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Volumn 34, Issue 6, 2012, Pages 525-535

Predicting skin penetration of actives from complex cosmetic formulations: An evaluation of inter formulation and inter active effects during formulation optimization for transdermal delivery

Author keywords

actives; diffusivity; flux; formulation; partition coefficient; retention; skin penetration

Indexed keywords

ADJUVANT; COSMETIC; DRUG SOLVENT; EMOLLIENT AGENT; FLUOROURACIL; HYDROCORTISONE; KETOCONAZOLE; TESTOSTERONE;

EID: 84868203194     PISSN: 01425463     EISSN: 14682494     Source Type: Journal    
DOI: 10.1111/ics.12001     Document Type: Article
Times cited : (22)

References (30)
  • 1
  • 2
    • 0026606514 scopus 로고
    • Predicting skin permeability
    • Potts, R.O., and, Guy, R.H., Predicting skin permeability. Pharm. Res. 9, 663-669 (1992).
    • (1992) Pharm. Res. , vol.9 , pp. 663-669
    • Potts, R.O.1    Guy, R.H.2
  • 3
    • 0034868376 scopus 로고    scopus 로고
    • Probing the effect of vehicles on topical delivery: Understanding the basic relationship between solvent and active penetration using silicone membranes
    • Cross, S.E., Pugh, W.J., Hadgraft, J., and, Roberts, M.S., Probing the effect of vehicles on topical delivery: understanding the basic relationship between solvent and active penetration using silicone membranes. Pharm. Res. 18, 999-1005 (2001).
    • (2001) Pharm. Res. , vol.18 , pp. 999-1005
    • Cross, S.E.1    Pugh, W.J.2    Hadgraft, J.3    Roberts, M.S.4
  • 5
    • 0141789947 scopus 로고    scopus 로고
    • Effect of vehicle pre-treatment on the flux, retention and diffusion of topically applied penetrants in vitro
    • Rosado, C., Cross, S.E., Pugh, W.J., Roberts, M.S., and, Hadgraft, J., Effect of vehicle pre-treatment on the flux, retention and diffusion of topically applied penetrants in vitro. Pharm. Res. 20, 1502-1507 (2003).
    • (2003) Pharm. Res. , vol.20 , pp. 1502-1507
    • Rosado, C.1    Cross, S.E.2    Pugh, W.J.3    Roberts, M.S.4    Hadgraft, J.5
  • 6
    • 34447253821 scopus 로고    scopus 로고
    • Influence of membrane-solvent-active interactions on active permeation in skin
    • Dias, M., Hadgraft, J., and, Lane, M.E., Influence of membrane-solvent-active interactions on active permeation in skin. Int. J. Pharm. 340, 65-70 (2007).
    • (2007) Int. J. Pharm. , vol.340 , pp. 65-70
    • Dias, M.1    Hadgraft, J.2    Lane, M.E.3
  • 7
    • 79960898776 scopus 로고    scopus 로고
    • Maximum transepidermal flux for similar size phenolic compounds is enhanced by solvent uptake into the skin
    • Zhang, Q., Li, P., and, Roberts, M.S., Maximum transepidermal flux for similar size phenolic compounds is enhanced by solvent uptake into the skin. J. Control Release 154, 50-57 (2011).
    • (2011) J. Control Release , vol.154 , pp. 50-57
    • Zhang, Q.1    Li, P.2    Roberts, M.S.3
  • 8
    • 58149280280 scopus 로고    scopus 로고
    • Formulation effects of topical emulsions on transdermal and dermal delivery
    • Otto, A., du Plessis, J., and, Wiechers, J.W., Formulation effects of topical emulsions on transdermal and dermal delivery. Int. J. Cosmet. Sci. 31, 1-19 (2009).
    • (2009) Int. J. Cosmet. Sci. , vol.31 , pp. 1-19
    • Otto, A.1    Du Plessis, J.2    Wiechers, J.W.3
  • 9
    • 0002246502 scopus 로고
    • Preparation of isolated sheets of human stratum corneum
    • Kligman, A.M., and, Christophers, E., Preparation of isolated sheets of human stratum corneum. Arch. Dermatol. 88, 702-705 (1963).
    • (1963) Arch. Dermatol. , vol.88 , pp. 702-705
    • Kligman, A.M.1    Christophers, E.2
  • 10
    • 0034941295 scopus 로고    scopus 로고
    • Can increasing the viscosity of formulations be used to reduce the human skin penetration of the sunscreen oxybenzone?
