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Volumn 120, Issue 1, 2012, Pages 36-44

Antidiabetic effects of SGLT2-selective inhibitor ipragliflozin in streptozotocin-nicotinamide-induced mildly diabetic mice

Author keywords

Diabetes; Hyperglycemia; Ipragliflozin; SGLT2; Urinary glucose excretion

Indexed keywords

INSULIN; IPRAGLIFLOZIN; SODIUM GLUCOSE COTRANSPORTER 2;

EID: 84866541730     PISSN: 13478613     EISSN: 13478648     Source Type: Journal    
DOI: 10.1254/jphs.12089FP     Document Type: Article
Times cited : (38)

References (29)
  • 1
    • 0033842027 scopus 로고    scopus 로고
    • Interactions between insulin resistance and insulin secretion in the development of glucose intolerance
    • Cavaghan MK, Ehrmann DA, Polonsky KS. Interactions between insulin resistance and insulin secretion in the development of glucose intolerance. J Clin Invest. 2000;106:329-333.
    • (2000) J Clin Invest , vol.106 , pp. 329-333
    • Cavaghan, M.K.1    Ehrmann, D.A.2    Polonsky, K.S.3
  • 2
    • 58149357463 scopus 로고    scopus 로고
    • Sodium-glucose co-transporter-2 inhibitors: An emerging new class of oral antidiabetic drug
    • Idris I, Donnelly R. Sodium-glucose co-transporter-2 inhibitors: an emerging new class of oral antidiabetic drug. Diabetes Obes Metab. 2009;11:79-88.
    • (2009) Diabetes Obes Metab , vol.11 , pp. 79-88
    • Idris, I.1    Donnelly, R.2
  • 3
    • 1242272759 scopus 로고    scopus 로고
    • The sodium/glucose cotransport family SLC5
    • Wright EM, Turk E. The sodium/glucose cotransport family SLC5. Pflugers Arch. 2004;447:510-518.
    • (2004) Pflugers Arch , vol.447 , pp. 510-518
    • Wright, E.M.1    Turk, E.2
  • 4
    • 0026761353 scopus 로고
    • Cloning and functional expression of a mammalian Na+/nucleoside cotransporter. A member of the SGLT family
    • Pajor AM, Wright EM. Cloning and functional expression of a mammalian Na+/nucleoside cotransporter. A member of the SGLT family. J Biol Chem. 1992;267:3557-3560.
    • (1992) J Biol Chem , vol.267 , pp. 3557-3560
    • Pajor, A.M.1    Wright, E.M.2
  • 5
    • 0025891622 scopus 로고
    • Glucose/galactose malabsorption caused by a defect in the Na+/glucose cotransporter
    • Turk E, Zabel B, Mundlos S, Dyer J, Wright EM. Glucose/galactose malabsorption caused by a defect in the Na+/glucose cotransporter. Nature. 1991;350:354-356.
    • (1991) Nature , vol.350 , pp. 354-356
    • Turk, E.1    Zabel, B.2    Mundlos, S.3    Dyer, J.4    Wright, E.M.5
  • 7
    • 0036937335 scopus 로고    scopus 로고
    • Autosomal recessive renal glucosuria attributable to a mutation in the sodium glucose cotransporter (SGLT2)
    • van den Heuvel LP, Assink K, Willemsen M, Monnens L. Autosomal recessive renal glucosuria attributable to a mutation in the sodium glucose cotransporter (SGLT2). Hum Genet. 2002;111: 544-547.
    • (2002) Hum Genet , vol.111 , pp. 544-547
    • Van Den Heuvel, L.P.1    Assink, K.2    Willemsen, M.3    Monnens, L.4
  • 8
    • 0025074647 scopus 로고
    • Insulin resistance in rats with non-insulin-dependent diabetes induced by neonatal (5 days) streptozotocin: Evidence for reversal following phlorizin treatment
    • Blondel O, Bailbe D, Portha B. Insulin resistance in rats with non-insulin-dependent diabetes induced by neonatal (5 days) streptozotocin: evidence for reversal following phlorizin treatment. Metabolism. 1990;39:787-793.
