A fluorescent reporter of ATP binding-competent receptor kinases

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 17, 2012, Pages 5532-5535

  Sicard, Renaud ^a   Dhuguru, Jyothi ^b   Liu, Wenjun ^a   Patel, Nirav ^a   Landgraf, Ralf ^a   Wilson, James N ^b  

^a UNIVERSITY OF MIAMI MILLER SCHOOL OF MEDICINE   (United States)

^b University of Miami   (United States)

Author keywords

EGFR; ERBB2; Fluorescent probes; Kinase inhibitors; Quinazoline

Indexed keywords

6 (4 DIMETHYL AMINOSTYRYL) N BENZYLQUINAZOLIN 4 AMINE; ADENOSINE TRIPHOSPHATE; EPIDERMAL GROWTH FACTOR RECEPTOR 2; FLUORESCENT DYE; UNCLASSIFIED DRUG;

ARTICLE; AUTOPHOSPHORYLATION; CONTROLLED STUDY; FLUORESCENCE; HUMAN; HUMAN CELL; HYDROPHOBICITY; IN VITRO STUDY; MOLECULAR PROBE; RECEPTOR BINDING; RECEPTOR OCCUPANCY;

ADENOSINE TRIPHOSPHATE; BINDING SITES; BREAST NEOPLASMS; CELL LINE, TUMOR; CELL SURVIVAL; FEMALE; FLUORESCENT DYES; HUMANS; MODELS, MOLECULAR; PHOSPHORYLATION; QUINAZOLINES; RECEPTOR, ERBB-2; SPECTROMETRY, FLUORESCENCE;

EID: 84865107223     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.07.034     Document Type: Article

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