    • Cross, S.E., Jiang, R., Benson, H.A.E., and, Roberts, M.S., Can increasing the viscosity of formulations be used to reduce the human skin penetration of the sunscreen oxybenzone? J. Invest. Dermatol. 117, 147-150 (2001).
    • (2001) J. Invest. Dermatol. , vol.117 , pp. 147-150
    • Cross, S.E.1    Jiang, R.2    Benson, H.A.E.3    Roberts, M.S.4
  • 11
    • 0024424743 scopus 로고
    • Bioavailability assessment of topical delivery systems: Effect of vehicle evaporation upon in vitro delivery of minoxidil from solution formulations
    • Chiang, C.M., Flynn, G.L., Weiner, N.D., and, Szpunar, G.J., Bioavailability assessment of topical delivery systems: effect of vehicle evaporation upon in vitro delivery of minoxidil from solution formulations. Int. J. Pharm. 55, 229-236 (1989).
    • (1989) Int. J. Pharm. , vol.55 , pp. 229-236
    • Chiang, C.M.1    Flynn, G.L.2    Weiner, N.D.3    Szpunar, G.J.4
  • 12
    • 2342599148 scopus 로고    scopus 로고
    • Molecular weight as the main determinant of maximum flux across the skin
    • Magnusson, B.M., Anissimov, Y.G., Cross, S.E., and, Roberts, M.S., Molecular weight as the main determinant of maximum flux across the skin. J. Invest. Dermatol. 22, 993-999 (2004).
    • (2004) J. Invest. Dermatol. , vol.22 , pp. 993-999
    • Magnusson, B.M.1    Anissimov, Y.G.2    Cross, S.E.3    Roberts, M.S.4
  • 14
    • 84861094256 scopus 로고    scopus 로고
    • An integrated approach to optimizing skin delivery of cosmetic and pharmaceutical actives
    • Abbott, S., An integrated approach to optimizing skin delivery of cosmetic and pharmaceutical actives. Int. J. Cosmet. Sci. 34, 217-222 (2012).
    • (2012) Int. J. Cosmet. Sci. , vol.34 , pp. 217-222
    • Abbott, S.1
  • 15
    • 84864283652 scopus 로고    scopus 로고
    • The influence of volatile solvents on transport across model membranes and human skin
    • Oliveira, G., Hadgraft, J., and, Lane, M.E., The influence of volatile solvents on transport across model membranes and human skin. Int. J. Pharm. 435, 38-49 (2012).
    • (2012) Int. J. Pharm. , vol.435 , pp. 38-49
    • Oliveira, G.1    Hadgraft, J.2    Lane, M.E.3
  • 16
    • 74049132487 scopus 로고    scopus 로고
    • Relative uptake of minoxidil into appendages and stratum corneum and permeation through human skin in vitro
    • Grice, J.E., Ciotti, S.N., Weiner, N., Lockwood, P., Cross, S.E., and, Roberts, M.S., Relative uptake of minoxidil into appendages and stratum corneum and permeation through human skin in vitro. J. Pharm. Sci. 99, 712-718 (2010).
    • (2010) J. Pharm. Sci. , vol.99 , pp. 712-718
    • Grice, J.E.1    Ciotti, S.N.2    Weiner, N.3    Lockwood, P.4    Cross, S.E.5    Roberts, M.S.6
  • 17
    • 85027932244 scopus 로고    scopus 로고
    • Effect of vehicles on the maximum transepidermal flux of similar size phenolic compounds
    • DOI: 10.1007/s11095-012-0846-x
    • Zhang, Q., Li, P., Liu, D., and, Roberts, M.S., Effect of vehicles on the maximum transepidermal flux of similar size phenolic compounds. Pharm. Res. DOI: 10.1007/s11095-012-0846-x (2012).
    • (2012) Pharm. Res.
    • Zhang, Q.1    Li, P.2    Liu, D.3    Roberts, M.S.4
  • 18
    • 0002113356 scopus 로고    scopus 로고
    • The relationship between structure and barrier function of skin
    • (Roberts, M.S. and Walters, K.A. eds), Marcel Dekker, New York
    • Roberts, M.S., and, Walters, K.A., The relationship between structure and barrier function of skin. In: Dermal Absorption and Toxicity Assessment (, Roberts, M.S., and, Walters, K.A., eds), pp. 1-42. Marcel Dekker, New York (1998).
    • (1998) Dermal Absorption and Toxicity Assessment , pp. 1-42
    • Roberts, M.S.1    Walters, K.A.2
  • 19
    • 0024375494 scopus 로고
    • Effect of several enhancers on the skin permeation of water soluble drugs
    • Okumura, M., Sugibayashi, K., and, Morimoto, Y., Effect of several enhancers on the skin permeation of water soluble drugs. Chem. Pharm. Bull. 37, 1375-1378 (1989).