    • (1990) Metabolism , vol.39 , pp. 787-793
    • Blondel, O.1    Bailbe, D.2    Portha, B.3
  • 9
    • 0023275573 scopus 로고
    • Correction of hyperglycemia with phlorizin normalizes tissue sensitivity to insulin in diabetic rats
    • Rossetti L, Smith D, Shulman GI, Papachristou D, DeFronzo RA. Correction of hyperglycemia with phlorizin normalizes tissue sensitivity to insulin in diabetic rats. J Clin Invest. 1987; 79:1510-1515.
    • (1987) J Clin Invest , vol.79 , pp. 1510-1515
    • Rossetti, L.1    Smith, D.2    Shulman, G.I.3    Papachristou, D.4    DeFronzo, R.A.5
  • 10
    • 0026033325 scopus 로고
    • Normalization of blood glucose in diabetic rats with phlorizin treatment reverses insulin-resistant glucose transport in adipose cells without restoring glucose transporter gene expression
    • Kahn BB, Shulman GI, DeFronzo RA, Cushman SW, Rossetti L. Normalization of blood glucose in diabetic rats with phlorizin treatment reverses insulin-resistant glucose transport in adipose cells without restoring glucose transporter gene expression. J Clin Invest. 1991;87:561-570.
    • (1991) J Clin Invest , vol.87 , pp. 561-570
    • Kahn, B.B.1    Shulman, G.I.2    DeFronzo, R.A.3    Cushman, S.W.4    Rossetti, L.5
  • 12
    • 0032850016 scopus 로고    scopus 로고
    • T-1095, an inhibitor of renal Na+-glucose cotransporters, may provide a novel approach to treating diabetes
    • Oku A, Ueta K, Arakawa K, Ishihara T, Nawano M, Kuronuma Y, et al. T-1095, an inhibitor of renal Na+-glucose cotransporters, may provide a novel approach to treating diabetes. Diabetes. 1999;48:1794-1800.
    • (1999) Diabetes , vol.48 , pp. 1794-1800
    • Oku, A.1    Ueta, K.2    Arakawa, K.3    Ishihara, T.4    Nawano, M.5    Kuronuma, Y.6
  • 13
    • 48249146624 scopus 로고    scopus 로고
    • Dapagliflozin, a selective SGLT2 inhibitor, improves glucose homeostasis in normal and diabetic rats
    • Han S, Hagan DL, Taylor JR, Xin L, Meng W, Biller SA, et al. Dapagliflozin, a selective SGLT2 inhibitor, improves glucose homeostasis in normal and diabetic rats. Diabetes. 2008;57: 1723-1729.
    • (2008) Diabetes , vol.57 , pp. 1723-1729
    • Han, S.1    Hagan, D.L.2    Taylor, J.R.3    Xin, L.4    Meng, W.5    Biller, S.A.6
  • 15
    • 58149119432 scopus 로고    scopus 로고
    • Effects of antidiabetic drugs on glucose tolerance in streptozotocin-nicotinamide-induced mildly diabetic and streptozotocin-induced severely diabetic mice
    • Tahara A, Matsuyama-Yokono A, Nakano R, Someya Y, Shibasaki M. Effects of antidiabetic drugs on glucose tolerance in streptozotocin-nicotinamide-induced mildly diabetic and streptozotocin-induced severely diabetic mice. Horm Metab Res. 2008;40:880-886.
    • (2008) Horm Metab Res , vol.40 , pp. 880-886
    • Tahara, A.1    Matsuyama-Yokono, A.2    Nakano, R.3    Someya, Y.4    Shibasaki, M.5
  • 16
    • 58749113105 scopus 로고    scopus 로고
    • Evaluation of the antidiabetic effects of dipeptidyl peptidase-IV inhibitor ASP8497 in streptozotocin-nicotinamide-induced mildly diabetic mice
    • Tahara A, Matsuyama-Yokono A, Nakano R, Someya Y, Hayakawa M, Shibasaki M. Evaluation of the antidiabetic effects of dipeptidyl peptidase-IV inhibitor ASP8497 in streptozotocin-nicotinamide-induced mildly diabetic mice. Pharmacology. 2009; 83:177-187.
