin Exp Metastasis , vol.28 , pp. 733-741
    • Antalis, C.J.1    Uchida, A.2    Buhman, K.K.3    Siddiqui, R.A.4
  • 19
    • 33748992624 scopus 로고    scopus 로고
    • The prototypical inhibitor of cholesterol esterification Sah 58-035 [3-[decyldimethylsilyl]-n-[2-(4-methylphenyl)-1-phenylethyl]propanamide], is an agonist of estrogen receptors
    • P. de Medina, N. Boubekeur, P. Balaguer, G. Favre, S. Silvente-Poirot, and M. Poirot The prototypical inhibitor of cholesterol esterification Sah 58-035 [3-[decyldimethylsilyl]-n-[2-(4-methylphenyl)-1-phenylethyl]propanamide], is an agonist of estrogen receptors J Pharmacol Exp Ther 319 2006 139 149
    • (2006) J Pharmacol Exp Ther , vol.319 , pp. 139-149
    • De Medina, P.1    Boubekeur, N.2    Balaguer, P.3    Favre, G.4    Silvente-Poirot, S.5    Poirot, M.6
  • 20
    • 0028835120 scopus 로고
    • Tamoxifen and toremifene lower serum cholesterol by inhibition of delta 8-cholesterol conversion to lathosterol in women with breast cancer
    • H. Gylling, S. Pyrhonen, E. Mantyla, H. Maenpaa, L. Kangas, and T.A. Miettinen Tamoxifen and toremifene lower serum cholesterol by inhibition of delta 8-cholesterol conversion to lathosterol in women with breast cancer J Clin Oncol 13 1995 2900 2905
    • (1995) J Clin Oncol , vol.13 , pp. 2900-2905
    • Gylling, H.1    Pyrhonen, S.2    Mantyla, E.3    Maenpaa, H.4    Kangas, L.5    Miettinen, T.A.6
  • 23
    • 77955799773 scopus 로고    scopus 로고
    • Identification and pharmacological characterization of cholesterol-5,6-epoxide hydrolase as a target for tamoxifen and AEBS ligands
    • P. de Medina, M.R. Paillasse, G. Segala, M. Poirot, and S. Silvente-Poirot Identification and pharmacological characterization of cholesterol-5,6-epoxide hydrolase as a target for tamoxifen and AEBS ligands Proc Natl Acad Sci USA 107 2010 13520 13525
    • (2010) Proc Natl Acad Sci USA , vol.107 , pp. 13520-13525
    • De Medina, P.1    Paillasse, M.R.2    Segala, G.3    Poirot, M.4    Silvente-Poirot, S.5
  • 24
    • 70349185445 scopus 로고    scopus 로고
    • Ligands of the antiestrogen-binding site induce active cell death and autophagy in human breast cancer cells through the modulation of cholesterol metabolism
    • P. de Medina, B. Payre, N. Boubekeur, J. Bertrand-Michel, F. Terce, S. Silvente-Poirot, and M. Poirot Ligands of the antiestrogen-binding site induce active cell death and autophagy in human breast cancer cells through the modulation of cholesterol metabolism Cell Death Differ 16 2009 1372 1384
    • (2009) Cell Death Differ , vol.16 , pp. 1372-1384
    • De Medina, P.1    Payre, B.2    Boubekeur, N.3    Bertrand-Michel, J.4    Terce, F.5    Silvente-Poirot, S.6    Poirot, M.7
  • 26
    • 65249139482 scopus 로고    scopus 로고
    • Autophagy facilitates the progression of ERalpha-positive breast cancer cells to antiestrogen resistance
    • P.V. Schoenlein, S. Periyasamy-Thandavan, J.S. Samaddar, W.H. Jackson, and J.T. Barrett Autophagy facilitates the progression of ERalpha-positive breast cancer cells to antiestrogen resistance Autophagy 5 2009 400 403
