SCOPUS 정보 검색 플랫폼

Volumn 3, Issue 9, 2012, Pages 1111-1116

Design and synthesis of trans-2-substituted-cyclopropane-1-carboxylic acids as the first non-natural small molecule inhibitors of O-acetylserine sulfhydrylase

(7) Amori, Laura a Katkevica, Sarmite a,c Bruno, Agostino a Campanini, Barbara a Felici, Paolo a Mozzarelli, Andrea a,b Costantino, Gabriele a

a UNIVERSITY OF PARMA (Italy)

b National Institute of Biostructure and Biosystems (Italy)

c LATVIAN INSTITUTE OF ORGANIC SYNTHESIS (Latvia)

Author keywords

[No Author keywords available]

Indexed keywords

CYCLOPROPANE DERIVATIVE; CYSTEINE SYNTHASE; ENZYME INHIBITOR; PENTAPEPTIDE; SYNTHETIC PEPTIDE; TRANS 2 SUBSTITUTED CYCLOPROPANE 1 CARBOXYLIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG DESIGN; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; HAEMOPHILUS INFLUENZAE TYPE A; MOLECULAR MODEL; MOLECULAR SIZE; NONHUMAN; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN BINDING;

BACTERIA (MICROORGANISMS); HAEMOPHILUS INFLUENZAE;

EID: 84865490293 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c2md20100c Document Type: Article

Times cited : (38)

References (35)

1
- 69549111337
- M. A. Fischbach C. T. Walsh Science 2009 325 1089 1093
- (2009) Science , vol.325 , pp. 1089-1093
- Fischbach, M.A.¹ Walsh, C.T.²

2
- 0038587681
- M. R. Barbachyn C. W. Ford Angew. Chem., Int. Ed. 2003 42 2010 2023
- (2003) Angew. Chem., Int. Ed. , vol.42 , pp. 2010-2023
- Barbachyn, M.R.¹ Ford, C.W.²

3
- 2342595765
- B. Spellberg J. H. Powers E. P. Brass L. G. Miller J. E. Edwards Jr Clin. Infect. Dis. 2004 38 1279 1286
- (2004) Clin. Infect. Dis. , vol.38 , pp. 1279-1286
- Spellberg, B.¹ Powers, J.H.² Brass, E.P.³ Miller, L.G.⁴ Edwards Jr., J.E.⁵

4
- 23444460075
- J. Conly B. Johnston Can. J. Infect. Dis. Med. Microbiol. 2005 16 159 160
- (2005) Can. J. Infect. Dis. Med. Microbiol. , vol.16 , pp. 159-160
- Conly, J.¹ Johnston, B.²

5
- 33644761913
- W. Kern Int. J. Clin. Pract. 2006 60 370 378
- (2006) Int. J. Clin. Pract. , vol.60 , pp. 370-378
- Kern, W.¹

6
- 0020686355
- A. J. Cooper Annu. Rev. Biochem. 1983 52 187 222
- (1983) Annu. Rev. Biochem. , vol.52 , pp. 187-222
- Cooper, A.J.¹

7
- 0033995794
- A. Sekowska H. F. Kung A. Danchin J. Mol. Microbiol. Biotechnol. 2000 2 145 177
- (2000) J. Mol. Microbiol. Biotechnol. , vol.2 , pp. 145-177
- Sekowska, A.¹ Kung, H.F.² Danchin, A.³

8
- 0033829523
- H. Beinert Eur. J. Biochem. 2000 267 5657 5664
- (2000) Eur. J. Biochem. , vol.267 , pp. 5657-5664
- Beinert, H.¹

9
- 33750083296
- D. Kessler FEMS Microbiol. Rev. 2006 30 825 840
- (2006) FEMS Microbiol. Rev. , vol.30 , pp. 825-840
- Kessler, D.¹

10
- 80054687027
- A. Mozzarelli S. Bettati B. Campanini E. Salsi S. Raboni R. Syngh F. Spyrakis V. P. Kumar P. F. Cook Biochim. Biophys. Acta, Proteins Proteomics 2011 1814 1497 1510
- (2011) Biochim. Biophys. Acta, Proteins Proteomics , vol.1814 , pp. 1497-1510
- Mozzarelli, A.¹ Bettati, S.² Campanini, B.³ Salsi, E.⁴ Raboni, S.⁵ Syngh, R.⁶ Spyrakis, F.⁷ Kumar, V.P.⁸ Cook, P.F.⁹