    • (2009) Pharmacology , vol.83 , pp. 177-187
    • Tahara, A.1    Matsuyama-Yokono, A.2    Nakano, R.3    Someya, Y.4    Hayakawa, M.5    Shibasaki, M.6
  • 17
    • 64549093267 scopus 로고    scopus 로고
    • Sergliflozin etabonate, a selective SGLT2 inhibitor, improves glycemic control in streptozotocin-induced diabetic rats and Zucker fatty rats
    • Fujimori Y, Katsuno K, Ojima K, Nakashima I, Nakano S, Ishikawa-Takemura Y, et al. Sergliflozin etabonate, a selective SGLT2 inhibitor, improves glycemic control in streptozotocin-induced diabetic rats and Zucker fatty rats. Eur J Pharmacol. 2009;609:148-154.
    • (2009) Eur J Pharmacol , vol.609 , pp. 148-154
    • Fujimori, Y.1    Katsuno, K.2    Ojima, K.3    Nakashima, I.4    Nakano, S.5    Ishikawa-Takemura, Y.6
  • 18
    • 0033619999 scopus 로고    scopus 로고
    • Na+-glucose cotransporter (SGLT) inhibitors as antidiabetic agents. 4. Synthesis and pharmacological properties of 4′-dehydroxyphlorizin derivatives substituted on the B ring
    • Tsujihara K, Hongu M, Saito K, Kawanishi H, Kuriyama K, Matsumoto M, et al. Na+-glucose cotransporter (SGLT) inhibitors as antidiabetic agents. 4. Synthesis and pharmacological properties of 4′-dehydroxyphlorizin derivatives substituted on the B ring. J Med Chem. 1999;42:5311-5324.
    • (1999) J Med Chem , vol.42 , pp. 5311-5324
    • Tsujihara, K.1    Hongu, M.2    Saito, K.3    Kawanishi, H.4    Kuriyama, K.5    Matsumoto, M.6
  • 20
    • 0032983666 scopus 로고    scopus 로고
    • Glycemic control with diet, sulfonylurea, metformin, or insulin in patients with type 2 diabetes mellitus: Progressive requirement for multiple therapies (UKPDS 49)
    • Turner RC, Cull CA, Frighi V, Holman RR. Glycemic control with diet, sulfonylurea, metformin, or insulin in patients with type 2 diabetes mellitus: progressive requirement for multiple therapies (UKPDS 49). JAMA. 1999;281:2005-2012.
    • (1999) JAMA , vol.281 , pp. 2005-2012
    • Turner, R.C.1    Cull, C.A.2    Frighi, V.3    Holman, R.R.4
  • 21
    • 0028232045 scopus 로고
    • Secondary failure of oral hypoglycaemic agents: Frequency, possible causes, and management
    • Pontiroli AE, Calderara A, Pozza G. Secondary failure of oral hypoglycaemic agents: frequency, possible causes, and management. Diabetes Metab Rev. 1994;10:31-43.
    • (1994) Diabetes Metab Rev , vol.10 , pp. 31-43
    • Pontiroli, A.E.1    Calderara, A.2    Pozza, G.3
  • 22
    • 0031972156 scopus 로고    scopus 로고
    • UKPDS 26: Sulphonylurea failure in non-insulin-dependent diabetic patients over six years
    • UK Prospective Diabetes Study (UKPDS) Group
    • Matthews DR, Cull CA, Stratton IM, Holman RR, Turner RC. UKPDS 26: Sulphonylurea failure in non-insulin-dependent diabetic patients over six years. UK Prospective Diabetes Study (UKPDS) Group. Diabet Med. 1998;15:297-303.
    • (1998) Diabet Med , vol.15 , pp. 297-303
    • Matthews, D.R.1    Cull, C.A.2    Stratton, I.M.3    Holman, R.R.4    Turner, R.C.5
  • 23
    • 59649108238 scopus 로고    scopus 로고
    • Antidiabetic effects of dipeptidyl peptidase-IV inhibitors and sulfonylureas in streptozotocin-nicotinamide-induced mildly diabetic mice
