Solid-state thermal behavior and stability studies of theophylline-citric acid cocrystals prepared by neat cogrinding or thermal treatment

Journal of Solid State Chemistry

Volumn 192, Issue , 2012, Pages 238-245

  Hsu, Po Chun ^a   Lin, Hong Liang ^a   Wang, Shun Li ^b   Lin, Shan Yang ^a  

^a YUANPEI UNIVERSITY   (Taiwan)

^b NATIONAL CHIAYI UNIVERSITY   (Taiwan)

Author keywords

Anhydrous citric acid; Anhydrous theophylline; Cocrystal; Cogrinding; Stepwise mechanism; Thermal treatment

Indexed keywords

ANHYDROUS THEOPHYLLINE; CO-CRYSTAL FORMATION; CO-CRYSTALS; CO-GRINDING; FTIR MICROSPECTROSCOPY; PHYSICAL MIXTURES; SOLVENT EVAPORATION METHOD; SPECTRAL PEAK; STABILITY BEHAVIOR; STABILITY STUDY; STORAGE TIME; THERMAL BEHAVIORS;

CURVE FITTING; HEAT TREATMENT; HYDROGEN BONDS; MIXTURES;

CITRIC ACID;

EID: 84864121752     PISSN: 00224596     EISSN: 1095726X     Source Type: Journal    
DOI: 10.1016/j.jssc.2012.04.010     Document Type: Article

References (40)

1. US FDA, The Biopharmaceutics Classification System (BCS) Guidance, 〈http://www.fda.gov/AboutFDA/CentersOffices/CDER/ucm128219.htm〉
2. G.L. Amidon, H. Lennernäs, V.P. Shah, and J.R. Crison Pharm. Res. 12 1995 413
3. J. Emami J. Pharm. Pharmaceut. Sci. 9 2006 169
4. R.S. Uppoor Am. Pharm. Rev. 8 2005 42
5. B.K. Nanjwade, G.K. Derkar, H.M. Bechra, V.K. Nanjwade, and F.V. Manvi J. Nanomed. Nanotechnol. 2 2 2011 2
6. E.H. Kerns J. Pharm. Sci. 90 2001 1838
7. P. Vishweshwar, J.A. McMahon, J.A. Bis, and M.J. Zaworotko J. Pharm. Sci. 95 2006 499
8. N. Schultheiss, and A. Newman Cryst. Growth Des. 9 2009 2950
9. I. Miroshnyk, S. Mirza, and N. Sandler Expert Opin. Drug Deliv. 6 2009 333
10. A.V. Trask Mol Pharmaceutics 4 2007 301
11. B.S. Sekhon Ars. Pharm. 50 2009 99
12. T. Friščić, and W. Jones J. Pharm. Pharmacol. 62 2010 1547
13. N. Blagden, M. de Matas, P.T. Gavan, and P. York Adv. Drug Delivery Rev. 59 2007 617
14. T.K. Wu, S.Y. Lin, H.L. Lin, and Y.T. Huang Bioorg. Med. Chem. Lett. 21 2011 3148
15. C. Medina, D. Daurio, K. Nagapudi, and F. Alvarez-Nunez J. Pharm. Sci. 99 2010 1693
16. A.V. Trask, and W. Jones Top. Curr. Chem. 254 2005 41
17. T. Friščić, and W. Jones Cryst. Growth Des. 9 2009 1621
18. G. Kaupp CrystEngComm 11 2009 388
19. N. Shan, F. Toda, and W. Jones Chem. Commun. 2002 2372
20. S.Y. Lin, W.T. Cheng, and S.L. Wang Int. J. Pharm. 318 2006 86
21. S.L. James, C.J. Adams, C. Bolm, D. Braga, P. Collier, T. Friščić, F. Grepioni, K.D. Harris, G. Hyett, W. Jones, A. Krebs, J. Mack, L. Maini, A.G. Orpen, I.P. Parkin, W.C. Shearouse, J.W. Steed, and D.C. Waddell Chem. Soc. Rev. 41 2012 413
22. V.V. Boldyrev J. Mater. Sci. 39 2004 5117
23. S. Karki, T. Friscić, W. Jones, and W.D. Motherwell Mol. Pharmaceutics 4 2007 347
24. A. Jayasankar, A. Somwangthanaroj, Z.J. Shao, and N. Rodríguez- Hornedo Pharm. Res. 23 2006 2381
25. W.T. Cheng, S.Y. Lin, and S.L. Wang Drug Dev. Ind. Pharm. 34 2008 1368
26. S.Y. Lin, C.H. Hsu, and M.T. Sheu J. Pharm. Biomed. Anal. 53 2010 799
27. C. Demitri, R. Del Sole, F. Scalera, A. Sannino, G. Vasapollo, A. Maffezzoli, L. Ambrosio, and L. Nicolais J. Appl. Polym. Sci. 110 2008 2453
28. J. Lu, and S. Rohani Org. Process Res. Dev. 13 2009 1269
29. E. Lu, N. Rodriguez-Hornedo, and R. Suryanarayanan Cryst EngComm 10 2008 665
30. J.S. Stevens, S.J. Byard, and S.L.M. Schroeder Cryst. Growth Des. 10 2010 1435
31. J.G. Kesavan, and G.E. Peckt Drug Dev. Ind. Pharm. 22 1996 189
32. T. Fujida Chem. Pharm. Bull. 30 1982 3461
33. L.C. Bichara, H.E. Lanús, E.G. Ferrer, M.B. Gramajo, and S.A. Brandán Adv. Phys. Chem. 2011 Article ID 347072
34. L.C. Bichara, H.E. Lanús, E.G. Ferrer, M.B. Gramajo, and S.A. Brandán Inorg. Chem. 28 1989 719
35. A.V. Trask, W.D. Sam Motherwell, and W. Jones Int. J. Pharm. 320 2006 114
36. W.I. Friesen, and K.H. Michaelian Appl. Spectrosc. 45 1991 50
37. US FDA, Guidance for industry, ICH Q1A (R2), Stability testing of new drug substances and products, Rockville, MD, USA. 2003.
38. G.A. Shabir, and S. Arain Am. Pharm. Rev. 7 2004 32
39. K. Huynh-Ba 2008 Springer New York
40. A. Jayasankar, L. Roy, and N. Rodríguez-Hornedo J. Pharm. Sci. 99 2010 3977