Utility of in situ sodium alginate/karaya gum gels to facilitate gastric retention in rodents

International Journal of Pharmaceutics

Volumn 434, Issue 1-2, 2012, Pages 406-412

  Foster, Kimberly A ^a   Morgen, Mike ^b   Murri, Brice ^b   Yates, Ian ^b   Fancher, R Marcus ^a   Ehrmann, Jon ^a   Gudmundsson, Olafur S ^a   Hageman, Michael J ^a  

^a BRISTOL MYERS SQUIBB   (United States)

^b Bend Research Incorporated   (United States)

Author keywords

Alginate; Controlled release; Digital imaging; Formulation; Gastroretention; Hydrogels

Indexed keywords

ALGINIC ACID; BARIUM SULFATE; KARAYA GUM; TRACER;

ANIMAL EXPERIMENT; ARTICLE; AUTOPSY; DIGITAL RADIOGRAPHY; DRUG ABSORPTION; DRUG FORMULATION; DRUG RETENTION; FLOW KINETICS; GEL; NONHUMAN; PRIORITY JOURNAL; RAT; STOMACH; VISCOSITY;

ALGINATES; ANIMALS; BARIUM SULFATE; FEASIBILITY STUDIES; GELS; GLUCURONIC ACID; HEXURONIC ACIDS; KARAYA GUM; RATS; RATS, SPRAGUE-DAWLEY; SUSPENSIONS; TIME FACTORS;

EID: 84864136507     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2012.06.009     Document Type: Article

References (22)

1. I. Ahmed, and J. Ayres Bioavailability of riboflavin from a gastric retention formulation Int. J. Pharm. 330 2007 146 154
2. Q. Ain, S. Sharma, G. Khuller, and S. Garg Alginate-based oral drug delivery system for tuberculosis: pharmacokinetics and therapy effects J. Antimicrob. Chemother. 51 2003 931 938
3. K. Albrecht, M. Greindl, C. Kremser, C. Wolf, P. Debbage, and A. Bernkop-Schnurch Comparative in vivo mucoadhesion studies of thiomer formulations using magnetic resonance imaging and fluorescence detection J. Control. Release 115 2006 78 84
4. M. Burke, S. Staton, A. Vickers, E. Peters, and M. Coffin A novel method to radiolabel gastric retentive formulations for gamma scinigraphy assessment Pharm. Res. 24 2007 695 704
5. P. Choudhury, M. Kar, and C. Chauhan Cellulose acetate microspheres as floating depot systems to increase gastric retention of anti-diabetic drug. Formulation, characterization, and in vitro-in vivo evaluation Drug Dev. Ind. Pharm. 34 2008 349 354
6. S. Davis Formulation strategies for absorption windows Drug Discov. Today 10 2005 249 257
7. A. Hoffman, D. Stepensky, E. Lavy, S. Eyal, E. Klausner, and M. Friedman Pharmacokinetic and pharmacodynamic aspects of gastroretentive dosage forms Int. J. Pharm. 277 2004 141 153
8. S. Jagdale, A. Agavekar, S. Pandya, B. Kuchekar, and A. Chabukswar Formulation and evaluation of gastroretentive drug delivery system of propanolol hydrochloride AAPS PharmSciTech 10 2009 1071 1079
9. H. Katayama, T. Nishimura, S. Ochi, Y. Tsuruta, Y. Yamazaki, K. Shibata, and H. Yoshitomi Sustained release liquid preparation using sodium alginate for eradication of Helicobacter pylori Biol. Pharm. Bull. 22 1999 55 60
10. Y.S. Khotimchenko, V.V. Koralev, O.V. Savchenko, and O.A. Ziganshina Physical-chemical properties, physiological activity, and usage of alginates, the polysaccharides of brown algae Russ. J. Mar. Biol. 27 2001 533 564
11. E. Klausner, E. Lavy, D. Stepensky, M. Friedman, and A. Hoffman Novel gastroretentive dosage forms: evaluation of gastroretentivity and its effect on riboflavin absorption in dogs Pharm. Res. 19 2002 1516 1523
12. W. Kubo, S. Miyazaki, and D. Attwood Oral sustained delivery of paracetamol from in situ gelling gellan and sodium alginate formulations Int. J. Pharm. 258 2003 55 64
13. A. Lalloo, E. McConnell, L. Jin, R. Eikes, C. Seiler, and Y. Wu Decoupling the role of image size and calorie intake on gastric retention of swelling-based gastric retentive formulations: pre-screening in the dog model Int. J. Pharm. 431 2012 90 100
14. S. Miyazaki, W. Kubo, and D. Attwood Oral sustained delivery of theophylline using in situ gelation of sodium alginate J. Control. Release 67 2000 275 280
15. R. Perry, C. Carrig, J. Williams, C. Johnson, and J. Kaneene Anatomic features and radiographic observations of gastric emptying and small intestine motility in rat Lab. Anim. Sci. 43 1993 586 593
16. R. Rastogi, Y. Sultana, M. Aqil, A. Ali, S. Kumar, K. Chuttani, and A.K. Mishra Alginate microspheres of isoniazid for oral sustained drug delivery Int. J. Pharm. 334 2007 71 77
17. S. Saphier, A. Rosner, R. Brandeis, and Y. Karton Gastro intestinal tracking and gastric emptying of solid dosage forms in rats using X-ray imaging Int. J. Pharm. 388 2010 190 195
18. T. Satapathy, P. Panda, A. Goyal, and G. Rath Evaluation of anti-GERD activity of gastro retentitve drug delivery system of itopride hydrochloride Artif. Cells Blood Substit. Immobil. Biotechnol. 38 2010 200 207
19. D. Stepensky, M. Friedman, W. Srour, I. Raz, and A. Hoffman Preclinical evaluation of pharmacokinetic-pharmacodynamic rationale for oral CR metformin formulation J. Control. Release 71 2001 107 115
20. F. Stops, J. Fell, J. Collett, L. Martini, H. Sharma, and A. Smith Citric acid prolongs the gastro-retention of a floating dosage form and increases the bioavailability of riboflavin in the fasted state Int. J. Pharm. 308 2006 14 24
21. G. Tripathi, S. Singh, and G. Nath Evaluation of pH trigger oil entrapped buoyant beads of acetohydroxamic acid for eradication of Helicobacter pylori Int. J. PharmTech Res. 3 2011 1359 1368
22. M. Uddin, P. Rathi, A. Siddiqui, A. Sonawane, and D. Gadade Recent development in floating delivery systems for gastric retention of drugs an overview Asian J. Biomed. Pharm. Sci. 1 2011 26 42