    • Matsuyama-Yokono A, Tahara A, Nakano R, Someya Y, Shiraki K, Hayakawa M, et al. Antidiabetic effects of dipeptidyl peptidase-IV inhibitors and sulfonylureas in streptozotocin-nicotinamide-induced mildly diabetic mice. Metabolism. 2009;58:379-386.
    • (2009) Metabolism , vol.58 , pp. 379-386
    • Matsuyama-Yokono, A.1    Tahara, A.2    Nakano, R.3    Someya, Y.4    Shiraki, K.5    Hayakawa, M.6
  • 24
    • 0030907293 scopus 로고    scopus 로고
    • Parallel reduction of pancreas insulin content and insulin secretion in 48-h tolbutamide-infused normoglycemic rats
    • Hosokawa YA, Leahy JL. Parallel reduction of pancreas insulin content and insulin secretion in 48-h tolbutamide-infused normoglycemic rats. Diabetes. 1997;46:808-813.
    • (1997) Diabetes , vol.46 , pp. 808-813
    • Hosokawa, Y.A.1    Leahy, J.L.2
  • 25
    • 0029783411 scopus 로고    scopus 로고
    • Beta-cell dysfunction with chronic hyperglycemia: "overworked beta-cell" hypothesis
    • Leahy JL. Beta-cell dysfunction with chronic hyperglycemia: "overworked beta-cell" hypothesis. Diabetes Rev. 1996;4:298-319.
    • (1996) Diabetes Rev , vol.4 , pp. 298-319
    • Leahy, J.L.1
  • 26
    • 0034845814 scopus 로고    scopus 로고
    • Beta-cell function evaluated by HOMA as a predictor of secondary sulphonylurea failure in Type 2 diabetes
    • Taverna MJ, Pacher N, Bruzzo F, Slama G, Selam JL. Beta-cell function evaluated by HOMA as a predictor of secondary sulphonylurea failure in Type 2 diabetes. Diabet Med. 2001;18: 584-588.
    • (2001) Diabet Med , vol.18 , pp. 584-588
    • Taverna, M.J.1    Pacher, N.2    Bruzzo, F.3    Slama, G.4    Selam, J.L.5
  • 27
    • 0032835391 scopus 로고    scopus 로고
    • Unresponsiveness to glibenclamide during chronic treatment induced by reduction of ATP-sensitive K+ channel activity
    • Kawaki J, Nagashima K, Tanaka J, Miki T, Miyazaki M, Gonoi T, et al. Unresponsiveness to glibenclamide during chronic treatment induced by reduction of ATP-sensitive K+ channel activity. Diabetes. 1999;48:2001-2006.
    • (1999) Diabetes , vol.48 , pp. 2001-2006
    • Kawaki, J.1    Nagashima, K.2    Tanaka, J.3    Miki, T.4    Miyazaki, M.5    Gonoi, T.6
  • 28
    • 77953181310 scopus 로고    scopus 로고
    • Dapagliflozin treatment in patients with different stages of type 2 diabetes mellitus: Effects on glycaemic control and body weight
    • Zhang L, Feng Y, List J, Kasichayanula S, Pfister M. Dapagliflozin treatment in patients with different stages of type 2 diabetes mellitus: effects on glycaemic control and body weight. Diabetes Obes Metab. 2010;12:510-516.
    • (2010) Diabetes Obes Metab , vol.12 , pp. 510-516
    • Zhang, L.1    Feng, Y.2    List, J.3    Kasichayanula, S.4    Pfister, M.5
  • 29
    • 84864371186 scopus 로고    scopus 로고
    • Weight loss induced by chronic dapagliflozin treatment is attenuated by compensatory hyperphagia in diet-induced obese (DIO) rats
    • Silver Spring
    • Devenny JJ, Godonis HE, Harvey SJ, Rooney S, Cullen MJ, Pelleymounter MA. Weight loss induced by chronic dapagliflozin treatment is attenuated by compensatory hyperphagia in diet-induced obese (DIO) rats. Obesity (Silver Spring). 2012;20:1645-1652.
    • (2012) Obesity , vol.20 , pp. 1645-1652
    • Devenny, J.J.1    Godonis, H.E.2    Harvey, S.J.3    Rooney, S.4    Cullen, M.J.5    Pelleymounter, M.A.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.