    • (1989) Chem. Pharm. Bull. , vol.37 , pp. 1375-1378
    • Okumura, M.1    Sugibayashi, K.2    Morimoto, Y.3
  • 21
    • 33750507126 scopus 로고    scopus 로고
    • Microemulsions as transdermal drug delivery vehicles
    • Kogan, A., and, Garti, N., Microemulsions as transdermal drug delivery vehicles. Adv. Colloid Interface Sci., 123-126, 369-385 (2006).
    • (2006) Adv. Colloid Interface Sci. , vol.123-126 , pp. 369-385
    • Kogan, A.1    Garti, N.2
  • 22
    • 0034602595 scopus 로고    scopus 로고
    • NMR characterization and transdermal drug delivery potential of microemulsion systems
    • Kreilgaard, M., Pedersen, E.J., and, Jaroszewski, J.W., NMR characterization and transdermal drug delivery potential of microemulsion systems. J. Control Release 69, 421-433 (2000).
    • (2000) J. Control Release , vol.69 , pp. 421-433
    • Kreilgaard, M.1    Pedersen, E.J.2    Jaroszewski, J.W.3
  • 24
    • 0029869326 scopus 로고    scopus 로고
    • Effect of nonionic surfactants on the percutaneous absorption of tenoxicam
    • Endo, M., Yamamoto, T., and, Ijuin, T., Effect of nonionic surfactants on the percutaneous absorption of tenoxicam. Chem. Pharm. Bull. (Tokyo) 44, 865-867 (1996).
    • (1996) Chem. Pharm. Bull. (Tokyo) , vol.44 , pp. 865-867
    • Endo, M.1    Yamamoto, T.2    Ijuin, T.3
  • 25
    • 0036025240 scopus 로고    scopus 로고
    • Transdermal delivery of physostigmine: Effects of enhancers and pressure sensitive adhesives
    • Kim, J.H., Lee, C.H., and, Choi, H.K., Transdermal delivery of physostigmine: effects of enhancers and pressure sensitive adhesives. Drug Dev. Ind. Pharm. 28, 833-839 (2002).
    • (2002) Drug Dev. Ind. Pharm. , vol.28 , pp. 833-839
    • Kim, J.H.1    Lee, C.H.2    Choi, H.K.3
  • 26
    • 34248586701 scopus 로고    scopus 로고
    • Development and evaluation of carvedilol transdermal patches
    • Tanwar, Y.S., Chauhan, C.S., and, Sharma, A., Development and evaluation of carvedilol transdermal patches. Acta Pharm. 57, 151-159 (2007).
    • (2007) Acta Pharm. , vol.57 , pp. 151-159
    • Tanwar, Y.S.1    Chauhan, C.S.2    Sharma, A.3
  • 27
    • 0035902683 scopus 로고    scopus 로고
    • Effects of non-ionic surfactants as permeation enhancers towards piroxicam from the poloxamer gel through rat skins
    • Shin, S.-C., Cho, C.-W., and, Oh, I.-J., Effects of non-ionic surfactants as permeation enhancers towards piroxicam from the poloxamer gel through rat skins. Int. J. Pharm. 222, 199-203 (2001).
    • (2001) Int. J. Pharm. , vol.222 , pp. 199-203
    • Shin, S.-C.1    Cho, C.-W.2    Oh, I.-J.3
  • 28
    • 34547676276 scopus 로고    scopus 로고
    • Skin permeation of ketotifen applied from a stick-type formulation
    • Kimura, C., Nakanishi, T., and, Tojo, K., Skin permeation of ketotifen applied from a stick-type formulation. Eur. J. Pharm. Biopharm. 67, 420-424 (2007).
    • (2007) Eur. J. Pharm. Biopharm. , vol.67 , pp. 420-424
    • Kimura, C.1    Nakanishi, T.2    Tojo, K.3
  • 29
    • 0032427652 scopus 로고    scopus 로고
    • In vitro human epidermal and polyethylene membrane and penetration of the sunscreen benzophenone-3 from a range of solvents
    • Jiang, R., Benson, H.A.E., Cross, S.E., and, Roberts, M.S., In vitro human epidermal and polyethylene membrane and penetration of the sunscreen benzophenone-3 from a range of solvents. Pharm. Res. 15, 1863-1868 (1998).
    • (1998) Pharm. Res. , vol.15 , pp. 1863-1868
    • Jiang, R.1    Benson, H.A.E.2    Cross, S.E.3    Roberts, M.S.4
  • 30
    • 70349521554 scopus 로고    scopus 로고
    • (Accessed August 2012)
    • Anon. J.M. Keynes. In Wikiquote http://en.wiki.quote.org/wiki/John- Maynard-Keynes (Accessed August 2012)
    • Wikiquote
    • Keynes, A.J.M.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.