The development of first Staphylococcus aureus SplB protease inhibitors: Phosphonic analogues of glutamine

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 17, 2012, Pages 5574-5578

  Ewa, Burchacka ^a   MacIej, Walczak ^a   Marcin, Sieńczyk ^a   Grzegorz, Dubin ^b   Michał, Zdzalik ^b   Jan, Potempa ^b   Józef, Oleksyszyn ^a  

^a WROCLAW UNIVERSITY OF TECHNOLOGY   (Poland)

^b JAGIELLONIAN UNIVERSITY   (Poland)

Author keywords

Aminoalkylphosphonates; Serine protease inhibitors; SplB protease; Staphylococcus aureus

Indexed keywords

BACTERIAL ENZYME; CHYMOTRYPSIN; GLUTAMINE DERIVATIVE; PHOSPHORAMIDIC ACID DERIVATIVE; SERINE PROTEINASE; SERINE PROTEINASE INHIBITOR; SPLB SERINE PROTEINASE; SPLB SERINE PROTEINASE INHIBITOR; SUBTILISIN; UNCLASSIFIED DRUG;

ARTICLE; ENZYME INHIBITION; NONHUMAN; PROTEIN FUNCTION; STAPHYLOCOCCUS AUREUS;

GLUTAMINE; HUMANS; SERINE PROTEASES; SERINE PROTEINASE INHIBITORS; STAPHYLOCOCCAL INFECTIONS; STAPHYLOCOCCUS AUREUS;

STAPHYLOCOCCUS AUREUS;

EID: 84865115539     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.07.011     Document Type: Article

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