11
- 77957256320
- A. L. Turnbull M. G. Surette Res. Microbiol. 2010 161 643 650
- (2010) Res. Microbiol. , vol.161 , pp. 643-650
- Turnbull, A.L.¹ Surette, M.G.²

12
- 77952310116
- R. Schnell G. Schneider Biochem. Biophys. Res. Commun. 2010 396 33 38
- (2010) Biochem. Biophys. Res. Commun. , vol.396 , pp. 33-38
- Schnell, R.¹ Schneider, G.²

13
- 0027183564
- C. H. Tai S. R. Nalabolu T. M. Jacobson D. E. Minter P. F. Cook Biochemistry 1993 32 6433 6644
- (1993) Biochemistry , vol.32 , pp. 6433-6644
- Tai, C.H.¹ Nalabolu, S.R.² Jacobson, T.M.³ Minter, D.E.⁴ Cook, P.F.⁵

14
- 77951212184
- E. Salsi B. Campanini S. Bettati S. Raboni S. L. Roderick P. F. Cook A. Mozzarelli J. Biol. Chem. 2010 285 12813 12822
- (2010) J. Biol. Chem. , vol.285 , pp. 12813-12822
- Salsi, E.¹ Campanini, B.² Bettati, S.³ Raboni, S.⁴ Roderick, S.L.⁵ Cook, P.F.⁶ Mozzarelli, A.⁷

15
- 23644440099
- B. Campanini F. Speroni E. Salsi P. F. Cook S. L. Roderick B. Huang S. Bettati A. Mozzarelli Protein Sci. 2005 14 2115 2124
- (2005) Protein Sci. , vol.14 , pp. 2115-2124
- Campanini, B.¹ Speroni, F.² Salsi, E.³ Cook, P.F.⁴ Roderick, S.L.⁵ Huang, B.⁶ Bettati, S.⁷ Mozzarelli, A.⁸

16
- 32344445371
- C. Zhao Y. Moriga B. Feng Y. Kumada H. Imanaka K. Imamura K. Nakanishi Biochem. Biophys. Res. Commun. 2006 341 911 916
- (2006) Biochem. Biophys. Res. Commun. , vol.341 , pp. 911-916
- Zhao, C.¹ Moriga, Y.² Feng, B.³ Kumada, Y.⁴ Imanaka, H.⁵ Imamura, K.⁶ Nakanishi, K.⁷

17
- 65649133057
- S. Kumaran H. Yi H. B. Krishnan J. M. Jez J. Biol. Chem. 2010 284 10268 10275
- (2010) J. Biol. Chem. , vol.284 , pp. 10268-10275
- Kumaran, S.¹ Yi, H.² Krishnan, H.B.³ Jez, J.M.⁴

18
- 57349162179
- A. L. Turnbull M. G. Surette Microbiology 2008 154 3410 3419
- (2008) Microbiology , vol.154 , pp. 3410-3419
- Turnbull, A.L.¹ Surette, M.G.²

19
- 0034278207
- K. Mino K. Hiraoka K. Imamura T. Sakiyama N. Eisaki A. Matsuyama K. Nakanishi Biosci., Biotechnol., Biochem. 2000 64 1874 1880
- (2000) Biosci., Biotechnol., Biochem. , vol.64 , pp. 1874-1880
- Mino, K.¹ Hiraoka, K.² Imamura, K.³ Sakiyama, T.⁴ Eisaki, N.⁵ Matsuyama, A.⁶ Nakanishi, K.⁷

20
- 0344157394
- P. Burkhard G. S. Rao E. Hohenester K. D. Schnackerz P. F. Cook J. N. Jansonius J. Mol. Biol. 1998 283 121 133
- (1998) J. Mol. Biol. , vol.283 , pp. 121-133
- Burkhard, P.¹ Rao, G.S.² Hohenester, E.³ Schnackerz, K.D.⁴ Cook, P.F.⁵ Jansonius, J.N.⁶

21
- 0033609810
- P. Burkhard C. H. Tai C. M. Ristroph P. F. Cook J. N. Jansonius J. Mol. Biol. 1999 291 941 953
- (1999) J. Mol. Biol. , vol.291 , pp. 941-953
- Burkhard, P.¹ Tai, C.H.² Ristroph, C.M.³ Cook, P.F.⁴ Jansonius, J.N.⁵

22
- 16644396746
- J. Gorman L. Shapiro Acta Crystallogr., Sect. D: Biol. Crystallogr. 2004 60 1600 1605
- (2004) Acta Crystallogr., Sect. D: Biol. Crystallogr. , vol.60 , pp. 1600-1605
- Gorman, J.¹ Shapiro, L.²