    • (2009) Autophagy , vol.5 , pp. 400-403
    • Schoenlein, P.V.1    Periyasamy-Thandavan, S.2    Samaddar, J.S.3    Jackson, W.H.4    Barrett, J.T.5
  • 27
    • 84870512029 scopus 로고    scopus 로고
    • Abstract 956: The liver-X-receptor-α is involved in the induction by Tamoxifen of breast cancer cell differentiation and death
    • Abstract nr
    • G. Segala, P. de Medina, M.R. Paillasse, V.C. Jordan, S. Silvente-Poirot, and M. Poirot Abstract 956: The liver-X-receptor-α is involved in the induction by Tamoxifen of breast cancer cell differentiation and death Cancer Res 72 2012 956 Abstract nr
    • (2012) Cancer Res , vol.72 , pp. 956
    • Segala, G.1    De Medina, P.2    Paillasse, M.R.3    Jordan, V.C.4    Silvente-Poirot, S.5    Poirot, M.6
  • 28
    • 57749092180 scopus 로고    scopus 로고
    • Microsomal antiestrogen-binding site ligands induce growth control and differentiation of human breast cancer cells through the modulation of cholesterol metabolism
    • B. Payre, P. de Medina, N. Boubekeur, L. Mhamdi, J. Bertrand-Michel, F. Terce, I. Fourquaux, D. Goudouneche, M. Record, and M. Poirot Microsomal antiestrogen-binding site ligands induce growth control and differentiation of human breast cancer cells through the modulation of cholesterol metabolism Mol Cancer Ther 7 2008 3707 3718
    • (2008) Mol Cancer Ther , vol.7 , pp. 3707-3718
    • Payre, B.1    De Medina, P.2    Boubekeur, N.3    Mhamdi, L.4    Bertrand-Michel, J.5    Terce, F.6    Fourquaux, I.7    Goudouneche, D.8    Record, M.9    Poirot, M.10
  • 29
    • 79955979073 scopus 로고    scopus 로고
    • MUC1-C oncoprotein suppresses reactive oxygen species-induced terminal differentiation of acute myelogenous leukemia cells
    • L. Yin, Z. Wu, D. Avigan, J. Rosenblatt, R. Stone, S. Kharbanda, and D. Kufe MUC1-C oncoprotein suppresses reactive oxygen species-induced terminal differentiation of acute myelogenous leukemia cells Blood 117 2011 4863 4870
    • (2011) Blood , vol.117 , pp. 4863-4870
    • Yin, L.1    Wu, Z.2    Avigan, D.3    Rosenblatt, J.4    Stone, R.5    Kharbanda, S.6    Kufe, D.7
  • 31
    • 10344229445 scopus 로고    scopus 로고
    • Regulation of cellular response to oncogenic and oxidative stress by Seladin-1
    • C. Wu, I. Miloslavskaya, S. Demontis, R. Maestro, and K. Galaktionov Regulation of cellular response to oncogenic and oxidative stress by Seladin-1 Nature 432 2004 640 645
    • (2004) Nature , vol.432 , pp. 640-645
    • Wu, C.1    Miloslavskaya, I.2    Demontis, S.3    Maestro, R.4    Galaktionov, K.5
  • 32
    • 84874107079 scopus 로고    scopus 로고
    • Cholesterol-5,6-epoxides: Chemistry, biochemistry, metabolic fate and cancer
    • doi:10.1016/j.biochi.2012.05.006 in press
    • Poirot M, Silvente-Poirot S: Cholesterol-5,6-epoxides: Chemistry, biochemistry, metabolic fate and cancer. Biochimie 2012, in press, http://dx.doi.org/10.1016/j.biochi.2012.05.006.