23
- 2442644099
- L. R. Olsen B. Huang M. W. Vetting S. L. Roderick Biochemistry 2004 43 6013 6019
- (2004) Biochemistry , vol.43 , pp. 6013-6019
- Olsen, L.R.¹ Huang, B.² Vetting, M.W.³ Roderick, S.L.⁴

24
- 4644272171
- V. E. Pye A. P. Tingey R. L. Robson P. C. Moody J. Biol. Chem. 2004 279 40729 40736
- (2004) J. Biol. Chem. , vol.279 , pp. 40729-40736
- Pye, V.E.¹ Tingey, A.P.² Robson, R.L.³ Moody, P.C.⁴

25
- 17644423923
- B. Huang M. W. Vetting S. L. Roderick J. Bacteriol. 2005 187 3201 3205
- (2005) J. Bacteriol. , vol.187 , pp. 3201-3205
- Huang, B.¹ Vetting, M.W.² Roderick, S.L.³

26
- 74849085165
- E. Salsi A. S. Bayden F. Spyrakis A. Amadasi B. Campanini S. Bettati T. Dodatko P. Cozzini G. E. Kellogg P. F. Cook S. L. Roderick A. Mozzarelli J. Med. Chem. 2010 53 345 356
- (2010) J. Med. Chem. , vol.53 , pp. 345-356
- Salsi, E.¹ Bayden, A.S.² Spyrakis, F.³ Amadasi, A.⁴ Campanini, B.⁵ Bettati, S.⁶ Dodatko, T.⁷ Cozzini, P.⁸ Kellogg, G.E.⁹ Cook, P.F.¹⁰ Roderick, S.L.¹¹ Mozzarelli, A.¹²

27
- 33746898558
- A. Reichelt S. F. Martin Acc. Chem. Res. 2006 39 433 442
- (2006) Acc. Chem. Res. , vol.39 , pp. 433-442
- Reichelt, A.¹ Martin, S.F.²

28
- 0028999843
- J. Salaun M. S. Baird Curr. Med. Chem. 1995 2 511 542
- (1995) Curr. Med. Chem. , vol.2 , pp. 511-542
- Salaun, J.¹ Baird, M.S.²

29
- 33846191100
- S. I. Kozhushkov H. Schill Chem. Rev. 2006 106 4926 4996
- (2006) Chem. Rev. , vol.106 , pp. 4926-4996
- Kozhushkov, S.I.¹ Schill, H.²

30
- 33646765763
- R. Pellicciari R. C. Rizzo G. Costantino M. Marinozzi L. Amori P. Guidetti H. Q. Wu R. Schwarcz ChemMedChem 2006 1 528 531
- (2006) ChemMedChem , vol.1 , pp. 528-531
- Pellicciari, R.¹ Rizzo, R.C.² Costantino, G.³ Marinozzi, M.⁴ Amori, L.⁵ Guidetti, P.⁶ Wu, H.Q.⁷ Schwarcz, R.⁸

31
- 0028174296
- G. D. McClure Jr P. F. Cook Biochemistry 1994 33 1674 1683
- (1994) Biochemistry , vol.33 , pp. 1674-1683
- McClure Jr., G.D.¹ Cook, P.F.²

32
- 23944514165
- John Wiley & Sons, Inc.
- R. A. Copeland, Evaluation of Enzyme Inhibitors in Drug Discovery: a Guide for Medicinal Chemists and Pharmacologists, John Wiley & Sons, Inc., 2005
- (2005) Evaluation of Enzyme Inhibitors in Drug Discovery: A Guide for Medicinal Chemists and Pharmacologists
- Copeland, R.A.¹

33
- 0003760238
- John Wiley & Sons, Inc.
- I. H. Segel, Enzymes Kinetics. Behavior and Analysis of Rapid Equilibrium and Steady-State Enzyme Systems, John Wiley & Sons, Inc., 1993
- (1993) Enzymes Kinetics. Behavior and Analysis of Rapid Equilibrium and Steady-State Enzyme Systems
- Segel, I.H.¹

34
- 84857099645
- I. Nagpal I. Raj N. Subbarao S. Gourinath PLoS One 2012 7 e30305
- (2012) PLoS One , vol.7 , pp. 30305
- Nagpal, I.¹ Raj, I.² Subbarao, N.³ Gourinath, S.⁴

35
- 84865513144
- LLC, New York
- Maestro, Version 9.1, Schroedinger, LLC, New York, 2010
- (2010) Maestro, Version 9.1, Schroedinger

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.