    • (2012) Biochimie
    • Poirot, M.1    Silvente-Poirot, S.2
  • 33
  • 36
    • 57349194627 scopus 로고    scopus 로고
    • The selective Alzheimer's disease indicator-1 gene (Seladin-1/DHCR24) is a liver X receptor target gene
    • Y. Wang, P.M. Rogers, K.R. Stayrook, C. Su, G. Varga, Q. Shen, S. Nagpal, and T.P. Burris The selective Alzheimer's disease indicator-1 gene (Seladin-1/DHCR24) is a liver X receptor target gene Mol Pharmacol 74 2008 1716 1721
    • (2008) Mol Pharmacol , vol.74 , pp. 1716-1721
    • Wang, Y.1    Rogers, P.M.2    Stayrook, K.R.3    Su, C.4    Varga, G.5    Shen, Q.6    Nagpal, S.7    Burris, T.P.8
  • 37
    • 42049109699 scopus 로고    scopus 로고
    • MCF7 side population cells with characteristics of cancer stem/progenitor cells express the tumor antigen MUC1
    • K. Engelmann, H. Shen, and O.J. Finn MCF7 side population cells with characteristics of cancer stem/progenitor cells express the tumor antigen MUC1 Cancer Res 68 2008 2419 2426
    • (2008) Cancer Res , vol.68 , pp. 2419-2426
    • Engelmann, K.1    Shen, H.2    Finn, O.J.3
  • 38
    • 52049109180 scopus 로고    scopus 로고
    • Mucin1 expression is enriched in the human stem cell fraction of cord blood and is upregulated in majority of the AML cases
    • S. Fatrai, H. Schepers, H. Tadema, E. Vellenga, S.M. Daenen, and J.J. Schuringa Mucin1 expression is enriched in the human stem cell fraction of cord blood and is upregulated in majority of the AML cases Exp Hematol 36 2008 1254 1265
    • (2008) Exp Hematol , vol.36 , pp. 1254-1265
    • Fatrai, S.1    Schepers, H.2    Tadema, H.3    Vellenga, E.4    Daenen, S.M.5    Schuringa, J.J.6
  • 40
    • 83555168180 scopus 로고    scopus 로고
    • Clomiphene as a novel modality for the treatment of acute myeloid leukemia: A pilot phase II study
    • G. Yom-Tov, I. Nathan, O. Shpilberg, A. Polliack, and I. Levi Clomiphene as a novel modality for the treatment of acute myeloid leukemia: a pilot phase II study Leuk Res 36 2012 42 45
    • (2012) Leuk Res , vol.36 , pp. 42-45
    • Yom-Tov, G.1    Nathan, I.2    Shpilberg, O.3    Polliack, A.4    Levi, I.5
  • 41
    • 0033856062 scopus 로고    scopus 로고
    • Synthesis, binding and structure-affinity studies of new ligands for the microsomal anti-estrogen binding site (AEBS)
    • M. Poirot, P. De Medina, F. Delarue, J.J. Perie, A. Klaebe, and J.C. Faye Synthesis, binding and structure-affinity studies of new ligands for the microsomal anti-estrogen binding site (AEBS) Bioorg Med Chem 8 2000 2007 2016
    • (2000) Bioorg Med Chem , vol.8 , pp. 2007-2016
    • Poirot, M.1    De Medina, P.2    Delarue, F.3    Perie, J.J.4    Klaebe, A.5    Faye, J.C.6
  • 42
    • 1342311015 scopus 로고    scopus 로고
    • Phase III study of N N-diethyl-2-[4-(phenylmethyl) phenoxy]ethanamine (BMS-217380-01) combined with doxorubicin versus doxorubicin alone in metastatic/recurrent breast cancer: National Cancer Institute of Canada Clinical Trials Group Study MA 19
    • L. Reyno, L. Seymour, D. Tu, S. Dent, K. Gelmon, B. Walley, A. Pluzanska, V. Gorbunova, A. Garin, and J. Jassem Phase III study of N N-diethyl-2-[4- (phenylmethyl) phenoxy]ethanamine (BMS-217380-01) combined with doxorubicin versus doxorubicin alone in metastatic/recurrent breast cancer: National Cancer Institute of Canada Clinical Trials Group Study MA 19 J Clin Oncol 22 2004 269 276
    • (2004) J Clin Oncol , vol.22 , pp. 269-276
    • Reyno, L.1    Seymour, L.2    Tu, D.3    Dent, S.4    Gelmon, K.5    Walley, B.6    Pluzanska, A.7    Gorbunova, V.8    Garin, A.9    Jassem, J.10
  • 43
    • 58849097669 scopus 로고    scopus 로고
    • Preferential killing of breast tumor initiating cells by N,N-diethyl-2-[4-(phenylmethyl)phenoxy]ethanamine/tesmilifene
    • T. Deng, J.C. Liu, K.I. Pritchard, A. Eisen, and E. Zacksenhaus Preferential killing of breast tumor initiating cells by N,N-diethyl-2-[4- (phenylmethyl)phenoxy]ethanamine/tesmilifene Clin Cancer Res 15 2009 119 130
    • (2009) Clin Cancer Res , vol.15 , pp. 119-130
    • Deng, T.1    Liu, J.C.2    Pritchard, K.I.3    Eisen, A.4    Zacksenhaus, E.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.